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3-ethyl-5-hydroxy-N-{3-[methyl(phenyl)amino]propyl}adamantane-1-carboxamide
5-[4-(2-phenylethyl)piperidine-1-carbonyl]-N-[(2R)-pyrrolidin-2-ylmethyl]pyridin-2-amine
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-4-phenylbenzamide
2-(2-{[(3,4-dimethylphenyl)methyl]amino}-4-(morpholin-4-yl)pyrimidin-5-yl)-2-methylpropanoic acid
N-cyclopropyl-3-[5-(5-methylthiophene-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanamide
N-({3-[4-(2-methoxyethoxy)phenyl]phenyl}methyl)propanamide
(1S,5R)-3-benzyl-N-[(2-methylphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
(2S,4S,5R)-1,2-dimethyl-4-[methyl(pyridin-3-ylmethyl)carbamoyl]-5-(2-methylphenyl)pyrrolidine-2-carboxylic acid
3-(2,3-dihydro-1H-inden-4-yl)-1-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-1-(pyridin-4-ylmethyl)urea
3-methoxy-1-[(2-methoxypyridin-3-yl)methyl]-1,2-dihydropyridin-2-one
N-[(7-{[4-(benzyloxy)-3-methoxyphenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]pyridine-2-carboxamide
N4-[(4,6-dimethylpyridin-2-yl)methyl]-N4-methyl-6-(propan-2-yl)pyrimidine-2,4-diamine
(2S,4S)-4-amino-N-(propan-2-yl)-1-(pyridine-2-carbonyl)pyrrolidine-2-carboxamide
4-{[2-(1H-indol-3-yl)ethyl]amino}-N-(1-methoxypropan-2-yl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
3-fluoro-N,4-dimethyl-N-{2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}benzamide
1-(cyclohex-3-en-1-ylmethyl)-4-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
1-[4-(3-hydroxyphenyl)piperazin-1-yl]-2-(morpholin-2-yl)ethan-1-one
6-[(2S)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-2-[(4-methoxyphenyl)methyl]-1,3-benzoxazole
1-ethyl-N-methyl-N-(1,3-thiazol-4-ylmethyl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperazine
4-[1-benzyl-5-(2,6-dimethoxypyridine-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
N-[5-(2-ethoxyethyl)-1,3,4-thiadiazol-2-yl]-3-phenylpiperidine-1-carboxamide
1-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]-4-[(1-propyl-1H-imidazol-2-yl)methyl]piperazine
N,N-dimethyl-3-[1-(6-methylquinolin-4-yl)piperidin-3-yl]propanamide
1-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-methoxy-2,2-dimethylpropan-1-one
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-{[1-(propan-2-yl)piperidin-4-yl]formamido}acetic acid
dimethyl(1-{3-[3-(1-methyl-1H-imidazole-2-carbonyl)phenyl]phenyl}ethyl)amine
N-[1-(pyridin-3-yl)propyl]pyrimidin-2-amine
4-(4-chlorophenyl)-N-methyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}butanamide
3-{[4-methyl-6-({pyrazolo[1,5-a]pyrimidin-3-ylmethyl}amino)pyrimidin-2-yl]amino}phenol
4-methyl-5-(3-phenylpiperazine-1-carbonyl)pyrimidine
3-{5-[1-(4-methoxyphenyl)cyclopentyl]-1,2,4-oxadiazol-3-yl}pyridazine
3-(1,3-dimethyl-1H-pyrazol-5-yl)-1-[(1-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)methyl]urea
4-(prop-2-en-1-yl)-1-{[4-(pyrrolidin-1-yl)phenyl]methyl}-1,4-diazepan-5-one
(1R,7S)-3-(2-ethylbutyl)-N-methyl-N-(1,2-oxazol-3-ylmethyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-[(3S,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-tert-butyl-1-methyl-1H-pyrazole-5-carboxamide
N-[(1S,2S)-1,3-dihydroxy-1-phenylpropan-2-yl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
[(2S,4R,5R)-5-(2-fluorophenyl)-4-[({[4-methoxy-3-(methoxymethyl)phenyl]methyl}amino)methyl]-1-methylpyrrolidin-2-yl]methanol
3-ethyl-1-[(1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-3-yl)methyl]urea
5-methyl-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)pyrazine-2-carboxamide
N-[(3S,4R)-4-(4-methylphenyl)-1-(6-oxo-1,6-dihydropyrimidine-5-carbonyl)pyrrolidin-3-yl]cyclopropanecarboxamide
N-methyl-2-[2-oxo-3-(trifluoromethyl)-1,2-dihydropyridin-1-yl]-N-(quinolin-2-ylmethyl)acetamide
[(1-cyclopentylpiperidin-4-yl)methyl][(2,4-dimethoxy-3-methylphenyl)methyl](pyridin-3-ylmethyl)amine
(3R,4R)-N-[2-(2-fluorophenyl)ethyl]-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidine-1-carboxamide
4-(2,3-dihydro-1H-inden-2-yl)-3-{2-oxo-2-[4-(pyridin-3-ylmethyl)piperazin-1-yl]ethyl}piperazin-2-one
4-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}thiomorpholine
2-(ethoxymethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-cyclohexyl-1-{1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-azaspiro[2.5]octan-6-yl}ethan-1-one
({4-ethyl-5-[1-(5-methylthiophene-3-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide