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(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(2-chloro-6-fluorophenyl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
(3S,9aR)-8-(2,5-dimethylbenzenesulfonyl)-3-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
7-amino-4-(2-fluoro-4,5-dimethoxyphenyl)-1,2,3,4-tetrahydro-1,8-naphthyridin-2-one
[(3R,4R)-1-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
2-methyl-4-{3-[3-(pyridin-4-yl)azetidine-1-carbonyl]phenyl}but-3-yn-2-ol
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-4-(pyridin-3-yl)pyrimidin-2-amine
8-(6-methylpyridazin-3-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
methyl({[5-(pyrimidin-2-ylsulfanyl)furan-2-yl]methyl})[1-(pyrimidin-4-yl)ethyl]amine
(2S)-1-[2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetyl]pyrrolidine-2-carboxamide
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-2-(1H-pyrrol-1-yl)propanamide
8-(2-methyl-5-propylpyrimidin-4-yl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
(4aS,8aR)-1-(2-aminoethyl)-6-[1-(2-fluorophenyl)cyclopropanecarbonyl]-decahydro-1,6-naphthyridin-2-one
2-(3-hydroxypropyl)-9-(2-{methyl[(4-methylphenyl)methyl]amino}acetyl)-2,9-diazaspiro[5.5]undecan-3-one
(1S,5R)-6-(cyclobutylmethyl)-3-(6-methoxypyrimidin-4-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl 6-({[2-(1H-pyrazol-1-yl)phenyl]methyl}amino)pyridine-3-carboxylate
1-[3-({3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}methyl)phenyl]-1H-pyrazole
N3-methyl-4-oxo-1-(2-phenylethyl)-N5-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
N-[1-(7-{[4-(furan-2-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-2-methylpropanamide
1-(2-{1-[(2-chloro-5-fluorophenyl)methyl]piperidin-2-yl}ethyl)-4-methylpiperazine
5-[1-(1,3-benzothiazole-2-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
N-cyclopropyl-3-(5-{imidazo[1,2-a]pyrimidine-2-carbonyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanamide
phenyl (7S,9aR)-7-[(2S)-butan-2-yl]-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
(4aS,7aR)-1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-methanesulfonyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-[1-(5-methyl-1,3-oxazole-4-carbonyl)pyrrolidin-2-yl]-N-(1-methyl-1H-pyrazol-5-yl)thiophene-2-carboxamide
1-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-(oxan-2-ylmethoxy)ethan-1-one
1-acetyl-N-[2-(5-chloro-2-methyl-1H-indol-3-yl)ethyl]piperidine-3-carboxamide
1-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-3-(1,2-oxazinan-2-yl)propan-1-one
2-amino-2-methyl-1-[2-(3-phenylpropyl)morpholin-4-yl]propan-1-one
1-cyclopentyl-3-({1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}methyl)urea
1-[(6-chloroquinolin-2-yl)methyl]-N-ethyl-N-(pyridin-4-ylmethyl)piperidin-3-amine
N-(2-ethoxyphenyl)-3-[4-(1-methyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]propanamide
(2S,4R)-4-(4-cyanobenzamido)-N-ethyl-1-[3-(methylsulfanyl)propyl]pyrrolidine-2-carboxamide
N-[2-(4-methoxybenzenesulfonamido)ethyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
3-(2-fluorophenyl)-3-{[4-hydroxy-2-(pyridin-4-yl)pyrimidin-5-yl]formamido}propanoic acid
N-[(1R,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-1-methyl-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-hydroxypiperidin-1-yl)methyl]pyrrolidin-1-yl]-2-(phenylsulfanyl)ethan-1-one
1-(3-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}-3-oxopropyl)piperidin-2-one
(3S,4S)-4-propyl-1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}pyrrolidine-3-carboxylic acid
(4aS,8aR)-6-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-1-(3-methylbutyl)-decahydro-1,6-naphthyridin-2-one
1-methyl-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-2-oxo-1,2-dihydropyridine-4-carboxamide
{[2-cyclohexylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[3-(pyrrolidin-1-yl)propyl]amine
N-[3-(1H-imidazol-1-yl)propyl]-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
(3aS,6aR)-3-[3-(morpholin-4-yl)propyl]-5-(1H-pyrrole-2-carbonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-[4-(5-{1-[(2E)-4-methylpent-2-en-1-yl]pyrrolidin-2-yl}thiophene-2-carbonyl)piperazin-1-yl]ethan-1-one
{[2-cyclohexylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)(pyridin-2-ylmethyl)amine
3-(furan-2-yl)-N-[1-(pyrimidin-2-yl)piperidin-3-yl]propanamide
N-(1-{7-[(4-fluoro-3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)pyridine-3-carboxamide
2-cyclopropyl-N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]acetamide
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2-(4-fluorophenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide