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3-({4-[(2-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)-4H-chromen-4-one
1-(azocan-1-yl)-3-(2-{[(2-hydroxyethyl)(methyl)amino]methyl}-5-methoxyphenoxy)propan-2-ol
7-(3-cyclopropyl-1-phenyl-1H-1,2,4-triazol-5-yl)-3,4-dihydro-2H-1,4-benzoxazin-3-one
3-(3-methylpiperidine-1-carbonyl)-N-[2-(pyridin-4-yl)ethyl]benzene-1-sulfonamide
8-(2-phenylpyrimidine-5-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-chloro-N-(1,1-dioxo-1λ6-thian-4-yl)-4-fluoro-N-methyl-1-benzothiophene-2-carboxamide
2-amino-N-(2-methylpropyl)-4-phenyl-N-(pyridin-2-ylmethyl)pyrimidine-5-carboxamide
4-(6-{[1-(pyrrolidin-1-yl)hex-5-en-2-yl]oxy}pyridazin-3-yl)thiomorpholine
3-[(4-fluorophenyl)methyl]-5-methyl-5-[1-(2-methyl-1H-1,3-benzodiazole-6-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
8-[(2-aminopyridin-3-yl)methyl]-2-[(dimethyl-1,2-oxazol-4-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
(4aS,8aR)-6-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2,5-dimethylthiophene-3-sulfonamide
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(3-chlorophenyl)methyl]-4-{[(2,5-dimethylphenyl)methyl]amino}pyrrolidine-2-carboxamide
N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-2-(1H-1,2,4-triazol-1-yl)benzamide
8-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-[9-oxo-8-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecane-2-carbonyl]cyclopropane-1-carboxamide
1-ethyl-8-[(4-phenyl-1,3-thiazol-2-yl)methyl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(3S,4S)-3-hydroxy-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-1-yl]-2-(4-methyl-1H-pyrazol-1-yl)ethan-1-one
7-hydroxy-4-(3-methyl-1H-indol-2-yl)-2-oxo-1,2,3,4-tetrahydroquinoline-6-carboxylic acid
1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}-4-(thiophen-2-ylmethyl)-1,4-diazepane
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-1-[(3,4-dimethoxyphenyl)methyl]-N5-[2-(morpholin-4-yl)ethyl]piperidine-3,5-dicarboxamide
1-{[2-(2,5-dimethoxyphenyl)-8-methylquinolin-3-yl]methyl}piperidin-3-ol
N-[(2-chloro-6-fluorophenyl)methyl]-4-methylpyrimidin-2-amine
2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-1-[1-(propan-2-yl)piperidine-4-carbonyl]piperidine
3-{imidazo[1,2-a]pyridin-2-yl}-5-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1,2,4-oxadiazole
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-3-oxo-3,4-dihydro-2H-1,4-benzoxazine-6-sulfonamide
1-cyclohexyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-1H-1,2,3-triazole-4-carboxamide
4-ethyl-1-methyl-3-(1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
ethyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]{[3-(methylsulfanyl)phenyl]methyl}amine
methyl({[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}){[4-(trifluoromethyl)phenyl]methyl}amine
(1S,6R)-9-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-ethyl-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazole
1-(3-chlorophenyl)-4-(1-phenyl-1H-pyrazole-4-carbonyl)piperazin-2-one
2-{methyl[4-(morpholin-4-yl)butyl]amino}-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
2-hydroxy-2-methyl-N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)propanamide
N'1-{2-[benzyl(methyl)amino]-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl}cyclopropane-1,1-dicarboxamide
4-{2-[3-(pyridin-2-yl)azetidine-1-carbonyl]phenyl}morpholine
N-({4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-3-chlorobenzamide
3-[cyclopropyl(thiophen-3-ylmethyl)amino]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
4-[3-(3-chlorophenyl)pyrrolidine-1-carbonyl]-1-cyclopropanecarbonylpiperidine
1-[1-(1-benzothiophen-2-ylmethyl)piperidin-3-yl]-N-cyclopentyl-1H-1,2,3-triazole-4-carboxamide
2-(3-methyl-1,2-oxazol-5-yl)-N-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]pyrrolidine-1-carboxamide
(2S)-2-[3-cyclopropyl-1-(1-methyl-2-oxo-1,2-dihydroquinolin-4-yl)-1H-1,2,4-triazol-5-yl]pyrrolidine-1-carboxamide
N-(1-methyl-1H-1,2,3-triazol-4-yl)-3-({methyl[1-(pyridin-2-yl)propan-2-yl]amino}methyl)benzamide
6-({[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)-1,4-oxazepan-6-ol
5-[(1S,5R)-6-(cyclobutylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]propanamide
(3R)-1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}pyrrolidin-3-ol
methyl (2S,4R)-4-(dimethylamino)-1-(2-methyl-1-benzofuran-7-carbonyl)pyrrolidine-2-carboxylate
2-[(3-{[4-(pyridin-2-yl)butyl]carbamoyl}phenyl)amino]acetic acid