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5-(oxane-2-carbonyl)-3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2-fluoro-6-hydroxy-N-{[(1r,4r)-4-(methylcarbamoyl)cyclohexyl]methyl}benzamide
4,6-dimethyl-2-{pyrazolo[1,5-a]pyridin-7-yl}pyridine-3-carbonitrile
1-benzyl-3,8-bis(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(3-chloro-4-fluorophenyl)-3-[1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]propanamide
2-{[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl](pyridin-3-ylmethyl)amino}butan-1-ol
2-[2-(2,4-dichlorophenyl)-4-methylphenoxy]acetamide
1-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
4-(4-{[(1S,2S)-2-[(4-fluorophenyl)methyl]cyclopentyl]amino}piperidin-1-yl)-6-methylpyrimidin-2-amine
N-(3,4-dimethylphenyl)-4-[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
2-[8-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carbonyl)-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl]acetic acid
3-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}pyridin-2-amine
3-{[methyl({[3-(1H-pyrazol-1-yl)phenyl]methyl})amino]methyl}pyridin-2-ol
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-ethyl-4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
(1S,4R)-2-[(3-chloro-2-fluorophenyl)methyl]-2-azabicyclo[2.2.1]heptan-3-one
2-(2,6-dimethoxyphenyl)-7-phenyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-(5-phenyl-1,2-oxazole-4-carbonyl)-1,4-oxazepan-6-ol
8-[(2S)-2-aminopentanoyl]-2-[(3,5-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
5-[1-(2H-1,3-benzodioxol-5-yl)-1H-imidazol-2-yl]-2-(pyrrolidin-1-yl)-1,3-thiazole
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-2-(dimethyl-1,3-thiazol-5-yl)acetamide
4-(5-methyl-1H-indazole-3-carbonyl)-7-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-ylmethyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-{[4-(dimethylamino)-1-methylpiperidin-4-yl]methyl}-5-ethylpyrimidin-2-amine
2-methyl-4-{3-[3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]phenyl}but-3-yn-2-ol
1-(cyclohex-3-en-1-ylmethyl)-4-(4-phenyl-1H-pyrazol-5-yl)piperidine
1-(2-ethoxyethyl)-2-oxo-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]pyrrolidine-3-carboxylic acid
N-(prop-2-en-1-yl)-3-propanamido-N-(pyridin-3-ylmethyl)benzamide
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-2,3,6-trimethylquinoline-4-carboxamide
ethyl 4-[5-(2-chloro-4-fluorophenoxymethyl)-1,2-oxazole-3-carbonyl]piperazine-1-carboxylate
2-[4-(2-methyl-1H-imidazol-1-yl)butanoyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
1-(4-{[2-(5-methylfuran-2-yl)ethyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
6-{1-[1-(pyridin-2-yl)piperidine-3-carbonyl]piperidin-4-yl}-3,4-dihydropyrimidin-4-one
(3aS,6aS)-2-cyclobutanecarbonyl-5-[2-(1,3-thiazol-4-yl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
8-(4-hydroxypiperidine-1-carbonyl)-2-methyl-1,4-dihydroquinolin-4-one
4-(2-{7-[2-hydroxy-4-(1H-pyrazol-1-yl)butan-2-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-oxoethyl)-7-methyl-2H-chromen-2-one
4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]-1-(2-phenylethyl)piperidine
2-[8-(1,3-benzothiazol-2-ylmethyl)-1-ethyl-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
1-[1-(5-chloropyridin-2-yl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-3-carboxamide
2-(methoxymethyl)-5-({4-[(4-phenyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}methyl)pyrimidine
1-ethyl-4-{4-[(3-methylphenyl)methyl]piperazine-1-carbonyl}-1,2-dihydropyridin-2-one
2,6-dimethyl-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)pyridine-4-carboxamide
2-(2,4-dimethoxybenzenesulfonyl)-2,7-diazaspiro[4.5]decane
7-[5-(4-methylphenyl)furan-2-carbonyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
2-{1-[(4-fluorophenyl)methyl]-4-{[4-(propan-2-yloxy)phenyl]methyl}piperazin-2-yl}ethan-1-ol
8-[(benzylsulfamoyl)amino]quinoline-2-carboxylic acid
2-{3-methyl-5-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]-1H-1,2,4-triazol-1-yl}pyridine
[(2-ethoxyphenyl)methyl]({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}(methyl)(oxan-4-ylmethyl)amine
2-[2-(2-methoxyphenyl)pyrrolidine-1-carbonyl]-6-methyl-4H-pyran-4-one