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1-(oxane-4-carbonyl)-3-(4-phenoxybenzoyl)piperidine
4-({N-ethyl-1-[3-(3-fluorophenyl)-1H-pyrazol-4-yl]formamido}methyl)benzoic acid
N-[(2,5-dimethylphenyl)(pyridin-3-yl)methyl]-2-ethyl-4-methyl-1,3-oxazole-5-carboxamide
{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]methylamine
2-(5-acetylthiophen-3-yl)-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]ethan-1-one
2-{4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperazin-1-yl}pyridine-3-carboxamide
5-ethanesulfonamido-N,1-dimethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-phenyl-1H-1,3-benzodiazole-7-carboxamide
2-({3-[(oxolan-2-ylmethyl)carbamoyl]phenyl}amino)acetic acid
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-4-(1H-pyrazol-3-yl)benzamide
(3S,4R)-1-[6-(dimethylamino)pyridine-3-carbonyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
3-(2-methoxyethyl)-1-[3-(1H-pyrazol-1-yl)propanoyl]piperidine-3-carboxylic acid
2-(1H-1,3-benzodiazol-1-yl)-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}propanamide
5-[4-(thian-4-yl)piperazine-1-carbonyl]thiophene-2-carboxylic acid
5-methoxy-2-{[2-(morpholin-4-ylmethyl)piperidin-1-yl]methyl}-4H-pyran-4-one
8-(4-methylpyridine-3-carbonyl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-{1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-4-(2-methylphenyl)piperazine
1-[(5-amino-1,3,4-thiadiazol-2-yl)methyl]-3-(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)urea
3-(5-amino-1H-1,2,4-triazol-3-yl)-1-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]propan-1-one
(1R,5S,6R,7S)-3-methyl-4-oxo-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-[(1r,4r)-4-hydroxycyclohexyl]acetamide
4-{[5-(1-cyclopentylpiperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}morpholine
N-[(4-phenyl-1,3-thiazol-5-yl)methyl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
3-[4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]-1,2,5,6,7,8-hexahydroquinolin-2-one
2-ethyl-8-[(4-oxo-1,4-dihydroquinolin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
2-(4-hydroxyphenyl)-1-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
(2S,4S)-4-amino-1-{3-[(3-fluorophenyl)carbamoyl]propanoyl}-N-methylpyrrolidine-2-carboxamide
4-(2-fluorophenoxy)-1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidine-4-carboxylic acid
(3R,4R)-3-methyl-1-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]-4-(oxan-4-yl)piperidin-4-ol
6-(4-fluorophenyl)-N-methyl-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
5-[3-(1H-indol-3-yl)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonitrile
methyl 3-[(2E)-3-phenylprop-2-enamido]-5-{[2-(1H-1,2,4-triazol-1-yl)acetamido]methyl}benzoate
1-(cyclohexylmethyl)-3-hydroxy-3-({methyl[(3-methylpyridin-2-yl)methyl]amino}methyl)piperidin-2-one
(2S)-2-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]piperidine
3-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)-2,3-dihydro-1λ6-thiophene-1,1-dione
(1R,6S)-3-(2-ethylpyrimidine-5-carbonyl)-9-methyl-3,9-diazabicyclo[4.2.1]nonane
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-methoxypropanamide
5-(2-fluorophenyl)-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1,2,4-triazin-3-amine
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-N,2,2,6,6-pentamethylpiperidin-4-amine
N-[(5-amino-1,3,4-thiadiazol-2-yl)(phenyl)methyl]-1-(4-fluorophenyl)cyclopropane-1-carboxamide
8-(4-methylphthalazin-1-yl)-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
2-[4-(3-chloro-4-methylbenzoyl)morpholin-3-yl]-N-(pyridin-3-yl)acetamide
N-(3-hydroxypropyl)-N-[(2-methoxyphenyl)methyl]-2,5-dimethyl-1,3-thiazole-4-carboxamide
N-{[1-(dimethylsulfamoyl)piperidin-3-yl]methyl}-4-phenylbenzamide
7-chloro-N,3,5-trimethyl-N-[4-(morpholin-4-yl)butyl]-1-benzofuran-2-carboxamide
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
methyl 3-[(3S,4R)-1-[(4-oxo-4H-chromen-3-yl)methyl]-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanoate
N-methyl-6-(piperidin-1-yl)-N-[2-(1H-pyrazol-4-yl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
3-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-2-methylphenol
N-(2-{[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]amino}ethyl)acetamide
2-[9-(oxan-2-ylmethyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]acetamide