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1-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}hexan-1-one
14-(2,2-dimethyl-2,3-dihydro-1-benzofuran-7-yl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
N-(cyclohex-1-en-1-ylmethyl)-2-(ethanesulfonyl)propanamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]acetamide
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}-3-(methylsulfanyl)propanamide
5-[1-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-4-yl]-5-[(4-fluorophenyl)methyl]-3-(2-methoxyethyl)imidazolidine-2,4-dione
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]({[2-(2-fluorophenoxy)pyridin-3-yl]methyl})amine
5-[5-(2-benzyl-1,3-thiazol-4-yl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
4-[(3,4-dimethoxypyridin-2-yl)methyl]-3,4-dihydro-2H-1,4-benzoxazin-3-one
4-(3,5-dimethoxyphenyl)-N-methyl-1H-pyrrolo[2,3-b]pyridin-6-amine
1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
4-(4-chlorophenyl)-N-methyl-N-[1-(1,3-thiazol-5-yl)ethyl]butanamide
N-[3-(1H-imidazol-1-yl)propyl]-N-(pyridin-4-ylmethyl)-2,3-dihydro-1H-indene-2-carboxamide
2-methyl-5-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyrimidine
methyl 5-[(2,3-dihydroxypropyl)amino]-1-(2-methoxyethyl)-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(3-hydroxypropyl)-9-[(2,4,5-trimethylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
5,7-dichloro-2-{5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}-1,2,3,4-tetrahydroisoquinoline
N-(furan-2-ylmethyl)-3-{4-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}propanamide
1-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine
2-methyl-5-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}phenol
(2S,4R)-N-[2-(3-chlorophenyl)ethyl]-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
N-[(2,6-difluorophenyl)methyl]-2-(3-methoxyphenoxymethyl)-1,3-oxazole-4-carboxamide
3-[2-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-2-oxoethyl]-1-(2-methoxyethyl)-3-(2-methoxyphenyl)pyrrolidine-2,5-dione
3-propyl-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-5-carboxamide
1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-cyclopropyl-3-({1-[(2,4-difluorophenyl)methyl]piperidin-4-yl}oxy)-4-methoxybenzamide
6-[4-(2-methylpropanamido)phenyl]pyrazine-2-carboxylic acid
N-butyl-2-[methyl(pyridin-3-ylmethyl)amino]-N-[(5-methylthiophen-2-yl)methyl]acetamide
2-amino-7-(2-methoxyquinoline-4-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-{[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]formamido}-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetic acid
(3R,5S)-1-benzyl-N-[3-(morpholin-4-yl)propyl]-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
1-[3-(2-fluorophenyl)pyrrolidin-1-yl]-2-{[3-(pyridin-3-yl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]sulfanyl}ethan-1-one
N-[2-(dimethylamino)ethyl]-6-methyl-N-[(5-methylthiophen-2-yl)methyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
(4aR,7aS)-1-acetyl-4-{pyrazolo[1,5-a]pyridine-3-carbonyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(2-methoxyethyl)(propan-2-yl)amine
4-({4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}methyl)-1,4-oxazepane
N-methyl-N-(1-methylpiperidin-4-yl)-3-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-3-yl)propanamide
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-1,5-dimethyl-1H-pyrazole-3-carboxamide
(5-{[(butan-2-yl)[(2-chlorophenyl)methyl]amino]methyl}furan-2-yl)methanol
(2S,4S)-4-[(4-methylpyrimidin-2-yl)sulfanyl]-1-(naphthalen-2-ylmethyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
7-[3-(1H-imidazol-4-yl)-2-(1H-pyrrol-1-yl)propanoyl]-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
8-(5-propyl-1,3,4-oxadiazole-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(4-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)propan-1-ol
4-(3-phenylbutyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-(2,3-dimethyl-1H-indole-7-carbonyl)-7-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-cyclobutanecarbonyl-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]piperidine
3-(2,3-dimethoxyphenyl)-1-{5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carbonyl}pyrrolidine
N-({1-[(6-ethoxyquinolin-2-yl)methyl]pyrrolidin-3-yl}methyl)acetamide
4-(2-methyl-1,3-benzothiazole-5-carbonyl)piperazin-2-one