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N-(2-{7-[(2-phenyl-1,3-thiazol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-3-carboxamide
1-(2-fluorophenyl)-N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]cyclopropane-1-carboxamide
1-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-4-(4-methoxyphenyl)piperazine
2-(2-{[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
4-{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}thiomorpholine
2-({6-[4-(pyridin-2-yl)piperazin-1-yl]pyridazin-3-yl}oxy)-1-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
2-amino-6-[1-(2-fluorophenyl)-1H-pyrazol-4-yl]-4-(oxolan-3-yl)pyridine-3-carbonitrile
5-(4-fluorophenyl)-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
N,N-diethyl-1-[(1s,4s)-4-(2,3,4-trimethoxybenzamido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
(2S)-2-amino-N-(propan-2-yl)-3-(1,3-thiazol-4-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]propanamide
3-acetamido-N-(2-methoxyphenyl)-5-({[(5-methylfuran-2-yl)methyl]amino}methyl)benzamide
N-[4-({[(2-methylphenyl)methyl]carbamoyl}methyl)phenyl]butanamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-1-(2-methylpropyl)piperidin-4-amine
4-{4-[2-(dimethylamino)-2-(4-methylphenyl)acetyl]piperazin-1-yl}benzonitrile
4-(2,8-dimethylquinoline-4-carbonyl)-1λ6-thiomorpholine-1,1-dione
1-[1-(cyclopropylmethyl)piperidin-3-yl]-4-(4-methoxyphenyl)piperazine
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
(2S)-4-methyl-1-(4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzoyl)-2-(propan-2-yl)piperazine
4-[(3-fluorophenyl)methyl]-11-{[2-(2-methoxyphenyl)ethyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
7-(2-methoxyethyl)-2-(4-methoxypyrimidin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
2-cyclopropyl-9-(2,2-dimethyloxane-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(1H-indol-3-ylmethyl)-6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-methyl-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
5-(1H-imidazol-1-ylmethyl)-N-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]furan-2-carboxamide
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-N-[(1S,2R)-1-hydroxy-1-(4-hydroxyphenyl)propan-2-yl]propanamide
1-(3-chloro-4-methoxybenzoyl)-3-(1H-imidazol-1-ylmethyl)piperidine
N-[(3R,5S)-1-butyl-5-(methylcarbamoyl)pyrrolidin-3-yl]-3-(thiophen-3-yl)-1H-pyrazole-5-carboxamide
2-methyl-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]quinoline
3-methyl-3-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1-[2-methyl-5-(4H-1,2,4-triazol-4-yl)phenyl]urea
(1s,4s)-4-{4-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}cyclohexan-1-amine
4-(4-methoxy-2-methylphenyl)-1-(oxan-2-ylmethyl)-1H-1,2,3-triazole
2-(pyrrolidin-1-yl)-1-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
2-(morpholin-4-yl)-1-(4-{1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)ethan-1-ol
N-[(3R,4S)-4-cyclopropyl-1-[3-(methylsulfanyl)propyl]pyrrolidin-3-yl]-4-(hydroxymethyl)benzamide
1-ethyl-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-N-[2-(pyridin-2-yl)ethyl]piperidin-4-amine
(3S,4R)-1-(2-ethylpyridine-4-carbonyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
1-(2-methyl-1,3-benzothiazol-5-yl)-3-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}urea
[(3R,4R)-4-[(dimethylamino)methyl]-1-[4-(hydroxymethyl)benzoyl]pyrrolidin-3-yl]methanol
(2E)-1-{3-[benzyl(methyl)amino]piperidin-1-yl}-3-(furan-2-yl)prop-2-en-1-one
1-ethyl-4-{[methyl({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)amino]methyl}pyrrolidin-2-one
8-[(2E)-2-methylbut-2-en-1-yl]-3-{2-[4-(propan-2-yl)piperazin-1-yl]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-cyclohexyl-N-(oxan-4-yl)-1H-pyrazole-4-carboxamide
7-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-methyl-N-(pyrazin-2-ylmethyl)benzamide
1-(azocan-1-yl)-3-{2-methoxy-4-[({[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}amino)methyl]phenoxy}propan-2-ol
1-[(4-chlorophenyl)methyl]-4-[2-(4-methyl-1,4-diazepane-1-carbonyl)-1-benzofuran-5-yl]piperidin-4-ol
(3aS,6aS)-2-propyl-5-[2-(1H-1,2,4-triazol-3-yl)benzoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
ethyl 4-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperazine-1-carboxylate
N-[2-(2-ethoxyphenyl)ethyl]-5-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine