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(1-{[3-(2-aminoethyl)phenyl]methyl}-3-(cyclopropylmethyl)piperidin-3-yl)methanol
3-hydroxy-S-[2-(1H-pyrazole-3-carbonyl)-1,2,3,4-tetrahydroisoquinolin-6-yl]butane-1-sulfonamido
N1,N1-dimethyl-N4-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}piperidine-1,4-dicarboxamide
2-oxo-N-[1-(thian-4-yl)piperidin-4-yl]-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
(2S)-2-{[6-(4-fluorophenyl)-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazin-2-yl]formamido}propanamide
methyl 2-[3-oxo-1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)piperazin-2-yl]acetate
1-(2-fluoro-4-methylbenzoyl)-4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine
3-[({[1-(hydroxymethyl)cyclobutyl]methyl}(methyl)carbamoyl)methyl]-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-{2-[1-(3-cyanobenzenesulfonyl)piperidin-2-yl]ethyl}acetamide
N-cyclopentyl-4-[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
1-benzyl-5-methanesulfonamido-N,2-dimethyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1H-1,3-benzodiazole-7-carboxamide
1-[(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-cyclopropylpropan-1-one
7-(2-phenylbenzoyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-[1-(azepane-1-sulfonyl)piperidin-3-yl]benzoic acid
2,6-dimethyl-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}quinoline-4-carboxamide
1-[(1-phenyl-1H-pyrazol-4-yl)methyl]-4-[2-(piperidine-1-carbonyl)phenoxy]piperidine
5-[2-(methylsulfanyl)phenoxymethyl]-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
5-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-N-methyl-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-3,4,7-trimethyl-1H-indole-2-carboxamide
N-cycloheptyl-3-[(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)amino]propanamide
(1-{1-[(2,6-difluoro-3-methoxyphenyl)methyl]piperidin-4-yl}piperidin-3-yl)methanol
{[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(methyl)[(5-methylfuran-2-yl)methyl]amine
1-{2-[(2,5-dimethyl-1-phenyl-1H-pyrrol-3-yl)formamido]ethyl}piperidine-3-carboxamide
(3-{2-[1-(3,5-difluoropyridine-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
3-methoxy-N-(1-{7-[(2-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
4-(2-phenylphenyl)pyridin-2-amine
N1-(pyridin-3-yl)-N2-{8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-yl}ethane-1,2-diamine
4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}-N-[2-(pyridin-3-yloxy)propyl]benzamide
{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}(methyl)(pyridin-2-ylmethyl)amine
2-(2,3-dihydro-1H-inden-1-yl)-N-[1-(thian-4-yl)piperidin-4-yl]acetamide
(2S)-2-amino-N-butyl-4-(methylsulfanyl)-N-[(3-methylthiophen-2-yl)methyl]butanamide
5-methyl-N-({5-[3-(trifluoromethoxy)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-1,2-oxazole-3-carboxamide
(2R,6R)-10-methoxy-4-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-methyl-2-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine
N-[3-(pyridin-3-yloxy)propyl]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-[(5,8-dimethoxy-4-methylquinolin-2-yl)(methyl)amino]ethan-1-ol
N4-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]pyrimidine-4,6-diamine
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]-decahydro-1,6-naphthyridin-2-one
N-[(3S,5S)-1-cyclopentyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]-1-methyl-1H-pyrazole-5-carboxamide
5-[(2-chlorophenyl)methyl]-3-(2-methoxyethyl)-5-[1-(4-methyl-2-oxopentanoyl)piperidin-4-yl]imidazolidine-2,4-dione
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-3-ethyl-1,2-oxazole-5-carboxamide
N-(3-cyclohexyl-1H-1,2,4-triazol-5-yl)-2-(2-methoxyphenyl)pyrrolidine-1-carboxamide
4-{[(4aS,7aR)-4-ethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
1-[(4aR,8aR)-1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-decahydro-1,6-naphthyridin-6-yl]-3-phenylpropan-1-one
{2-[4-(2-methoxyphenoxy)piperidin-1-yl]quinolin-3-yl}methanol
2-(2,5-dioxoimidazolidin-1-yl)-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}acetamide
N-[(4-fluorophenyl)methyl]-N-(3-methoxypropyl)-5,6-dimethylpyridine-3-carboxamide
4-methyl-5-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,3-thiazol-2-amine
8-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(3R,4S)-1-[2-oxo-2-(piperidin-1-yl)ethyl]-4-propylpyrrolidin-3-yl]methanesulfonamide