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N-[1-(pyrazin-2-yl)propan-2-yl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
ethyl 1-(3,5-dimethylfuran-2-carbonyl)-4-[(4-methoxyphenyl)methyl]piperidine-4-carboxylate
2-{4-[(6-fluoro-4-hydroxyquinolin-2-yl)methyl]piperazin-1-yl}-N-(propan-2-yl)acetamide
methyl 9-(cyclopentyloxy)-7-oxo-3-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[(3R,4S)-1-acetyl-4-(propan-2-yl)pyrrolidin-3-yl]-1-(3-chlorophenyl)methanesulfonamide
2-({[(1-cyclopropanecarbonylpiperidin-4-yl)methyl]amino}methyl)-6-methylquinolin-4-ol
2-(5-chloro-6-methyl-1-benzofuran-3-yl)-1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}ethan-1-one
N-(2-ethyl-3-methyl-1-benzofuran-7-yl)-4-(pyrimidin-2-yl)-1,4-diazepane-1-carboxamide
1-{[4-(benzyloxy)phenyl]methyl}-3-(4H-1,2,4-triazol-3-yl)piperidine
(3aS,6aS)-2-(3-cyanopyridin-2-yl)-5-cyclopentyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[2-(1-tert-butyl-3-methyl-1H-1,2,4-triazol-5-yl)ethyl]-5-methyl-1H-1,2,3,4-tetrazole
N-(1-{7-[(8-methoxyquinolin-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)propanamide
N-({2,3-dimethylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
methyl({[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl})[1-(thiophen-2-yl)ethyl]amine
3-{[2-(hydroxymethyl)-2,5-dihydro-1H-pyrrol-1-yl]methyl}-N,8-dimethyl-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
8-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(quinolin-2-ylmethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetamide
(3S,4S)-4-(dimethylamino)-1-{[3-(2-methylphenyl)phenyl]methyl}pyrrolidin-3-ol
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-2-(2-oxoazepan-1-yl)acetamide
1-[3-(2H-1,3-benzodioxol-5-yl)-1-methyl-1H-1,2,4-triazol-5-yl]piperidine
3-cyclopropyl-5-[2-(2-methyl-1H-imidazol-1-yl)propyl]-1-propyl-1H-1,2,4-triazole
N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,2-dimethylpropanamide
2-{[3-(2-hydroxyethyl)-4-methylpiperazin-1-yl]methyl}-3,5-dimethoxybenzoic acid
N-[(2-{4-[5-(methoxymethyl)furan-2-amido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-3-methyl-5,6-dihydro-1,4-dioxine-2-carboxamide
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
6-fluoro-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
7-(1,3-benzothiazol-2-yl)-9-hydroxy-N,N-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxamide
5-{[3-(4-methyl-1,3-thiazol-5-yl)propanamido]methyl}thiophene-2-carboxylic acid
1-[(2-chloro-6-fluorophenyl)methyl]-N-methylpyrrolidine-3-carboxamide
N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
5-(2,2-diethylmorpholine-4-carbonyl)-1-[(2-fluorophenyl)methyl]piperidin-2-one
2-[3-(3-methoxypropyl)piperidine-1-carbonyl]benzonitrile
N-ethyl-5-(propan-2-yl)-N-(pyridin-4-ylmethyl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
1-[5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-2-carbonyl]-3-(1H-pyrazol-5-yl)piperidine
8-{1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(3-chloro-1,2-oxazol-5-yl)-1-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]propan-1-one
3-cyclopropyl-1-[2-methoxy-4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-[(5-methylthiophen-2-yl)methyl]urea
5-{2-[3-(1H-imidazol-1-yl)propoxy]-3-methoxyphenyl}-4-phenyl-1H-imidazole
2-(3-fluorophenyl)-1-[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]ethan-1-one
N-methyl-N-{[5-({methyl[(3-methyl-1H-indol-2-yl)methyl]amino}methyl)furan-2-yl]methyl}methanesulfonamide
({2,4-dimethyl-5-[(4-methylpiperazin-1-yl)methyl]phenyl}methyl)(methyl)(pyridin-3-ylmethyl)amine
1-[(3-methylpyridin-2-yl)methyl]-4-[(2,3,4-trimethoxyphenyl)methyl]piperazine
2-methoxy-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
(3aS,6aS)-2-(dimethylsulfamoyl)-5-(furan-2-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[(2-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxylic acid
2-[1-(4-methylphenyl)pyrrolidin-3-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[(2-fluorophenyl)methyl]-1-methyl-5-[(pyridin-3-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(3R,4R)-4-(hydroxymethyl)-1-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}piperidin-3-ol
2-[3-benzyl-1-(4-methoxyphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(2-hydroxyethyl)-N-methylacetamide