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1-methyl-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)-1H-pyrazole-4-carboxamide
N-[1-(pyrazin-2-yl)piperidin-4-yl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
5-(azepane-1-carbonyl)-1-(butan-2-yl)-N-[2-(3-fluorophenyl)ethyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
N-(2-{7-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclohexanecarboxamide
N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-oxo-S-(thiophen-2-yl)ethane-1-sulfonamido
2-{3-[3-(isoquinolin-4-yl)phenyl]-1H-pyrazol-1-yl}ethan-1-ol
1-ethyl-N-methyl-3-(2-methylpropyl)-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1H-pyrazole-5-carboxamide
{2-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-1,3-thiazol-4-yl}methanol
5-{[2-(oxolan-3-yl)-1H-imidazol-1-yl]methyl}-1-phenyl-1H-1,2,3,4-tetrazole
4-(4-chlorophenyl)-N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)butanamide
2-[N-(1-methylpiperidin-4-yl)-1-(3,4,7-trimethyl-1H-indol-2-yl)formamido]acetic acid
N-[2-(2-methoxyphenyl)ethyl]-2-{[4-(propan-2-yl)piperazin-1-yl]methyl}quinazolin-4-amine
5-(oxolan-2-yl)-N-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)thiophene-2-carboxamide
6-[8-(3-methoxypropyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-3-carbonitrile
4-[4-(2-chlorophenyl)piperidin-4-yl]-2-(3-methylbutyl)pyrimidine
3-{ethyl[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}propane-1,2-diol
1-(3-chlorophenyl)-4-(1-cyclobutylpiperidin-3-yl)piperazine
N,8-dimethyl-3-[(4-methylpiperidin-1-yl)methyl]-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
4-[2-(1-{[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl}piperidin-2-yl)ethyl]morpholine
N-[3-(cyclohexyloxy)-2-hydroxypropyl]-1-(furan-2-ylmethyl)piperidine-4-carboxamide
4-(5-acetylthiophene-2-carbonyl)-5-methyl-1-(2-methylphenyl)piperazin-2-one
2-[6-(2,2-dimethylpropanamido)pyridin-3-yl]-2-{[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl](methyl)amino}acetic acid
5-[(3,4-dimethoxyphenyl)methyl]-5-(3-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}-3-oxopropyl)pyrrolidin-2-one
6-[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]pyridine-2-carbonitrile
(3aS,6aS)-2-methyl-5-({2-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[4-({4-[(2S)-4-methyl-2-phenylpiperazine-1-carbonyl]-1,3-oxazol-2-yl}methyl)piperazin-1-yl]pyrimidine
2-{1-cyclopentyl-4-[(2,3,4-trimethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-(2,3-dihydroxypropyl)-5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carboxamide
1-[8-chloro-2-(furan-2-yl)quinoline-4-carbonyl]pyrrolidin-3-ol
6-oxo-1-(3-phenylpropyl)-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}piperidine-3-carboxamide
6-(8-methoxy-2-methylquinolin-5-yl)pyrazine-2-carboxylic acid
4-({2-[1-(2-chloro-4-fluorobenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]amine
1-(4-methylpyridine-3-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
N-[4-(methylsulfanyl)phenyl]-2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carboxamide
8-[(3-hydroxy-4-methoxyphenyl)methyl]-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
{5-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}methanol
ethyl 2-{1-[2-(4-fluorophenoxy)acetyl]piperidin-2-yl}acetate
4-(2H-1,3-benzodioxol-5-yloxy)-1-(pyrimidin-2-yl)piperidine-4-carboxylic acid
N-tert-butyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
3-{[(1H-imidazol-2-ylmethyl)(methyl)amino]methyl}-N-{2-methyl-2H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}benzamide
2-methyl-6-[1-(5-propyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]pyrimidin-4-ol
3-{5-[3-(2-oxoazepan-1-yl)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
methyl 4-{[2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]methyl}-1H-pyrazole-3-carboxylate
2-(4-tert-butylphenoxymethyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(3R,5S)-N-[2-(1,3-benzothiazol-2-yl)ethyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
1-[3-(2-methoxybenzoyl)piperidin-1-yl]-4-(thiophen-2-yl)butan-1-one
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-3-(1H-pyrazol-4-yl)benzamide
3-fluoro-N-({7-[(2E)-4-methylpent-2-enoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzamide