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1-(3-methylbut-2-en-1-yl)-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol
1-(2-methoxybenzoyl)-4-[3-(2-phenylethyl)-4,5-dihydro-1,2-oxazole-5-carbonyl]piperazine
1-methyl-4-phenyl-5-[2-(prop-2-yn-1-yloxy)phenyl]-1H-imidazole
3-(3,4-difluorophenyl)-5-methanesulfonyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
8-[(2R)-2-hydroxy-2-(naphthalen-2-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
(3S,4R)-1-(3-fluoropyridine-4-carbonyl)-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-3-(2-methylphenyl)propan-1-one
1-(2-methoxyphenyl)-4-{1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}piperazine
1-(4-{[(3-cyclopentylpropyl)amino]methyl}-2-methoxyphenoxy)-3-(4-ethylpiperazin-1-yl)propan-2-ol
1-(carbamoylmethyl)-N-(2-methanesulfonamidoethyl)piperidine-3-carboxamide
1-methyl-N-[3-(morpholin-4-yl)propyl]-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-{3-[(4-hydroxy-4-methylazepan-1-yl)methyl]phenoxy}acetamide
8-(3-chloropyridin-2-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-{1-azabicyclo[3.2.1]octan-5-yloxy}pyridine-3-carboxamide
N-[(3R,4R)-1-(2-amino-9H-purin-6-yl)-3-hydroxypiperidin-4-yl]pyrazine-2-carboxamide
1-{2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]morpholin-4-yl}-3-methyl-3-phenylbutan-1-one
N-{1-[(8-methoxy-2H-chromen-3-yl)methyl]piperidin-4-yl}methanesulfonamide
N-[(3S,5S)-1-methyl-5-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)pyrrolidin-3-yl]furan-2-carboxamide
N-[(2-chlorophenyl)methyl]-2-oxo-6-(thiomorpholin-4-ylmethyl)-1,2-dihydropyridine-3-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-1-{4-[(pyridin-2-yl)amino]piperidin-1-yl}ethan-1-one
1-cyclopropanecarbonyl-N-{2-[(pyridin-3-yl)amino]ethyl}piperidine-4-carboxamide
1-[1-(2-methoxyethyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
4-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-2-methoxypyridine-3-carbonitrile
2-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-2,8-diazaspiro[4.5]decane
(5S,9aS,9bS)-5-(5-methylfuran-2-yl)-2-[(2-methylphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-(pyridin-3-ylmethyl)-8-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
2-(4-chloro-2-methylphenoxy)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]acetamide
N-propyl-3-(pyridin-3-yl)-N-(pyridin-3-ylmethyl)propanamide
1-(2-methyloxolane-2-carbonyl)-4-phenoxypiperidine-4-carboxylic acid
2-{4-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-1-(thiophen-3-ylmethyl)piperazin-2-yl}ethan-1-ol
methyl (2S)-2-{[1-(3-ethanesulfonamidophenyl)piperidin-4-yl]amino}-2-phenylacetate
8-ethyl-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
N-methyl-2-propyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,3-thiazole-4-carboxamide
3-[(3R,4S)-1-(furan-2-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N-[4-fluoro-3-({[1-(pyrimidin-2-yl)piperidin-3-yl]carbamoyl}amino)phenyl]propanamide
3-{[3-(2,4-dimethylphenoxy)-2-hydroxypropyl]amino}butan-1-ol
1-(carbamoylmethyl)-N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]piperidine-4-carboxamide
4-[6-oxo-1-(2-phenylethyl)piperidine-3-carbonyl]-1,4-diazepane-1-carbaldehyde
6-[(diethylamino)methyl]-N-methyl-N-[1-(pyridin-4-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
4-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-5-ethyl-2-methylpyrimidine
2-{[(3-ethoxyphenyl)methyl](isoquinolin-5-ylmethyl)amino}ethan-1-ol
methyl 6-[4-(2H-1,3-benzodioxol-5-ylmethyl)-3-oxopiperazin-1-yl]pyridine-3-carboxylate
methyl 2-[2-(1-methylpiperidin-2-yl)ethyl]-1-oxo-1,2-dihydroisoquinoline-7-carboxylate
3-[5-(ethanesulfonyl)thiophen-2-yl]-1H-pyrazole
2-methyl-N-[1-(1-{spiro[2.3]hexane-1-carbonyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-3-(pyridin-3-yl)propanamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)pyridine-4-carboxamide
{1-[2-(2,6-dimethoxyphenoxy)ethyl]-3-ethylpiperidin-3-yl}methanol
2-(3-methylbutyl)-8-(4-methylpyridine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
2-{1-[2-(3-fluoro-2,4-dimethylphenyl)-1H-imidazol-1-yl]ethyl}-1,3-thiazole