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3-(1-cyclopentanecarbonylpiperidin-3-yl)-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
1-{2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxybenzoyl}-N,N-diethylpyrrolidin-3-amine
N-[2-(pyrrolidin-1-yl)ethyl]-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
2-{[3-cyclopropyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1H-1,3-benzodiazole
2-[3-(cycloheptylcarbamoyl)propanamido]-2-(3-methylphenyl)acetic acid
4-[(3R,4S)-3-amino-4-propylpyrrolidine-1-carbonyl]-1,2-dihydroisoquinolin-1-one
N-(prop-2-en-1-yl)-N-(pyridin-3-ylmethyl)-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
N-(1,4-dioxan-2-ylmethyl)-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
(8R,9aS)-8-hydroxy-2-{[2-(1H-imidazol-1-yl)phenyl]methyl}-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
(4aS,7aR)-1-(1H-imidazol-4-ylmethyl)-4-(3-methylbutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1R,6S)-9-methyl-3-[3-(piperidin-4-ylmethyl)benzoyl]-3,9-diazabicyclo[4.2.1]nonane
5-methoxy-2-[2-(pyridin-3-yl)piperidine-1-carbonyl]-1,4-dihydropyridin-4-one
1-(2-{4-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperazin-1-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
methyl 1-benzyl-3-(oxolane-2-amido)-5-[(propan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-{1-[1-(2-fluorophenyl)cyclopropanecarbonyl]piperidin-3-yl}benzoic acid
[1-(4-{1-[2-(1H-imidazol-1-yl)ethyl]-1H-imidazol-2-yl}phenyl)ethyl]dimethylamine
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-5-(1,5-dimethyl-1H-pyrazol-4-yl)-1,2-oxazole-3-carboxamide
N3-tert-butyl-1-(3-methylbutyl)-4-oxo-N5-[2-(pyridin-4-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
3-{1,2-dihydrospiro[indole-3,4'-piperidine]-1'-ylmethyl}piperidin-3-ol
1-tert-butyl-3-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1H-pyrrole
4-ethyl-3-{1-[4-(2-methylpropyl)benzoyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
(2S,4R)-4-amino-N,N-diethyl-1-{3-methyl-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carbonyl}pyrrolidine-2-carboxamide
(3S,4S)-1-[(5-fluoro-1-methyl-1H-indol-2-yl)methyl]-4-methylpiperidine-3,4-diol
N-[3-(dimethylamino)-2,2-dimethylpropyl]-2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
7-(2,2-dimethyloxane-4-carbonyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
N5-(2-methoxyethyl)-N6-(1-phenylpiperidin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
1-[4-(4-propyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-2-(2,2,6,6-tetramethylpiperidin-4-yl)ethan-1-one
2-[4-(2-amino-9H-purin-6-yl)-1-[(4-fluorophenyl)methyl]piperazin-2-yl]ethan-1-ol
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(2-methoxyethyl)[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]amine
(1R,5R)-6-(2-aminopyridine-4-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
7-chloro-N,3,5-trimethyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-1-benzofuran-2-carboxamide
N-[(2-chloro-6-fluorophenyl)methyl]-1-[2-(dimethylamino)ethyl]-5-oxopyrrolidine-3-carboxamide
1-(cyclohexylmethyl)-5-(cyclopentylamino)-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-tert-butyl-2-{[(1S,4S)-3,3-dimethyl-2-methylidenebicyclo[2.2.1]heptan-1-yl]formamido}acetamide
1-(2-methylpyridin-4-yl)-4-{2-methylthieno[2,3-d]pyrimidin-4-yl}-1,4-diazepane
2-(3,5-dimethoxyphenyl)-1-[(3S,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]ethan-1-one
1-[3-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-(pyrimidin-2-ylsulfanyl)ethan-1-one
N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]pyrrolidine-1-sulfonamide
N-[(3R,4S)-4-cyclopropyl-1-(3-hydroxypropyl)pyrrolidin-3-yl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
N-({5-fluoro-7-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-3-(3-methyl-1H-pyrazol-1-yl)propanamide
N-[2-(3-chlorophenyl)ethyl]-1-propyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1,3,5-trimethyl-N-(1-phenylcyclopropyl)-1H-pyrazole-4-carboxamide
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-(3-methoxy-4-methylbenzoyl)pyrrolidin-3-yl]methanol
3-[2-(1H-indol-7-yl)ethyl]-1λ6-thiolane-1,1-dione
3-{[1-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
6-[9-methoxy-7-(quinolin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pyrimidin-4-amine
N-butyl-2-(pyridin-3-yloxy)-N-(thiophen-3-ylmethyl)acetamide
methyl (2S,4R)-4-hydroxy-1-(2-methyl-1-benzofuran-5-carbonyl)pyrrolidine-2-carboxylate
N2-(4-methylphenyl)-6-(1H-pyrazol-4-yl)-1,3,5-triazine-2,4-diamine
N-[2-(dimethylamino)-2-(2-methylphenyl)ethyl]-5-methylpyrazolo[1,5-a]pyrimidin-7-amine