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N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-3-fluoro-2-methoxybenzamide
1-(2-phenylethyl)-5-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}piperidin-2-one
N-{1-[(3,4-difluorophenyl)methyl]piperidin-4-yl}-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
3-(1,3-benzothiazol-2-yl)-N-[1-(pyrimidin-2-yl)piperidin-3-yl]propanamide
5-(2-chloro-4-methoxyphenoxymethyl)-N-(1-hydroxybutan-2-yl)-1H-pyrazole-3-carboxamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-methyl-1,5-diazatricyclo[5.2.2.02,6]undecane
1-butyl-4-[2-(2-chlorophenyl)-2-hydroxyacetyl]piperazin-2-one
6-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carbonyl]-1,2,3,4-tetrahydroquinoxaline-2,3-dione
3-(1H-indol-3-yl)-N-[(4-oxo-3,4-dihydrophthalazin-1-yl)methyl]propanamide
N-(4-chloro-3-methoxyphenyl)-2-{[1-(1H-pyrazol-1-yl)propan-2-yl]amino}acetamide
6-[(3-methoxyphenyl)methoxy]-1-(2-phenylethyl)-4-(quinoxaline-5-carbonyl)-1,4-diazepan-2-one
4-(2-{1-[2-(3-fluorophenyl)ethyl]piperidin-2-yl}ethyl)morpholine
4-{[4-(1-propyl-1H-imidazol-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}quinoline
1-methyl-4-phenyl-3-[1-(thiophen-2-ylmethyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[3-(azepan-1-yl)-2-hydroxypropyl]-2-(1H-pyrazol-1-yl)benzamide
1-[2-(1-tert-butyl-3-cyclopentyl-1H-1,2,4-triazol-5-yl)ethyl]-6-methyl-1,2-dihydropyridin-2-one
2-{1-[6-(2-methylphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperidin-2-yl}ethan-1-ol
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]acetamide
1-methyl-5-{4-[2-oxo-2-(pyrrolidin-1-yl)ethyl]piperazine-1-carbonyl}-1,2-dihydropyridin-2-one
1-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one
5-[(methylsulfanyl)methyl]-N-[2-(pyridin-3-yl)ethyl]furan-2-carboxamide
(2S,4R)-4-(cycloheptylamino)-1-(2,2-diphenylethyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
5-cyclobutanecarbonyl-1'-[(1-methyl-1H-imidazol-2-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-{2-[1-(2-methyl-1-benzofuran-7-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
N-[2-(dimethylsulfamoyl)ethyl]-3-(3-methylphenyl)-1H-pyrazole-4-carboxamide
N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-2-(methylamino)-1,3-thiazole-4-carboxamide
(3R,4R)-3-methyl-1-[1-(3-methylphenyl)piperidin-4-yl]-4-(oxan-4-yl)piperidin-4-ol
N-[2-(dimethylamino)ethyl]-N-[(5-methylthiophen-2-yl)methyl]morpholine-2-carboxamide
N-(2-methylphenyl)-1-(2-{[(3,4,5-trimethoxyphenyl)methyl]amino}ethyl)-1H-1,2,3-triazole-4-carboxamide
8-(5-amino-1H-pyrazole-3-carbonyl)-2-cyclopentyl-2,8-diazaspiro[5.5]undecan-3-one
[(5-phenyl-1H-pyrazol-3-yl)methyl]({[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl})amine
3-(4-methoxyphenyl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-3-phenylpropanamide
1-(2-{1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}-2-oxoethyl)imidazolidine-2,4-dione
5-chloro-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-2,3-dihydro-1H-indole-2-carboxamide
1-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-ol
[1-(4-{[(3-methoxyphenyl)methyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carbonyl)piperidin-3-yl]methanol
5-{1-[3-(carbamoylmethoxy)phenyl]-1H-imidazol-2-yl}thiophene-2-carboxylic acid
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-3,5-dimethoxybenzamide
{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}(pyridin-3-ylmethyl)amine
N-butyl-4-(1H-pyrazol-3-yl)-N-(pyridin-3-ylmethyl)benzamide
N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N,2-dimethyl-1,3-benzothiazole-5-carboxamide
N-methyl-4-oxo-4-phenyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}butanamide
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N,2,4-trimethyl-1,3-thiazole-5-carboxamide
N-(1-methyl-1H-pyrazol-4-yl)-2-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)acetamide
3-({[(6-chloropyridin-3-yl)methyl](methyl)amino}methyl)-N-(1,3-thiazol-2-yl)benzamide
(3S,4R)-1-{imidazo[1,2-a]pyrimidine-2-carbonyl}-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
7-[(3-ethoxy-4-methoxyphenyl)methyl]-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
1-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-hydroxyethan-1-one
8-methoxy-2-methyl-5-[5-(morpholine-4-carbonyl)pyridin-2-yl]quinoline