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1-{[5-(1-benzofuran-2-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-3,3-dimethylurea
2-(2-methoxyphenyl)-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]acetamide
2-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-1-(4-methylpiperazin-1-yl)ethan-1-one
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-[2-(pyridin-2-yl)ethyl]benzamide
3-[3-(3-methoxyphenoxymethyl)piperidine-1-carbonyl]benzonitrile
2-[(cyclopropylmethyl)sulfanyl]-1-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
5-[4-(3-hydroxy-3-methylbutyl)benzoyl]-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
1-ethyl-N-methyl-3-(propan-2-yl)-N-{[4-(trifluoromethyl)phenyl]methyl}-1H-pyrazole-5-carboxamide
1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
1-tert-butyl-4-{[methyl({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amino]methyl}pyrrolidin-2-one
2-ethyl-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,4-dimethyl-1,3-oxazole-5-carboxamide
N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
6-chloro-2-(2-oxo-2-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}ethyl)-2,3-dihydropyridazin-3-one
4-[(4-fluorophenyl)methyl]-N,N-dimethyl-5-oxo-3-(propan-2-yl)-1,4-diazepane-1-sulfonamide
2-amino-4-(4-hydroxyphenyl)-6-[1-(2-methylphenyl)-1H-pyrazol-4-yl]pyridine-3-carbonitrile
2-methyl-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-[1-(2-chloro-6-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
5-{[7-acetyl-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}-1-methylpiperidin-2-one
N-({7-[(3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-phenoxyacetamide
N,6-dimethyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}pyridine-2-carboxamide
1-(3-{[methyl(pyrimidin-4-ylmethyl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-{ethyl[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]carbamoyl}benzoic acid
1-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-3-{2-methyl-[1,2,4]triazolo[1,5-a]pyridin-8-yl}urea
2-amino-6-tert-butyl-4-(4-methyl-1H-imidazol-5-yl)pyridine-3-carbonitrile
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(1-ethyl-1H-pyrazole-3-carbonyl)piperidin-3-ol
1-[1'-(2,4-dimethylpyrimidine-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
1-(3-cyano-4-ethoxyphenyl)-3-[3-(methylsulfanyl)propyl]urea
3-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)propanoic acid
2-(dimethylamino)-8-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}-1,3,8-triazaspiro[4.5]dec-1-en-4-one
N-[(2,3-difluorophenyl)methyl]-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-4-carboxamide
1-cyclopropyl-4-{8-methyl-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}pyrrolidin-2-one
2-(phenylsulfanyl)-N-[1-({[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]acetamide
N-[2-(pyridin-3-ylformamido)ethyl]-2-(2,3,6-trimethylphenoxy)acetamide
4-[(2-amino-6-methylpyrimidin-4-yl)amino]-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-one
5-methoxy-2-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-4H-pyran-4-one
N-[(2S,4R,6R)-2-ethyl-6-heptyloxan-4-yl]acetamide
1-(pyridin-2-ylmethyl)-N-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-amine
1-{dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine
2-(3-{[3-(2-hydroxyethyl)-4-[1-(propan-2-yl)piperidin-4-yl]piperazin-1-yl]methyl}phenoxy)ethan-1-ol
1-[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(methylsulfanyl)ethan-1-one
3-methyl-1-[7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]piperidin-3-ol
5-{4-[(ethylcarbamoyl)amino]-3-methoxyphenyl}thiophene-2-carboxamide
1-(3-phenylpropyl)-5-(pyrrolidine-1-carbonyl)piperidin-2-one
5-(phenoxymethyl)-N-[1-(thiophen-3-yl)propan-2-yl]-1H-pyrazole-3-carboxamide
1-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
(2R)-1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}pyrrolidine-2-carboxamide
1-cyclohexyl-4-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperazine
4-(4-methanesulfonylphenyl)-5,6-dimethyl-2-(trifluoromethyl)pyrimidine
2-(benzyloxy)-N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methylacetamide