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2-(1H-indazol-3-yl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}acetamide
N-{[1-(methoxymethyl)cyclopropyl]methyl}-6-(3-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
(2E)-3-(4-methoxyphenyl)-1-[9-(oxan-2-ylmethoxy)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]prop-2-en-1-one
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-2-propoxyacetamide
2-(3-fluorophenyl)-1-[3-(4-fluorophenyl)-1H-pyrazole-5-carbonyl]azepane
1-[2-({[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}methyl)morpholin-4-yl]ethan-1-one
2-(8-methoxyquinolin-5-yl)-N,N-bis(propan-2-yl)benzamide
2-amino-6-(3,4-dimethoxyphenyl)-4-(furan-3-yl)pyridine-3-carbonitrile
4-(cyclopropylmethyl)-1-[3-(4-hydroxyphenyl)-1H-pyrazole-5-carbonyl]-3-(propan-2-yl)-1,4-diazepan-5-one
3-[(2-methylphenyl)methyl]-1-(pyridin-2-ylmethyl)piperidine-3-carboxylic acid
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(1-cyclopropyl-1H-pyrrole-2-carbonyl)pyrrolidin-3-yl]methanol
(3aS,6aS)-2-(oxan-4-yl)-5-[(phenylcarbamoyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
9-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-methyl-4-(4-{[methyl({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)amino]methyl}phenyl)but-3-yn-2-ol
N,N-dimethyl-5-(2-oxo-1,2-dihydroquinoline-4-carbonyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
4-{[3-(2,3-dimethoxyphenyl)pyrrolidin-1-yl]methyl}-1,3-thiazole
4-(1-{5-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-phenyl-1H-imidazol-1-yl}ethyl)pyrimidine
N-[(5-oxopyrrolidin-2-yl)methyl]-6-phenyl-N-(propan-2-yl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-[4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-6-(pyrrolidine-1-carbonyl)pyrazine
1-(4-methoxyphenyl)-5-[2-(oxolan-2-yl)ethyl]-1H-1,2,4-triazole
[(1R,3S,3aS,6aR)-5-benzyl-3-(2-fluoro-4-methylphenyl)-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
1-(azocan-1-yl)-3-(4-{[4-(cyclopropylmethyl)piperazin-1-yl]methyl}-2-methoxyphenoxy)propan-2-ol
N-{[1-(2-fluorophenyl)pyrrolidin-3-yl]methyl}-5-propyl-1,3,4-oxadiazol-2-amine
6-{4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}quinoxaline
4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-5-methyl-N-[2-(morpholin-4-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
3-{5-[2-(2-chloro-4-fluorophenyl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl){[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}amine
N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]acetamide
N-[3-(1H-indazol-1-yl)propyl]-2-(pyrrolidin-1-yl)-5,6,7,8-tetrahydroquinazoline-4-carboxamide
N-[(4-ethoxyphenyl)methyl]-N-(2-methoxyethyl)but-3-enamide
5-(methoxymethyl)-N-({7-[(3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)furan-2-carboxamide
N-[3-(methylsulfanyl)propyl]-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-(1-{4-[(oxolan-2-ylmethyl)(propyl)carbamoyl]phenyl}-1H-pyrazol-4-yl)pyridine-3-carboxamide
1-[2-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-oxoethyl]piperidin-2-one
(1S,5R)-3-(6-hydroxyhexyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(isoquinolin-5-ylmethyl)(methyl)(pyrrolidin-3-ylmethyl)amine
{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}[3-(1H-indazol-1-yl)propyl]amine
N-[(4-acetamidophenyl)methyl]-2-[2-(1,3-thiazol-2-yl)piperidin-1-yl]acetamide
1-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-3-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)urea
1-benzyl-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-1H-pyrazole-4-carboxamide
1-(2,6-diaminopyrimidin-4-yl)-4-(4-fluoro-2-methylphenoxy)piperidine-4-carboxylic acid
4-({4-methyl-5-[1-(2-phenylethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
(1S,5R)-3-(2-benzyl-1,3-thiazole-4-carbonyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(dimethylamino)-2-(2-methylphenyl)-1-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
4-[2-(aminomethyl)-5-methyl-2,3-dihydro-1-benzofuran-7-yl]-3-fluorobenzene-1-sulfonamide
1-(2-aminoethyl)-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-N'-(2-fluoro-5-methylphenyl)butanediamide
ethyl 4-benzyl-1-[(5-methylthiophen-2-yl)methyl]piperidine-4-carboxylate
2-(3-chlorophenyl)-N-[4-(4-{methyl[(5-propyl-1H-pyrazol-3-yl)methyl]amino}piperidin-1-yl)phenyl]acetamide