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3-(3-methoxypropyl)-1-[(6-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]piperidine-3-carboxylic acid
N-(4-chloro-2-methylphenyl)-4-({4-[(dimethylamino)methyl]-1H-1,2,3-triazol-1-yl}methyl)piperidine-1-carboxamide
4-fluoro-N-{[1-(furan-3-carbonyl)piperidin-3-yl]methyl}benzamide
6-[3-methyl-5-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-3-carboxamide
2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]benzamide
(3S)-4-[6-(3-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-1,3-dimethylpiperazin-2-one
N-cyclopropyl-5-[1-(2-hydroxyethyl)-1H-1,3-benzodiazol-2-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
3-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]pyridin-1-ium-1-olate
3-hexyl-8-[2-(1H-pyrazol-1-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(3S,4R)-1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
3-(2-methoxyethyl)-5-[(3-methoxyphenyl)methyl]-5-(piperidin-4-yl)imidazolidine-2,4-dione
1-{1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-(propan-2-yl)-1H-pyrazole-4-carbonyl}-4-methyl-1,4-diazepane
N4,6-dimethyl-N2-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]pyrimidine-2,4-diamine
2-[3-(4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-3,4-dihydroquinazolin-4-one
N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}-3-(pyridin-3-yl)propanamide
2-({4-benzyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)-1-propyl-1H-imidazole
4-[3-(2-chlorophenyl)-1H-pyrazol-5-yl]-1-(3-methyl-1,2-oxazole-5-carbonyl)piperidine
1-[(4-chlorophenyl)methyl]-4-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]piperazine
2-{3-[(4-benzoylpiperazin-1-yl)methyl]phenoxy}ethan-1-ol
5-ethyl-2-{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1H-imidazol-2-yl}pyridine
6-(1-benzofuran-2-yl)-2H-1,3-benzodioxole-5-carboxamide
1-(adamantan-1-yl)-4-(3-ethyl-1H-pyrazole-4-carbonyl)piperazine
N-methyl-2-[2-(propan-2-yl)-1H-imidazol-1-yl]-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
5-chloro-2-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidine-1-carbonyl]phenol
2-methoxy-1-[1'-(pyridine-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
(2S,4S)-1-benzyl-4-{[(2,6-difluorophenyl)methyl]amino}-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
N-{2-methyl-3-[(1,3-thiazol-2-yl)carbamoyl]phenyl}oxolane-3-carboxamide
2-(4-{1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}piperazin-1-yl)-1,3-benzoxazole
1-(3-chloro-4-methoxyphenyl)-5-oxo-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]pyrrolidine-3-carboxamide
2-(dimethylamino)-1-[(3S,4S)-3-hydroxy-4-[4-(2-methoxyphenyl)piperazin-1-yl]pyrrolidin-1-yl]ethan-1-one
2-chloro-4-[(3R,4R)-3-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-4-(hydroxymethyl)pyrrolidine-1-carbonyl]phenol
3-amino-N-[3-(2-methoxyacetamido)-2-methylphenyl]pyrrolidine-1-carboxamide
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-2-acetamidoacetamide
1-{4-[(2,3-dihydro-1H-inden-2-yl)amino]-2-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
9-methoxy-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-3-[2-(2-methylphenyl)acetyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[(4,6-dimethylpyridin-2-yl)methyl]-7-methanesulfonyl-N,4-dimethylquinazolin-2-amine
(2S,4R)-4-[2-(1H-imidazol-1-yl)acetamido]-N-methyl-1-[(2E)-3-phenylprop-2-en-1-yl]pyrrolidine-2-carboxamide
2-(2,2-dimethylpropanoyl)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-6-one
8-methyl-2-[3-(pyrimidin-2-yloxy)benzoyl]-2,8-diazaspiro[4.5]decane
ethyl 5-[(cyclopropylamino)methyl]-1-(4-phenyl-1,3-thiazol-2-yl)-1H-pyrazole-4-carboxylate
2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]-1-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]ethan-1-one
2-{5-[(1-propyl-1H-imidazol-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1H-1,3-benzodiazole
N-(2-{7-[(4-methoxy-2,3-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclobutanecarboxamide
N-[3-(3-chlorophenyl)phenyl]-1-[(4-hydroxy-3-methoxyphenyl)methyl]piperidine-4-carboxamide
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
3-[3-(4-phenyl-1H-imidazol-5-yl)-1H-indol-1-yl]propanamide
1-(4-fluorophenyl)-2,2-dimethyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]cyclopropane-1-carboxamide
7-(cyclopropylmethyl)-2-[2-(4-methoxyphenyl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
1-[(3-ethenylphenyl)methyl]-4-(3-fluoropyridin-2-yl)piperazine
2-(dimethyl-1,2-oxazol-4-yl)-N-[(3-methoxyphenyl)methyl]acetamide