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6-cyclopentyl-1-methyl-N-(oxolan-2-ylmethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(2S,4R)-N-ethyl-4-(2-phenylacetamido)-1-(pyridin-4-ylmethyl)pyrrolidine-2-carboxamide
N-(furan-2-ylmethyl)-N,1-dimethyl-5-({[1-(piperidin-1-yl)cyclopentyl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(4-methoxyphenyl)-3-methyl-4-[3-oxo-3-(pyrrolidin-1-yl)propyl]piperazin-2-one
2-(7-fluoro-2-methylquinoline-4-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
N-{[1-(ethoxymethyl)cyclopropyl]methyl}-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
5-methyl-N-[1-(1-propyl-1H-1,2,4-triazol-5-yl)ethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}-7-(3-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(1S,5R)-N-(4-fluorophenyl)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
(furan-3-ylmethyl)(methyl)({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amine
5-[3-(2-methylphenyl)phenyl]-5-(morpholin-4-yl)pent-3-yn-1-ol
2-{[(3aS,6aS)-5-(3-phenyl-1,2-oxazole-4-carbonyl)-octahydropyrrolo[3,4-b]pyrrol-1-yl]methyl}pyridine
{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amine
[2-(4-methoxyphenoxy)ethyl](methyl)[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amine
N-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}pyrazin-2-amine
2-{5-[(3-oxo-2,3-dihydro-1H-isoindol-1-yl)methyl]-3-(phenoxymethyl)-1H-1,2,4-triazol-1-yl}acetic acid
2-[(oxan-3-ylmethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
1-[(5-fluoro-2-methylphenyl)methyl]-2-(propan-2-yl)-1H-imidazole
5-(2-chloro-4-methoxyphenoxymethyl)-N-(2,3-dihydro-1H-inden-2-yl)-1,2-oxazole-3-carboxamide
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-{[1-(furan-2-yl)ethyl]amino}acetamide
2-{[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]methyl}benzoic acid
N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-1,3-benzothiazole-6-carboxamide
5-chloro-3-phenyl-2-[3-(1H-pyrazol-1-yl)azetidine-1-carbonyl]-1H-indole
1-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-3-yl]-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
N-{1-[(3-fluorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-3-(1H-1,2,4-triazol-1-yl)propanamide
3,5-dimethyl-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-1-benzofuran-2-carboxamide
N-[(2R)-1-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-1-oxobutan-2-yl]acetamide
2-{[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}-1,2-oxazolidine
6-[6-(dimethylamino)pyridin-3-yl]-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
2-ethyl-N-[2-(pyridin-3-ylformamido)ethyl]pyrimidine-5-carboxamide
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-benzyl-4-{[(3-methoxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
3-(diphenylmethyl)-5-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-1,2,4-oxadiazole
4-({4-[(3R)-3-methylpiperazine-1-carbonyl]furan-2-yl}methyl)morpholine
N-[1-(1H-imidazol-1-yl)butan-2-yl]-2,8-dimethylquinoline-4-carboxamide
N-[(3-ethoxyphenyl)methyl]-N-(2-hydroxyethyl)-1-oxo-1,2-dihydroisoquinoline-4-carboxamide
1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
1-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-3-phenoxypropan-1-one
N-[2-(3-methylthiophen-2-yl)ethyl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-1-[2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]propan-1-one
(1R,9S)-5-amino-3-(3,4-dihydroxyphenyl)-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
1-(cyclopropylmethyl)-4-(3-hydroxy-1,2-oxazole-5-carbonyl)-1,4-diazepane-6-carboxylic acid
3-[4-(3-chlorophenyl)-3-oxopiperazin-1-yl]-N-cyclohexylpropanamide
2-(2,4-dichlorophenoxy)-N-{1-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}acetamide
N-cyclohexyl-2-(3-fluorophenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
1-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-[(2-methoxyethyl)(methyl)amino]ethan-1-one
2-(2,3-difluorophenyl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
4-[(1-{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)methyl]morpholine
8-(5-ethyl-1,2,4-oxadiazol-3-yl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
3-(1-{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}piperidin-3-yl)propan-1-ol
2-(4-fluorophenyl)-N-(2-propoxyethyl)imidazo[1,2-a]pyridine-6-carboxamide