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4-{2-[2-(6-ethoxy-2,3-dihydro-1H-inden-5-yl)-1H-imidazol-1-yl]ethyl}-4H-1,2,4-triazole
(2S,4S)-4-amino-N,N-diethyl-1-[(4-methoxynaphthalen-1-yl)methyl]pyrrolidine-2-carboxamide
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
4-[(3-methoxypropyl)amino]-5-methyl-N-[2-phenyl-2-(piperidin-1-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
1-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-4-(furan-2-carbonyl)piperazine
4-[(2R,6S)-2,6-dimethylpiperidine-1-carbonyl]-2-(1-ethyl-1H-pyrazol-4-yl)-7-methylquinoline
3-(azepane-1-carbonyl)-1-methyl-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-cyclopropyl-1-{1-[(2-ethylpyrimidin-4-yl)methyl]piperidin-4-yl}piperidine-3-carboxamide
3-(dimethyl-1,2-oxazol-4-yl)-N-[2-(pyridin-3-ylformamido)ethyl]propanamide
5-(2,6-difluorophenoxymethyl)-N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
1-(2-methoxyphenyl)-4-[2-(methylamino)pyrimidine-5-carbonyl]piperazin-2-one
(1S,6R)-3-[3-(4-fluorophenoxy)propyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
2-({4-methyl-5-[1-(propan-2-yloxy)ethyl]-4H-1,2,4-triazol-3-yl}sulfanyl)acetic acid
2-(3-hydroxypropyl)-8-[(1-methyl-1H-imidazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-6-(methoxymethyl)-N,1-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-(ethylsulfanyl)-1-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
N-{1-[({2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}carbamoyl)methyl]-1H-pyrazol-4-yl}-2-(phenylsulfanyl)acetamide
6-({2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}amino)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
1-[2-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-oxoethyl]-4-ethylpiperazine-2,3-dione
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-ethyl-N-(pyridin-4-ylmethyl)-2,3-dihydro-1H-indene-2-carboxamide
2-(4-methylphenoxy)-N-[2-(1-methylpiperidin-3-yl)ethyl]acetamide
N-(1H-imidazol-2-ylmethyl)-N-methyl-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
2-methyl-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-2-(thiophen-2-ylformamido)propanamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-N'-(4-methyl-1,3-thiazol-2-yl)ethanediamide
8-fluoro-N-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]quinoline-2-carboxamide
2-{5-[(dimethylamino)methyl]furan-2-carbonyl}-2,7-diazaspiro[4.5]decan-6-one
{1-[(1-{[6-(trifluoromethyl)pyridin-3-yl]methyl}piperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}methanol
2-[8-(2,2-dimethylpropyl)-1-ethyl-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
2-{4-[(3,5-difluorophenyl)methyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-[2-({[2-fluoro-3-(trifluoromethyl)phenyl]methyl}amino)-4-methylpyrimidin-5-yl]ethan-1-one
N-[2-(1-benzofuran-2-ylmethyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]oxolane-2-carboxamide
propan-2-yl 5-[(2S)-2-amino-3-methoxypropanamido]-2-chlorobenzoate
N-[(3R,4S)-1-(cyclobutylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]-1-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)[(3-methoxyphenyl)methyl]methylamine
1-[2-(pyridin-2-yl)ethyl]-4-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine
N-[(2S,4R,6S)-2-(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)-6-ethyloxan-4-yl]benzamide
(1-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)(thiophen-2-yl)methanol
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-1-(4-methylphenyl)methanesulfonamide
4-{3-[4-(3-methylphenyl)piperazin-1-yl]propanoyl}-1λ6-thiomorpholine-1,1-dione
1-[3-(4-fluorophenyl)-1H-pyrazole-5-carbonyl]-4-(6-methylpyridin-2-yl)piperazine
[(3R,4R)-1-{[4-(5-methylfuran-2-yl)phenyl]methyl}-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
2-{1-[(4-ethylphenyl)methyl]-5-[1-(ethylsulfanyl)ethyl]-1H-1,2,4-triazol-3-yl}acetamide
methyl 1-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(3-methylbutyl)-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylate
1-methyl-4-[4-(pyrrolidine-1-carbonyl)phenyl]-1H-pyrazole
7-acetamido-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
1-({[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]carbamoyl}methyl)piperidine-4-carboxamide
3-(4-chlorophenyl)-N-(1H-imidazol-2-ylmethyl)-3-phenylpropanamide
1-{[4-(3-methylpiperidin-1-yl)phenyl]methyl}-3-(1-oxo-1,3-dihydro-2-benzofuran-5-yl)urea
5-(3-chlorothiophene-2-carbonyl)-3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
(3aR,6aS)-5-{2-[(2-ethyl-6-methylpyridin-3-yl)oxy]acetyl}-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid