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2-(1H-1,2,3,4-tetrazol-1-yl)-1-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
(1R,7S)-3-[2-(pyridin-4-yl)ethyl]-6-(5,6,7,8-tetrahydro-1,6-naphthyridine-6-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
(4aS,7aR)-1-{[4-(difluoromethoxy)phenyl]methyl}-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N,N-dimethyl-1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}azepan-4-amine
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-[methyl(propan-2-yl)amino]ethan-1-one
2-({3-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-ylmethyl]-6-methoxyquinolin-2-yl}sulfanyl)acetic acid
2-hydroxy-N-[(3R,4S)-1-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
3-({2-[1-(2,4-difluorobenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
2-{[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-5-ethylpyridine
(3aR,6aR)-2-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanoyl]-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[(4-methoxy-3-methylphenyl)methyl]-3-[2-(1,2-oxazinan-2-yl)-2-oxoethyl]piperazin-2-one
4-(methoxymethyl)-5-methyl-3-[1-(propan-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1,2-oxazole
4-[2-(1H-indazol-1-yl)acetyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
N-[4-chloro-2-(isoquinolin-5-yl)phenyl]acetamide
1-[5-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl](methyl)amino}methyl)-2-methoxyphenoxy]-3-(piperidin-1-yl)propan-2-ol
2-[(4aR,7aS)-4-(2-cyclohexylethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine
8-benzyl-1-(2-methylpropyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-methylpiperidine
1-(1-{4-[(2-methoxyphenyl)methyl]piperazine-1-carbonyl}-6-azaspiro[2.5]octan-6-yl)but-2-yn-1-one
N-{2-[7-(1H-indol-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-4-methylbenzamide
7-fluoro-3-[({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)methyl]-1,2-dihydroquinolin-2-one
1-[(diethylcarbamoyl)methyl]-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
1-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-2-(2-phenylethyl)piperidine
(2S)-2-amino-3-hydroxy-N-{[1-methyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-2-yl]methyl}propanamide
4-{7-[(2-methyl-1,3-oxazol-4-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}thiomorpholine
N-methyl-2-({6-[4-(pyridin-2-yl)piperazin-1-yl]pyridazin-3-yl}oxy)-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)acetamide
1-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-[(3-methylpyridin-2-yl)methyl]piperazine
N-benzyl-3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]-N-ethylpropanamide
3-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-3-methyl-1-[3-(2-methylpyrimidin-4-yl)phenyl]urea
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
4-[7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-2-yl]-N,N,5,6-tetramethylpyrimidin-2-amine
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(ethylsulfanyl)propan-1-one
5-[(4-methyl-1H-imidazol-1-yl)methyl]-3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazole
N-methyl-2-oxo-N-({4-oxo-3H,4H-thieno[3,2-d]pyrimidin-2-yl}methyl)-6-phenyl-1,2-dihydropyridine-3-carboxamide
2-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}acetamide
N-{[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-methoxybenzamide
3-{4-[(dimethyl-1,2-oxazol-4-yl)methyl]piperazin-1-yl}-2,5-dimethylpyrazine
6-[(3-fluorophenyl)methoxy]-1-(2-phenylethyl)-4-(1,3-thiazole-5-carbonyl)-1,4-diazepan-2-one
(1R,2S)-N-butyl-2-(3-phenoxyazetidine-1-carbonyl)cyclohexane-1-carboxamide
(2E)-3-(3-fluorophenyl)-1-[3-(4-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}phenoxymethyl)piperidin-1-yl]prop-2-en-1-one
N-[3-(furan-2-yl)phenyl]-1-(1-methyl-1H-pyrrole-2-carbonyl)piperidine-4-carboxamide
(2-methylpropyl)({[2-(morpholin-4-yl)pyridin-3-yl]methyl})(pyridin-2-ylmethyl)amine
dimethyl({6-[4-(methylsulfanyl)phenyl]pyridin-3-yl}methyl)amine
5-[1-(cyclohex-3-ene-1-carbonyl)piperidin-4-yl]-5-(pyridin-3-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
N-[(1S,2R,4R)-bicyclo[2.2.1]heptan-2-yl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-2-[4-(propan-2-yl)phenyl]acetic acid
N-{4-[2-(4-hydroxy-3-methoxyphenyl)-1H-imidazol-1-yl]-2-methylphenyl}-2-methoxyacetamide
N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-2,3-dimethyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1H-indole-7-carboxamide