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methyl 3-(furan-2-amido)-1-(2-methoxyethyl)-5-{[(4-methoxyphenyl)methyl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-{[2-(3-methoxyphenyl)pyrrolidin-1-yl]sulfonyl}-1,2,3,4-tetrahydroisoquinoline
3-{[3-(2-phenylethyl)piperidin-1-yl]methyl}pyridine
4-[(4aS,7aR)-4-(2-methylpropyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carbonyl]benzonitrile
(1S,5R)-6-(1H-indole-6-carbonyl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-2-(2-oxopyrrolidin-1-yl)acetamide
7-{[4-(benzyloxy)piperidin-1-yl]methyl}-4-[(1R,2R)-2-phenylcyclopropanecarbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
(1R,5R)-6-(cyclobutylmethyl)-3-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
(1S,5R)-6-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
1-[2-({[methyl(propan-2-yl)sulfamoyl]amino}methyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]ethan-1-one
(1R,7S)-3-(4-fluorophenyl)-6-(thiomorpholine-4-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
9-ethyl-4-{[4-(2-hydroxyethoxy)phenyl]methyl}-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-[(2-methylphenyl)methyl]-3-(pyrrolidin-1-yl)piperidine
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(1R,3S,5S)-8-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octane
N-cyclopropyl-2-[(1S,4S)-5-(2-methoxy-5-phenylphenyl)-6-oxo-2,5-diazabicyclo[2.2.1]heptan-2-yl]acetamide
N-[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
3-(1-{[2-(2,2-dimethylpropanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperidin-2-yl)pyridine
N-{[1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]methyl}-2-methyl-2-phenylpropanamide
2-[4-methyl-2-(3-methyl-1H-pyrazol-1-yl)phenoxy]acetamide
1-[(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-3-hydroxypiperidin-1-yl]-2-(1-methyl-1H-pyrrol-3-yl)ethan-1-one
N-({5-[(4-methoxy-2-methylphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
1-[2-(benzyloxy)ethyl]-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
1-{2-[(2-ethoxyphenyl)carbamoyl]acetyl}piperidine-3-carboxylic acid
4-(1-{2-methylthieno[3,2-d]pyrimidin-4-yl}piperidin-3-yl)pyrimidine
1-[5-(2,5-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]-4-(pyrrolidin-1-yl)piperidine
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-ethoxyethan-1-one
(3aS,6aS)-2-cyclopropanecarbonyl-5-(pentylcarbamoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(2S,4R,6S)-2-ethyl-6-(5-methyl-1-propyl-1H-pyrazol-4-yl)oxan-4-yl]benzamide
1-[3-(1H-imidazol-2-yl)benzoyl]-3-(3-methoxybenzoyl)piperidine
{3-[(3-chlorophenyl)methyl]-1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-3-yl}methanol
(3R,4R)-3-cyclopropyl-1-(5-fluoro-4-methoxypyrimidin-2-yl)-4-methylpyrrolidin-3-ol
2-[benzyl(methyl)amino]-N-[2-(1H-imidazol-1-yl)ethyl]-6-(thiophen-3-yl)pyridine-3-carboxamide
N-(dicyclopropylmethyl)-2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-methylacetamide
(1S,5R)-6-(cyclobutylmethyl)-3-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-methyl-2-(4H-1,2,4-triazol-4-yl)pyridine
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(propylamino)benzamide
6-methyl-4-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]-2-(1H-pyrazol-4-yl)quinoline
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]quinoline-3-carboxamide
(1S,5R)-3-(1-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
6-{[2-(piperidin-1-yl)phenyl]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
5-(4-benzylpiperidine-1-carbonyl)-N-ethyl-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3-carboxamide
3-(azocan-1-yl)-N-[4-(morpholin-4-yl)butan-2-yl]propanamide
7-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidine-1-carbonyl]quinolin-8-ol
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl]amine
N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]-1H-indole-6-carboxamide
1-(3-chloro-4-methylphenyl)-3-[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl]-3-methylurea
4-(2-methoxypyridine-4-carbonyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
1-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}ethan-1-one
(3aR,6aR)-2-benzyl-N-[2-(2-hydroxyethoxy)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide