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1-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}-3-propoxypiperidine
2-{4-[(3,4-difluorophenyl)methyl]-1-[(3,5-dimethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-cyclopropyl-N-{1-[1-(furan-3-ylmethyl)piperidin-4-yl]-2-phenylethyl}pyridine-2-carboxamide
4-cyclopentyl-3-oxo-N-(3-phenyl-1,2,4-thiadiazol-5-yl)piperazine-1-carboxamide
2-[(4-chlorophenyl)methyl]-8-(pyridin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
N-[(3S,4R)-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-2-(pyrrolidin-1-yl)benzamide
N-(pyridin-2-ylmethyl)-1-[2-(trimethyl-1H-pyrazol-1-yl)acetyl]piperazine-2-carboxamide
4-methyl-N-{2-[1-(2-methylpropyl)piperidin-3-yl]ethyl}-1H-imidazole-5-carboxamide
1-{4-[(4-methylpiperazin-1-yl)methyl]phenoxy}-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
3-(1-cyclopentyl-4-methyl-1H-pyrazol-5-yl)-1-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}urea
2-[1'-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-2-oxo-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-1-yl]acetamide
2-(2-methoxyethyl)-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,3-benzoxazole-6-carboxamide
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-{[4-(dimethylamino)oxan-4-yl]methyl}urea
2-(benzyloxy)-1-[4-(3-hydroxypiperidin-1-yl)piperidin-1-yl]ethan-1-one
5-[3-(2-chlorophenyl)pyrrolidine-1-carbonyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole
N-[1-(morpholine-4-carbonyl)piperidin-4-yl]-1H-1,2,3-benzotriazole-5-carboxamide
N-[4-(2-methoxyphenyl)-1,3-dimethyl-1H-pyrazol-5-yl]-3-oxopiperazine-1-carboxamide
methyl 3-({2-methyl-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}sulfonyl)thiophene-2-carboxylate
5-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyridine-2-carbonitrile
5-{[(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)amino]methyl}pyrimidin-2-amine
[(3R,4R)-1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
3-[4-(1-hydroxy-2-phenylethyl)piperidine-1-carbonyl]-2-methylphenol
2-{3,5-dimethyl-4-[4-(2-oxopyrrolidin-1-yl)benzamido]-1H-pyrazol-1-yl}acetic acid
[5-({4-[(4-chlorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}methyl)furan-2-yl]methanol
1-{[5-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-4,4-difluoropiperidine
3-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
N-(3,4-dimethylphenyl)-1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperidin-3-amine
1-{2-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-({3-hydroxy-1-[(3-methoxyphenyl)methyl]-2-oxopiperidin-3-yl}methyl)-3,3-dimethylpiperazin-2-one
8-(2-hydroxypropyl)-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)-6-methoxy-1H-indazole
6-(3-hydroxypiperidin-1-yl)-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
8-(5-chloro-2-methylbenzoyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(2S,4R,6S)-2-(3-cyanophenyl)-6-ethyloxan-4-yl]benzamide
1-(1-propyl-1H-pyrazole-5-carbonyl)-3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine
N-[(4-hydroxy-6-methylpyrimidin-2-yl)methyl]-2-(thiophen-2-yl)acetamide
6-(4-methylpiperazin-1-yl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
(2S)-1-{2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxybenzoyl}-4-methyl-2-(propan-2-yl)piperazine
2-(4-{[(1R,3S,5S)-3-(4-methoxyphenyl)-8-azabicyclo[3.2.1]octan-8-yl]methyl}-3-methyl-1H-pyrazol-1-yl)ethan-1-ol
5-{3-[1-(4,4,4-trifluorobutyl)-1H-pyrazol-3-yl]phenyl}pyrimidine
N-[1-({[2-methoxy-2-(thiophen-2-yl)ethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-3-phenoxypropanamide
2,6-dihydroxy-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]benzamide
4-(2-methylfuran-3-carbonyl)-N-[2-(pyridin-2-yl)ethyl]morpholine-2-carboxamide
N-cyclopropyl-4-methoxy-3-({1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}oxy)benzamide
1-{3-[benzyl(methyl)amino]piperidin-1-yl}-3-(4-methoxyphenyl)propan-1-one
3-{2-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
8-methyl-N-(oxolan-2-ylmethyl)-N-(2-phenoxyethyl)imidazo[1,2-a]pyridine-2-carboxamide
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-{1,4,6-trimethyl-1H-pyrazolo[3,4-b]pyridin-3-yl}acetamide
{4-[5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]morpholin-3-yl}methanol