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N-[(3R,4S)-1-(4-aminopyrimidin-2-yl)-4-(propan-2-yl)pyrrolidin-3-yl]pyrrolidine-1-sulfonamide
N-(cyclopropylmethyl)-4-[(2,5-dihydroxy-2-methylpentyl)sulfamoyl]benzamide
2-(2H-1,3-benzodioxol-5-yl)-1-{9-methoxy-7-[5-(trifluoromethyl)pyridin-2-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}ethan-1-one
9-[3-(azetidine-1-carbonyl)benzenesulfonyl]-3-oxa-9-azaspiro[5.5]undecane
4-(1H-imidazol-2-yl)-1-methyl-3-(4-phenoxyphenyl)-1H-pyrazole
3-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-6-ethyl-1,5-dimethyl-1,2-dihydropyridin-2-one
1-{4-[2-methoxy-5-(pyrrolidin-1-ylmethyl)phenoxy]phenyl}-1H-pyrazole
{1-[(2,3-difluoro-6-methoxyphenyl)methyl]azepan-2-yl}methanol
methyl 5-oxo-5-[6-oxo-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-2-yl]pentanoate
{[2-(furan-2-yl)pyrimidin-5-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
1-butyl-5-[(4,5-dimethyl-1H-imidazol-1-yl)methyl]-3-(furan-2-yl)-1H-1,2,4-triazole
N-[(3S,4R)-1-[3-(dimethylcarbamoyl)propanoyl]-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
N3-[(2,4-difluorophenyl)methyl]-1-(2-methoxyethyl)-4-oxo-N5-[1-(thiophen-2-yl)propyl]-1,4-dihydropyridine-3,5-dicarboxamide
(3S,4R)-1-[3-(dimethylsulfamoyl)propyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
N,N-dimethyl-3-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrazin-2-amine
ethyl 4-(4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-amido)piperidine-1-carboxylate
6-oxo-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]-1,4,5,6-tetrahydropyridazine-3-carboxamide
3-({3-[2-oxo-2-(thiomorpholin-4-yl)ethyl]morpholin-4-yl}methyl)-1,2-dihydroquinolin-2-one
4-[(2-fluorophenyl)methyl]-11-[4-(pyridin-3-ylmethyl)piperazin-1-yl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-(7-fluoro-2-methyl-1H-indol-3-yl)-1-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}ethan-1-one
3-[1-(1,1-dioxo-1λ6-thian-4-yl)piperidin-4-yl]-1-(4-methoxyphenyl)urea
N-methyl-2-[3-(pyridin-4-yl)azetidin-1-yl]-5H,6H,7H-cyclopenta[d]pyrimidin-4-amine
1-methyl-9-{2-[3-(trifluoromethyl)phenyl]acetyl}-1,4,9-triazaspiro[5.5]undecan-5-one
1-[3-(2,6-dimethylphenoxy)azetidin-1-yl]-2-(3-fluoro-4-hydroxyphenyl)ethan-1-one
1-cyclopentyl-4-{[(1H-indol-5-ylmethyl)(methyl)amino]methyl}pyrrolidin-2-one
9-methoxy-N-methyl-3-[2-(3-methylphenyl)acetyl]-7-oxo-N-(1,3-thiazol-4-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-(1,4-dioxan-2-ylmethyl)-1-{4-[2-(pyridin-2-yl)ethoxy]phenyl}urea
6-phenyl-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
(4-{[1-(3-fluoro-4-methylbenzoyl)pyrrolidin-3-yl]methyl}phenyl)methanol
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(5-methyl-1,2-oxazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
6,8-dimethyl-2-{[methyl(oxan-4-yl)amino]methyl}quinolin-4-ol
6-fluoro-2-{[4-(oxolane-2-carbonyl)piperazin-1-yl]methyl}quinolin-4-ol
3-(1,2-diethyl-1H-1,3-benzodiazol-5-yl)-1-[2-methoxy-1-(pyridin-2-yl)ethyl]-1-methylurea
N-(1H-1,3-benzodiazol-2-ylmethyl)-N-methyl-3-(5-phenyl-1,3,4-oxadiazol-2-yl)propanamide
5-{4-[(3,3,4-trimethylpiperazin-1-yl)methyl]phenoxymethyl}furan-2-carboxylic acid
ethyl 2-[methyl({[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]-1,3-oxazole-4-carboxylate
6-[(1R,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]hexan-1-ol
5-{2-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-oxoethyl}-2-methyl-3,4-dihydropyrimidin-4-one
(3S,4R)-4-methyl-1-[6-methyl-2-(morpholin-4-yl)pyrimidin-4-yl]piperidine-3,4-diol
4-{2-[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]-2-oxoethyl}-7-methyl-2H-chromen-2-one
2-(benzyloxy)-1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]ethan-1-one
3-(azocan-1-yl)-1-[4-(morpholin-4-ylmethyl)piperidin-1-yl]propan-1-one
9-[(4-methyl-1H-imidazol-5-yl)methyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(2-methoxyethyl)-6-oxo-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}piperidine-3-carboxamide
N-(4-{[3-(naphthalene-1-carbonyl)piperidin-1-yl]methyl}phenyl)acetamide
(2S)-3-methyl-2-({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)butanamide
[(4aS,8aR)-6-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}-decahydro-1,6-naphthyridin-4a-yl]methanol
5-methyl-3-phenyl-4-{1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-1,2-oxazole
4-[2-(2-chloro-4,5-difluorophenyl)acetyl]-1-(4-methylphenyl)piperazin-2-one
N,N-diethyl-2-{[2-oxo-1-(2-phenylethyl)-4-[3-(pyridin-4-yl)propanoyl]-1,4-diazepan-6-yl]oxy}acetamide