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9-methoxy-7-(2-methoxyphenyl)-4-(pyridine-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-(1,2-oxazinan-2-yl)-1-{4-[(propan-2-yl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}propan-1-one
5-chloro-N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}thiophene-2-carboxamide
(3S,9aR)-8-(2-chlorobenzoyl)-3-[(4-chlorophenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-cyclobutaneamido-N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)benzamide
3-(2-chlorophenyl)-1-cyclopentyl-3-{2-[4-(4-methyl-1,2,5-oxadiazol-3-yl)piperazin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
N-[1-(cyclohexylmethyl)piperidin-3-yl]-2-(2,4-difluorophenyl)acetamide
4-cyclopropyl-6-[4-(4H-1,2,4-triazol-4-yl)piperidin-1-yl]pyrimidine
2-(2-{[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
N-(6-fluoropyridin-3-yl)-6-oxa-9-azaspiro[4.5]decane-9-carboxamide
2-[9-(3-methoxybenzoyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]propanoic acid
N-(4-fluoro-2-methylphenyl)-2-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepin-9-ylformamido}acetamide
N-(4-{2-[2-(2-methylphenyl)pyrrolidin-1-yl]-2-oxoethoxy}phenyl)propanamide
(2-{[4-(furan-3-ylmethyl)piperazin-1-yl]methyl}phenyl)methanol
N-cyclopropyl-1-(1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperidin-4-yl)piperidine-3-carboxamide
6-fluoro-4-(6-methoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-2-(pyrimidin-5-yl)quinoline
2-(ethylsulfanyl)-5-[1-(3-methoxyphenyl)-1H-imidazol-2-yl]pyrimidine
4-(4-chlorophenoxy)-N-[2-(pyridin-2-yl)ethyl]piperidine-4-carboxamide
1-ethyl-5-[1-(pyrimidin-2-yl)piperidine-4-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
3-[(2-fluoroethyl)sulfamoyl]-N-[(1-methylpiperidin-2-yl)methyl]benzamide
(1S,5R)-6-(1-methyl-1H-pyrazole-4-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
3-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
2-{2-[2-(2-butyl-1H-imidazol-4-yl)-1H-imidazol-1-yl]ethyl}pyridine
1-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(thiophen-2-yl)propan-1-one
9-oxo-N-(propan-2-yl)-8-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecane-2-carboxamide
[(2,2-dimethyl-1-phenylcyclopropyl)methyl][(4-methanesulfonylphenyl)methyl]methylamine
2,3,5-trimethyl-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
2-({[(3R,4R)-1-(2-ethylpyridine-4-carbonyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-(2-{[1-(4-fluorophenyl)pyrrolidin-3-yl]amino}ethyl)-N-methylmethanesulfonamide
5-[1-(2,2-dimethylpropyl)piperidin-4-yl]-3-(2-methoxyethyl)-5-[(3-methoxyphenyl)methyl]imidazolidine-2,4-dione
5-[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidine-1-carbonyl]pyrazin-2-ol
4-{[1-(1-acetylpiperidin-4-yl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
3-{[3-(pyridin-3-yl)azetidin-1-yl]methyl}-1λ6-thiane-1,1-dione
3-(1-cyclopentyl-1H-pyrazol-5-yl)-1-({2-[(2-oxopyrrolidin-1-yl)methyl]phenyl}methyl)urea
2-oxo-5-{[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]methyl}-2,3-dihydro-1H-imidazole-4-carboxylic acid
1-[2-methoxy-5-({[2-(2-methylphenyl)ethyl]amino}methyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
3-(2-methoxybenzoyl)-1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidine
3-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N,N-dimethyl-3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]piperidine-1-carboxamide
6-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidine-1-carbonyl)-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-{[(1H-indazol-4-yl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-(2-{[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]amino}ethyl)-N-methylmethanesulfonamide
1-butyl-4-[2-(4-methoxypiperidin-1-yl)-2-oxo-1-phenylethyl]piperazine-2,3-dione
[4-(oxan-2-ylmethyl)-1-(6-phenylpyridazin-3-yl)piperidin-4-yl]methanol
N-[1-(2-chlorophenyl)cyclopropyl]-3-(1-methylpiperidin-2-yl)propanamide
1-(3-{2-[(2-chlorophenyl)methyl]morpholin-4-yl}-3-oxopropyl)azepan-2-one
1-[(1S,3R)-1-ethoxy-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propan-1-one
(3-{2-[1-(5-chloro-3-fluoropyridin-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
3-{2-[4-(3,5-dimethylphenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}-1-(2-methoxyethyl)-3-(2-methylphenyl)pyrrolidine-2,5-dione
N-cyclopropyl-3-[5-(oxan-2-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanamide