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(2S)-2-amino-N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3-hydroxypropanamide
9-ethyl-1-methyl-4-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
4-[(4-fluoro-3-methylphenyl)methyl]-9-(2-methoxyethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
5-{[bis(1,3-oxazol-4-ylmethyl)amino]methyl}-N,N-dimethylpyridin-2-amine
4-[1-(1-{[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)ethyl]morpholine
3-chloro-N-[2-(2-ethylphenoxy)ethyl]-N,6-dimethylpyrazolo[1,5-a]pyrimidine-2-carboxamide
1-[3-({[2-(4-acetylpiperazin-1-yl)-7-chloroquinolin-3-yl]methyl}amino)propyl]pyrrolidin-2-one
7-[(2,3-dimethoxyphenyl)methyl]-2-(pyridin-2-ylmethyl)-2,7-diazaspiro[4.5]decane
2-(2-aminoethyl)-N-[4-(4-methoxyphenyl)phenyl]morpholine-4-carboxamide
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
1-({5-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)-4-methylpiperazine
7-[(4-fluorophenyl)methyl]-2-(pyrrolidine-1-sulfonyl)-2,7-diazaspiro[4.5]decane
4-[(5-chloro-2,4-dimethoxyphenyl)methyl]-2-ethyl-1-(propan-2-yl)piperazine
6-[5-(methoxymethyl)furan-2-carbonyl]-4-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-amine
4-{5-[(4-acetylpiperazin-1-yl)methyl]-1,2,4-oxadiazol-3-yl}benzoic acid
3-{1-[(2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl)methyl]piperidin-3-yl}-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
4-[(3-fluorophenyl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[(2-chlorophenyl)methyl]-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-[2-(pyridin-3-yl)ethyl]pyrimidine-5-carboxamide
5-{1-[(2-methoxynaphthalen-1-yl)methyl]-1H-imidazol-2-yl}-1,2-dimethyl-1H-imidazole
2-fluoro-1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]-2-phenylethan-1-one
1-{5-cycloheptyl-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidin-3-ol
4-benzyl-2-{2-[(3S,4S)-3,4-dihydroxypiperidin-1-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
2-(5-chloro-6-methyl-1-benzofuran-3-yl)-1-[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]ethan-1-one
2,6-diamino-4-[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
dimethyl[(4-methyl-5-{1-[(5-propylfuran-2-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]amine
(1R,5R)-6-(cyclobutylmethyl)-3-(1H-pyrazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-[(dimethyl-1,2-oxazol-4-yl)methyl]-5-methyl-5-(4-methylpent-3-en-1-yl)piperidin-2-one
methyl (2S,4R)-1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-hydroxypyrrolidine-2-carboxylate
N-cyclopropyl-3-[1-(pyridin-4-ylmethyl)piperidin-4-yl]propanamide
3-[2-(3-aminopyrrolidin-1-yl)-2-oxoethyl]-1-[(4-fluorophenyl)methyl]-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
2-amino-4-(3,4-dihydroxyphenyl)-6-(1H-indol-3-yl)pyridine-3-carbonitrile
N,N-dimethyl-1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-sulfonamide
1-(1H-imidazol-2-ylmethyl)-8-(quinoxalin-2-yl)-1,8-diazaspiro[4.5]decane
N-[(6-ethoxyquinolin-2-yl)methyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
3-cyclopropyl-5-[(1S,4S)-3,3-dimethyl-2-methylidenebicyclo[2.2.1]heptan-1-yl]-1H-1,2,4-triazole
8-(6-oxo-1,6-dihydropyridine-3-carbonyl)-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-benzyl-2-{3-[3-(pyrazin-2-yl)phenyl]-1H-pyrazol-1-yl}acetamide
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methyl-1-phenyl-1H-1,2,3-triazole-5-carboxamide
1-(2-ethylbutanoyl)-N-[2-(4-methoxyphenyl)phenyl]pyrrolidine-2-carboxamide
5-cyclobutyl-N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N-methyl-1,3,4-oxadiazol-2-amine
ethyl 2-{4-[2-(3-phenylpropyl)-1,3-benzoxazole-5-carbonyl]morpholin-3-yl}acetate
2-[(3-methoxyphenyl)methyl]-8-[2-(oxolan-3-yl)ethyl]-2,8-diazaspiro[4.5]decan-3-one
5-methyl-2-[4-(methylsulfanyl)phenyl]-4-(1H-pyrazol-1-ylmethyl)-1,3-oxazole
7-(2-methylphenyl)-4-[2-(1-methylpyrrolidin-2-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(4-fluorophenyl)-5-[1-(1H-imidazol-1-yl)ethyl]-3-(2-methylpropyl)-1H-1,2,4-triazole
5-hydroxy-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-N-(prop-2-en-1-yl)pyrazine-2-carboxamide
2-(dimethylamino)-2-(4-methylphenyl)-N-[(1-propyl-1H-pyrazol-4-yl)methyl]acetamide
ethyl 2-[1-(1-methyl-2-oxo-1,2-dihydroquinoline-4-carbonyl)piperidin-2-yl]acetate
1-[5-(2-chlorophenyl)furan-2-carbonyl]-2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidine