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5-(2-methoxyphenoxymethyl)-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1H-pyrazole-3-carboxamide
2,6-dimethyl-N-[2-(N-methylmethanesulfonamido)ethyl]pyrimidine-4-carboxamide
3-methoxy-1-{4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}propan-1-one
4-({1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}amino)-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid
4-({4-methyl-5-[1-(3-methylpyrazin-2-yl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
N-cyclopropyl-4-(3,5-dimethyl-1H-pyrazol-4-yl)benzamide
4,6-dimethyl-2-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyridine-3-carboxamide
1-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-3-(piperidin-1-yl)propan-1-one
2-ethyl-6-(3-methanesulfonylbenzoyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
3-(2-chlorophenyl)-1-cyclopentyl-3-{2-[3-(methoxymethyl)piperidin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
6-fluoro-2-{[3-(2-methoxyphenoxy)azetidin-1-yl]methyl}quinoline
3-(1H-1,3-benzodiazol-2-yl)-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]propanamide
5-(2-chlorophenyl)-3-{[2-(oxolan-3-yl)-1H-imidazol-1-yl]methyl}-1,2-oxazole
ethyl 1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylate
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-[3-(pyridin-3-yloxy)propyl]acetamide
(2S,4S)-4-({[4-(dimethylamino)phenyl]methyl}amino)-N-[2-(2-fluorophenyl)ethyl]-1-(2-methylpropyl)pyrrolidine-2-carboxamide
(3S,5R)-1-(4-propylpyrimidine-5-carbonyl)-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxylic acid
1-{[2-(cyclopentyloxy)phenyl]methyl}-4-(pyridin-2-ylmethyl)-1,4-diazepane
4-[2-(3-{[3-(2-methylpiperidin-1-yl)azetidin-1-yl]methyl}phenoxy)ethyl]morpholine
4-(pyridin-2-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]pyrimidin-2-amine
6-[(1R,9aR)-octahydro-1H-quinolizin-1-ylmethoxy]-2,3-dihydro-1-benzofuran-3-one
7-(5-chloropyridin-2-yl)-4-cyclohexyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-3-(1H-pyrazol-1-ylmethyl)benzamide
3-{[3-(2-hydroxyethyl)-4-(3-methylbutyl)piperazin-1-yl]methyl}-4H-chromen-4-one
2-[3-methyl-5-(pyrrolidin-1-ylmethyl)phenoxy]-5-(trifluoromethyl)pyridine
2-{4-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}-N-methylacetamide
3-methyl-1-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1,2-dihydroquinoxalin-2-one
7-(2-methoxyphenyl)-2-[3-(methylsulfanyl)phenyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
8-[2-(azepan-1-yl)-2-oxoethyl]-2-cyclopropyl-2,8-diazaspiro[5.5]undecan-3-one
3-methyl-1-{5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}piperidin-3-ol
(3S,4S)-1-(2-amino-6-methoxypyrimidin-4-yl)-4-propylpyrrolidine-3-carboxylic acid
3-[(1-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidin-4-yl)oxy]pyridine
3-chloro-N-cyclopentyl-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
7-[(1S,4S)-3,3-dimethyl-2-methylidenebicyclo[2.2.1]heptane-1-carbonyl]-5H,6H,7H,8H-imidazo[1,5-a]pyrazine
6-methyl-5-(2-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-4-(1H-1,2,4-triazol-1-yl)butanamide
3-(2-fluorophenyl)-1-{imidazo[1,2-a]pyridine-6-carbonyl}pyrrolidine
{[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]sulfamoyl}dimethylamine
2-(dimethylamino)-2-(3-fluorophenyl)-N-{[(propan-2-yl)carbamoyl]methyl}acetamide
(2S,4S)-4-amino-1-[3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)propanoyl]-N-ethylpyrrolidine-2-carboxamide
5-amino-N-[(3R,5S)-1-cyclohexyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]-1H-pyrazole-3-carboxamide
6-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]quinoline
N,N-dimethyl-4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-sulfonamide
N-(1-{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2H-1,3-benzodioxole-5-carboxamide
2-(2-hydroxypropanoyl)-N-methyl-N-(1,3-thiazol-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
N-ethyl-5-[1-(1H-indol-6-ylmethyl)-1H-1,2,3-triazol-4-yl]pyrimidin-2-amine
N-[3-(1H-imidazol-5-yl)phenyl]-4-(oxan-4-yl)piperazine-1-carboxamide
2-[(1,4-oxazepan-6-ylmethyl)amino]pyridine-3-carboxamide
1-(1,3-dimethyl-4-phenyl-1H-pyrazol-5-yl)-3-[2-(dimethylsulfamoyl)ethyl]urea
methyl 2-[(3,4-difluorophenyl)sulfamoyl]-6-(2-ethylbutanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate