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6-{[3-(diethylcarbamoyl)piperidin-1-yl]methyl}-2-oxo-N-(thiophen-3-ylmethyl)-1,2-dihydropyridine-3-carboxamide
cyclopentyl 4-{[3-(4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]amino}benzoate
N-(2-{5-[(2-methoxyethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}ethyl)-3-(4-methylphenyl)propanamide
N-({7-[(4-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-(pyridin-3-yl)propanamide
8-(3-aminopropanoyl)-2-[(3,5-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
methyl 3-[2-(dimethylcarbamoyl)ethyl]-1-(2-methoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylate
5-methoxy-2-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine-1-carbonyl)-4H-pyran-4-one
2-(dimethylamino)-2-(3-fluorophenyl)-1-[4-(morpholin-4-yl)piperidin-1-yl]ethan-1-one
N-[3-(phenylsulfanyl)propyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
[(4-ethyl-5-{1-[(1-methyl-1H-indol-2-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
2-phenyl-4-(thiophen-3-ylmethyl)morpholine
{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-1-(4-methoxyphenyl)-N-methylcyclopropane-1-carboxamide
2-chloro-5-(1H-pyrazol-1-yl)-N-[2-(pyrrolidin-1-yl)ethyl]benzamide
1-(3-{3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}-3-oxopropyl)pyrrolidin-2-one
1-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]-4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-5-one
8-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazole-5-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-1,2,5-oxadiazole-3-carboxamide
5-{1-[(2,4-dimethylphenyl)methyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
methyl 6-[(6-hydroxy-1,4-oxazepane-4-carbonyl)amino]-1,2,3,4-tetrahydroquinoline-1-carboxylate
(3R,4S)-4-cyclopropyl-N,N-dimethyl-1-[4-(pyrrolidine-1-carbonyl)pyridin-2-yl]pyrrolidin-3-amine
N-[2-(dimethylamino)ethyl]-N-ethyl-1-[4-(furan-2-yl)pyrimidin-2-yl]-5-(propan-2-yl)-1H-pyrazole-4-carboxamide
4-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1,4-diazepane-1-carbaldehyde
2-ethyl-5-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}pyrimidine
N-(dimethyl-1,2-oxazol-4-yl)-4-(5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carboxamide
4-{4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]piperazin-1-yl}-2-{[3-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindole-1,3-dione
2-(5-methyl-1,2-oxazol-3-yl)-1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidine
(S)-cyclopropyl[3-(oxan-4-yl)-1-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methanamine
1-[3-({4-[4-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)phenyl]ethan-1-one
5-[2-(3-methylphenoxy)propan-2-yl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
4-cyclopentyl-9-methoxy-7-(6-methoxypyridazin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-phenoxy-2-[4-(thiophen-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]propan-2-ol
N-{2-[2-(trifluoromethoxy)phenyl]ethyl}-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
5-(2-{5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}-1H-imidazol-1-yl)-4,5,6,7-tetrahydro-1H-indazole
3-(2H-1,3-benzodioxole-5-carbonyl)-1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}piperidine
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}propanamide
4-[1-hydroxy-2-({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]phenol
N-[5-(2-fluorophenyl)-4H-1,2,4-triazol-3-yl]-4-(thiophene-2-carbonyl)piperazine-1-carboxamide
2-(methylamino)-1-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)ethan-1-one
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-3-(3,4-dimethoxyphenyl)propan-1-one
3-[(5-methylpyrazin-2-yl)methyl]-1-{3-[2-(morpholin-4-yl)-2-oxoethoxy]phenyl}urea
N-[2-(dimethylamino)ethyl]-5-(1H-indole-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-3-(4-fluorophenyl)-1H-pyrazole-5-carboxamide
1-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}-3-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]urea
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-1,2-oxazole-3-carboxamide
1-[(2,5-dimethylphenyl)methyl]-4-ethyl-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl 4-(5-{[3-(acetamidomethyl)piperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
5-oxo-N-[2-(4-phenylpyrimidin-2-yl)ethyl]-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
(3R,4R)-4-(morpholin-4-yl)-1-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}piperidin-3-ol