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3-[2-(4H-1,2,4-triazol-4-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazole
3-(2-oxo-2-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}ethyl)-3,4-dihydroquinazolin-4-one
N-cyclohexyl-3-[(3-propyl-1H-pyrazol-5-yl)formamido]propanamide
1-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-ol
4,6-dimethyl-2-(4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperazin-1-yl)pyrimidine
2-[(4-methoxyphenyl)methyl]-4-(7-methyl-1-benzofuran-2-carbonyl)morpholine
2-methoxy-N-{1-[1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-phenylacetamide
N-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]-8-fluoroquinoline-2-carboxamide
4-methyl-2-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
3-[2-(4-fluorophenyl)ethyl]-1-(5-propyl-1,2-oxazole-3-carbonyl)piperidine
methyl 5-{[(2-chloro-6-fluorophenyl)methyl]amino}-1-methyl-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(2S,4R,6R)-2-(2,1,3-benzoxadiazol-4-yl)-6-tert-butyloxan-4-yl]acetamide
N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-3-methoxypropanamide
N-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine-1-carboxamide
3-{[(5-acetylthiophen-3-yl)methyl](ethyl)amino}-1λ6-thiolane-1,1-dione
9-(1,3-benzothiazol-2-yl)-5-methoxy-1-oxa-9-azaspiro[5.5]undecane
4,6-dimethyl-2-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
4-methyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-3-(2-oxoimidazolidin-1-yl)benzamide
1-ethyl-4-{[2-(furan-2-yl)azepan-1-yl]methyl}-1H-pyrrole-2-carbonitrile
(1S,5R)-6-[(dimethylcarbamoyl)methyl]-N-[(4-methoxyphenyl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
9-(2-methoxy-4-methylbenzenesulfonyl)-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
5-[4-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperazin-1-yl]-2-methyl-2,3-dihydropyridazin-3-one
ethyl 1-[4-(methoxycarbonyl)benzoyl]-4-[(4-methoxyphenyl)methyl]piperidine-4-carboxylate
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
N-methyl-N-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}aniline
2-cyclopentyl-N-{[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}acetamide
(3R,4R)-4-amino-1-[2-amino-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-3-ol
N,N-dimethyl-3-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-4'-ylmethyl}-1,2,4-oxadiazole-5-carboxamide
3-{[1-(4-methylpiperidine-4-carbonyl)pyrrolidin-3-yl]methyl}benzamide
ethyl 1-(2,3-dihydroxypropyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-3-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}benzamide
2-(2-methylpropyl)-8-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-(quinolin-4-ylmethyl)piperidin-3-amine
3,5,7-trimethyl-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-1H-indole-2-carboxamide
4-benzyl-3-{1-[6-(dimethylamino)pyrazin-2-yl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(azepan-1-yl)-3-[2-methoxy-4-({[(2-methylphenyl)methyl]amino}methyl)phenoxy]propan-2-ol
4-(3-methylphenoxy)-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidine
3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-8-methoxy-2-(2-methylpyrimidin-5-yl)quinoline
7-[(3-methoxyphenyl)methyl]-2-[(5-methylfuran-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
3-(3-chlorophenyl)-1-[4-(methoxymethyl)piperidin-1-yl]-3-phenylpropan-1-one
1-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
1-(2-methyl-1,3-thiazole-4-carbonyl)-4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidine
N-[1-(4-methyl-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]furan-2-carboxamide
1-[(5-chloro-2,3-dimethoxyphenyl)methyl]-4-(1,2,4-oxadiazol-3-yl)piperidine
6-[4-(cyclopropylmethyl)-5-oxo-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-methyl-2-{1-[3-(4-methyl-1H-pyrazol-1-yl)propyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
3-(4-{5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]pyridin-2-yl}phenyl)propanoic acid
N-[1-(2,5-difluorophenyl)cyclopropyl]-2-methylimidazo[1,2-a]pyridine-6-carboxamide
{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}[(1-phenyl-1H-pyrazol-4-yl)methyl]amine