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1-[1-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-4-yl]-1,4-diazepan-5-one
N-(2,2-difluoroethyl)-6-(4-fluorophenyl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
8-butyl-N-[(3-fluorophenyl)methyl]-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
1-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}-4-(pyridin-4-yl)piperazine
1-[4-(1,3-benzoxazol-2-yl)piperazin-1-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one
N-[(3R,4S)-1-[(2-aminopyrimidin-5-yl)methyl]-4-cyclopropylpyrrolidin-3-yl]oxane-4-carboxamide
2-{[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)methyl]amino}-N-(1,3-thiazol-2-yl)propanamide
3-{8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-5-phenyl-1,2-oxazole
3-(1H-1,3-benzodiazol-2-ylmethyl)-N-(6-cyanopyridin-3-yl)piperidine-1-carboxamide
4-phenyl-3-[2-(trifluoromethyl)morpholine-4-carbonyl]-1H-pyrazol-5-amine
9-[2-(2-methoxyethoxy)acetyl]-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
(1S,5R)-3-[2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)acetyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[2-(1H-pyrazol-1-yl)ethyl]benzamide
methyl 2-(1-{5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]phenyl}-N-methylformamido)acetate
N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-cyclopropyl-N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N-methyl-1,3,4-oxadiazol-2-amine
1-(3-chloro-4-methoxyphenyl)-5-oxo-N-[2-(propylsulfanyl)ethyl]pyrrolidine-3-carboxamide
(3R,9aR)-8-(4-chlorobenzenesulfonyl)-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
methyl (2S,4R)-1-[(3-methylphenyl)methyl]-4-[4-(trifluoromethyl)benzamido]pyrrolidine-2-carboxylate
(2E)-3-(1-methyl-1H-pyrazol-4-yl)-1-[3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]prop-2-en-1-one
2-(methylsulfanyl)-1-[2-(2-phenylethyl)morpholin-4-yl]ethan-1-one
N-[2-(4-chlorobenzenesulfonamido)ethyl]-6-oxo-1-propylpiperidine-3-carboxamide
2-ethyl-6-(3-fluoro-2-methoxybenzoyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-6-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
5-chloro-N-[2-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)ethyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
1-(2-carbamoylethyl)-N-[3-(1H-indol-2-yl)phenyl]piperidine-4-carboxamide
(1R,2R,6S,7S)-4-(7-fluoroquinazolin-4-yl)-4-azatricyclo[5.2.1.02,6]decane
2-{1-[(6-methylpyridin-2-yl)methyl]-4-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
2-(4-acetylphenoxy)-1-[3-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]ethan-1-one
1-[2-(2-chlorophenyl)ethyl]-2-(methoxymethyl)-6-methyl-4-oxo-N-(thiophen-3-ylmethyl)-1,4-dihydropyridine-3-carboxamide
5-({ethyl[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-N-(propan-2-yl)pyrimidin-2-amine
6-{1-[(4-methoxyphenyl)methyl]-1H-pyrazol-4-yl}pyridine-3-carboxylic acid
N-{2-[1-(9-methyl-1-oxo-2,3,4,9-tetrahydro-1H-carbazol-6-yl)-1H-imidazol-4-yl]ethyl}acetamide
2-{3,5-dimethyl-4-[3-(trifluoromethyl)benzenesulfonamido]-1H-pyrazol-1-yl}acetic acid
(2S)-2-amino-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-phenylpropanamide
4-(4-chlorophenyl)-N-[2-(methylsulfamoyl)ethyl]butanamide
2-(1-methyl-6-oxo-1,6-dihydropyridazine-3-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
2-{4-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
5-{[4-(1,5-dimethyl-1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-2-hydroxybenzoic acid
N-({4-[4-(benzenesulfonyl)phenyl]phenyl}methyl)acetamide
(1S,3R)-N-(2-ethylbutyl)-3-[2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamido]cyclopentane-1-carboxamide
1-cyclohexyl-N3-ethyl-N5-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
4-(5-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl)morpholine
(2S,4S)-4-amino-1-methyl-N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]pyrrolidine-2-carboxamide
N-[(1-ethyl-5-oxopyrrolidin-3-yl)methyl]-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
3-[(furan-2-ylmethyl)sulfamoyl]-5-(pyridin-3-yl)benzoic acid
1-methyl-N-(3-phenylpropyl)-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-hydroxy-1,2-dimethyl-N-[2-(morpholin-4-yl)ethyl]-1H-indole-3-carboxamide
1-(2,2-dimethyloxane-4-carbonyl)-4-{2-[2-(3-methoxyphenyl)ethyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidine
1-(3-chloro-4-fluorophenyl)-5-[2-(1H-pyrazol-1-yl)ethyl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole