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4-chloro-N-ethyl-1-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
2-(butan-2-ylsulfanyl)-5-{[4-(1H-pyrrole-2-carbonyl)piperazin-1-yl]methyl}pyrimidine
N-ethyl-N-(2,2,2-trifluoroethyl)imidazo[1,2-a]pyrimidine-2-carboxamide
8-(2,3-difluoro-4-pentylphenyl)-3,7-dimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-dione
5-cyclobutanecarbonyl-1'-(pyrazin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
methyl 7-oxo-3-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-9-[2-(pyridin-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-methyl-N-[(3-methylpyridin-4-yl)methyl]-5-phenyl-1H-pyrrole-2-carboxamide
N-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-2-methoxy-N-(oxolan-2-ylmethyl)acetamide
benzyl({[2-cyclohexylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl})methylamine
2-[(4-fluorophenyl)methyl]-4-(piperidin-4-ylmethyl)morpholine
2-[(3-methoxyphenyl)methyl]-8-(morpholine-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
N-(1-{7-[(2,4-dimethoxy-3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-methylpropanamide
N-(1-{7-[(4-acetamidophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-phenylpropanamide
3-chloro-5-[4-(2-methylpyrimidin-4-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
N-(3-aminopropyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-methyl-8-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-cyclopentyl-4-[2-(morpholin-4-yl)pyrimidine-5-carbonyl]-1,4-diazepane
2-[4-methoxy-3-(methoxymethyl)benzoyl]-8-methyl-2,8-diazaspiro[4.5]decane
3-chloro-5-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
N5-cyclopentyl-N6-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
N-(5-chloro-2-methoxyphenyl)-3-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-3-yl}propanamide
N-[(5-ethylpyridin-2-yl)methyl]-4-hydroxy-N-methyl-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
2-butyl-8-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(5-chloro-2-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
6-methyl-1-{3-oxo-3-[4-(thian-4-yl)piperazin-1-yl]propyl}-1,2-dihydropyridin-2-one
N-[2-(2-chloro-4-methylphenoxy)ethyl]-5-ethoxy-N-methylfuran-2-carboxamide
1-(2-methylpropyl)-N-[(4-phenyloxan-4-yl)methyl]-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-{2-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]-2-oxoethyl}methanesulfonamide
(3S,5S)-5-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-1-methylpyrrolidin-3-amine
1-[1-(3,6-dimethylpyrazin-2-yl)piperidin-4-yl]-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
1-(naphthalen-2-yl)-3-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]urea
5-methoxy-3-methyl-N-[2-(2-methylpropanesulfonyl)ethyl]-1H-indole-2-carboxamide
2-(4-benzyl-2-oxopyrrolidin-1-yl)-N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}[(5-methylpyrazin-2-yl)methyl]amine
1-[1-(3-aminopropyl)-1H-1,2,3-triazole-4-carbonyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
6-(2-chlorophenyl)-7-methyl-8-oxo-N-[2-(1,3-thiazol-2-yl)ethyl]-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
9-(furan-2-carbonyl)-1-methyl-4-[(3-methylthiophen-2-yl)methyl]-1,4,9-triazaspiro[5.5]undecane
2-{[3-benzyl-3-(hydroxymethyl)piperidin-1-yl]methyl}-4-chlorophenol
2-(2,5-dimethylphenyl)-2-{methyl[4-(morpholin-4-yl)butyl]amino}acetic acid
8-[(4-methoxyphenyl)methyl]-1-methyl-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3R,4R)-1-[2-(dimethylamino)pyridine-3-carbonyl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
(5-{[3-(4-chlorobenzoyl)piperidin-1-yl]methyl}-2-ethoxyphenyl)methanol
(5R)-5-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]pyrrolidin-2-one
N4-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-6-methyl-5-(prop-2-en-1-yl)pyrimidine-2,4-diamine
1-(4-{[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
N-[(5-carbamoyl-1,2,4-oxadiazol-3-yl)methyl]-1-(cyclohexylmethyl)-6-oxopiperidine-3-carboxamide
5-fluoro-6-methyl-2-[2-(thiomorpholin-4-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
(3R,4S)-1-{[1-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-3,4-dimethylpiperidin-4-ol
1-(2-propyl-1,3-thiazole-4-carbonyl)-4-(4H-1,2,4-triazol-4-yl)piperidine
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]propanamide