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4-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}-1-(oxan-4-ylmethyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
N-benzyl-3-(2-{[(3,4-difluorophenyl)methyl]carbamoyl}ethyl)piperidine-1-carboxamide
N-(1-{1-[(2,5-dimethylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopentanecarboxamide
4-methyl-2-(propan-2-yl)-5-{3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}pyrimidine
2-methyl-4-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyrimidine
3-[9-oxo-8-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-2-yl]propanoic acid
2-(2-fluorophenoxymethyl)-N-[2-(1-hydroxycyclopentyl)ethyl]-N-methyl-1,3-oxazole-4-carboxamide
1-[4-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
N-methyl-2-(2-methyl-1,3-thiazol-4-yl)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]acetamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-methyl-1,5-diazatricyclo[5.2.2.02,6]undecane
5-fluoro-3-methyl-2-({4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}methyl)-1H-indole
5-methyl-5-phenyl-1-(piperidin-4-ylmethyl)piperidin-2-one
N-(3,3-diphenylpropyl)-6-[2-(thiophen-2-yl)acetyl]-6-azaspiro[2.5]octane-1-carboxamide
1-[(3-methylphenyl)methyl]-4-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
1-(4-fluorophenyl)-4-{4-methyl-3-oxo-1-oxa-4,9-diazaspiro[5.5]undecan-9-yl}butane-1,4-dione
1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine
1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-3-{3-methyl-3H-imidazo[4,5-b]pyridin-2-yl}propan-1-one
3-[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)propanamide
N-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-6-methoxy-1,3-benzothiazol-2-amine
N,N-bis(2-methoxyethyl)-5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
N3-cyclohexyl-1-cyclopropyl-N5-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
(1R,2S,9R)-11-(4-methoxypyrimidin-2-yl)-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
3-[5-({4-oxo-3H,4H-thieno[3,2-d]pyrimidin-2-yl}methyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
N,8-dimethyl-N-(2-phenylethyl)-3-(pyrrolidin-1-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
(1S,6R)-9-[(1-ethyl-1H-indol-4-yl)methyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
(4aR,7aS)-N,N-dimethyl-4-[3-(4-methyl-1H-pyrazol-1-yl)propanoyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
2-(dimethylamino)-2-(3-methylphenyl)-N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}acetamide
5-(4-acetyl-2-methoxyphenoxymethyl)-N-[2-(pyrrolidin-1-yl)ethyl]-1,2-oxazole-3-carboxamide
(4aS,7aR)-4-ethyl-N-(5-fluoro-2-methylphenyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N-[2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]-2-(phenylamino)pyrimidine-5-carboxamide
4,4,4-trifluoro-1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]butan-1-one
1-(5-methoxy-2-{[(2-phenylethyl)amino]methyl}phenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-ethylpiperidine-3-carboxamide
6-(1-methyl-1H-imidazol-2-yl)-N-[4-(1H-pyrazol-1-yl)butan-2-yl]pyridazin-3-amine
2-{1-[(2-ethoxyphenyl)methyl]-4-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperazin-2-yl}ethan-1-ol
N-cyclopropyl-4-methoxy-3-({[(5-oxopyrrolidin-2-yl)methyl](propan-2-yl)carbamoyl}amino)benzamide
4-(3-hydroxy-3-methylbutyl)-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}benzamide
3-(3,5-difluorophenyl)-5-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-[(2-fluorophenyl)methyl]-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]-1H-1,2,3-triazole-4-carboxamide
3-(4-chloro-1H-pyrazol-1-yl)-1-[4-(quinazolin-4-yl)piperazin-1-yl]propan-1-one
5-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-methyl-3-[2-methyl-4-(4-methylphenyl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
N-cyclopropyl-1-{1-[1-(2-methoxyphenyl)piperidin-4-yl]piperidin-4-yl}piperidine-4-carboxamide
methyl 2-(piperidine-1-sulfonyl)-6-(4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[5,8-dimethoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-3-(3-methyl-1H-pyrazol-1-yl)propanamide
N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-6-methyl-2-(pyridin-3-yl)pyrimidin-4-amine
(4aR,7aS)-1-cyclobutanecarbonyl-4-(5-methyl-1,2-oxazole-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3,4-dimethoxy-N-(2-{4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)benzamide
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-(3-methoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonane
N,2,3-trimethyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}quinoxaline-6-carboxamide