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4-{4-[(4-chloro-3-fluorophenyl)methyl]piperazin-1-yl}-5,6-dimethylpyrimidine
4-hydroxy-2-[({2-[4-(propan-2-yl)-1,3-thiazol-2-yl]ethyl}amino)methyl]quinoline-6-carboxamide
5-(1H-1,3-benzodiazol-1-yl)-3-methylpyridin-2-amine
(1R,3s,6r,8S)-4-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-azatricyclo[4.3.1.13,8]undecane
6-methyl-N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)pyridine-2-carboxamide
2-amino-6-(2H-1,3-benzodioxol-5-yl)-4-(piperidin-4-yl)pyridine-3-carbonitrile
N-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-4-acetamido-N-(oxolan-2-ylmethyl)benzamide
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N-methyl-2-(1-oxo-1,2-dihydroisoquinolin-2-yl)acetamide
1-[1'-(furan-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
3-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}benzoic acid
3-benzoyl-1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}piperidine
1,3-dimethyl-N-[1-(1H-pyrazol-1-yl)propan-2-yl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-[(3S,4R)-4-(4-methylphenyl)-1-[3-(2-oxopiperidin-1-yl)propanoyl]pyrrolidin-3-yl]acetamide
(1R,5R)-3-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
4-cyclopentyl-2-[(4-fluorophenyl)methyl]morpholine
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]({[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl})amine
N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]-1H-imidazole-4-carboxamide
2-[(4aR,7aS)-4-[(2,5-difluorophenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
2-[2-({[(1-methylpiperidin-4-yl)methyl](2-phenylethyl)amino}methyl)phenoxy]ethan-1-ol
{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[4-(trifluoromethyl)phenyl]methyl}amine
6-(2-chlorophenyl)-7-methyl-N-(3-methylbutan-2-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-[(2S)-3-(1H-imidazol-4-yl)-1-oxo-1-[3-oxo-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-9-yl]propan-2-yl]acetamide
{2-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}urea
1-[(2-hydroxy-5-phenylphenyl)methyl]piperidin-3-ol
(3aR,6aR)-2-cyclopropanecarbonyl-N-(prop-2-en-1-yl)-N-(pyridin-2-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-tert-butyl-5-[1-(4-chloro-1H-pyrazol-1-yl)ethyl]-3-methyl-1H-1,2,4-triazole
1-cyclohexyl-4-[2-(1H-indazol-1-yl)acetyl]-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
1-[(4-chlorophenyl)methyl]-5-{2-[(prop-2-en-1-yl)amino]ethyl}pyrrolidin-2-one
dimethyl({5-[1-(thiophen-3-ylmethyl)-1H-imidazol-2-yl]thiophen-3-yl}methyl)amine
N-[(4-fluorophenyl)methyl]-3-{1-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]piperidin-4-yl}propanamide
(1S,5R)-6-(furan-3-ylmethyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
1-[3-(5-methylfuran-2-yl)butyl]-4-[2-(piperidine-1-carbonyl)phenoxy]piperidine
N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(thiomorpholine-4-sulfonyl)benzamide
1-[(4-chloro-3-fluorophenyl)methyl]-3-(pyrrolidin-1-yl)piperidine
4-[(5-ethylfuran-2-yl)methyl]-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[(3R,4S)-3-amino-4-(3-methoxyphenyl)pyrrolidin-1-yl]-2-(2,2,3,3-tetrafluoropropoxy)ethan-1-one
[9-(3-chloropyridin-2-yl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol
N-benzyl{[4-(1H-1,2,3,4-tetrazol-5-yloxy)phenyl]amino}sulfonamide
N-{2-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-2-oxoethyl}-2-methylpropanamide
methyl 2-(4-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-2-yl)acetate
3-{5-[(4-methoxypyridin-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-(propan-2-yl)propanamide
3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}-N-[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]propanamide
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamide
ethyl 4-[(4-chlorophenyl)methyl]-1-(1,4-dithiepan-6-yl)piperidine-4-carboxylate
N-{4-[({1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}amino)methyl]phenyl}acetamide
2-{4-[(3,5-dimethylphenyl)methyl]-1-(1-methylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]azepan-4-amine
4-[1-(3,4,5-trimethoxyphenyl)-1H-imidazol-2-yl]quinoline
(1,4-dioxan-2-ylmethyl)(methyl){[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine