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6-chloro-2-(2,4-dimethoxyphenyl)quinoline
1-tert-butyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-1H-pyrrole-3-carboxamide
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-[2-(1H-pyrazol-1-yl)benzoyl]piperidine
1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
2-{[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]({[4-(methylsulfanyl)phenyl]methyl})amino}ethan-1-ol
2-[2-({4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)-1H-pyrrol-1-yl]pyridine
1-benzyl-6-(pyridin-2-ylmethoxy)-4-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)-1,4-diazepan-2-one
N-[(2R,3R)-1'-(3-chloro-2-fluorobenzoyl)-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
(3R,4R)-4-ethyl-1-[3-(pyrrolidin-1-yl)pyrazin-2-yl]piperidine-3,4-diol
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-6-fluoro-N-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
(1H-imidazol-2-ylmethyl)(pyridin-3-ylmethyl)(thiophen-3-ylmethyl)amine
1-{6-chloroimidazo[1,2-a]pyrimidine-2-carbonyl}-2-(furan-2-yl)azepane
2-cyclopropyl-4-hydroxy-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]pyrimidine-5-carboxamide
1-{2-[cyclohexyl(methyl)amino]pyridine-3-carbonyl}-3-(hydroxymethyl)piperidin-3-ol
2-methyl-4-(pyrrolidin-1-yl)-6-{1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]piperidin-3-yl}pyrimidine
2-(3-methoxyphenyl)-1-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)azetidine
({3-methyl-1-[2-(thiomorpholin-4-yl)ethyl]-1H-pyrazol-4-yl}methyl)[(5-methylpyrazin-2-yl)methyl]amine
2-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}phenol
4-ethyl-1-methyl-3-{[1-(quinoline-5-carbonyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-methyl-2-({3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}methyl)pyridine
1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-4-(piperidin-1-yl)piperidine
2-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]-1-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]ethan-1-one
4-[1-(2H-1,3-benzodioxol-5-ylmethyl)-1H-1,2,4-triazol-5-yl]-2-ethylpyridine
6-(methoxymethyl)-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]pyrimidin-4-amine
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]amine
1-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-2-(1-propylpiperidin-4-yl)ethan-1-one
3-(2H-1,3-benzodioxol-5-yl)-1-{4-[2-(methoxymethyl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}propan-1-one
3-(1H-1,3-benzodiazol-1-yl)-N-(oxolan-3-yl)propanamide
1-[2-(dimethylamino)-4-[methyl(oxolan-2-ylmethyl)amino]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
N-[1-(4-fluorophenyl)piperidin-4-yl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1-(morpholin-4-yl)cyclohexane-1-carboxamide
1-(2-methoxyethyl)-3-(3-methoxyphenyl)-3-{2-[(2S,6S)-4-methyl-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
2-methyl-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}imidazo[1,2-a]pyrimidine-3-carboxamide
N-cyclopropyl-2-{6-hydroxy-4-[2-(1H-pyrazol-4-yl)ethyl]-1,4-diazepan-1-yl}acetamide
{[2-(2,2-dimethylpropanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(ethyl)(pyridin-4-ylmethyl)amine
[5-(1-{[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-1H-imidazol-2-yl)furan-2-yl]methanol
N,N-dimethyl-3-(1-{5-[(methylsulfanyl)methyl]pyridin-2-yl}piperidin-3-yl)propanamide
3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
1-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
N-[2-(1-methylpiperidin-2-yl)ethyl]-6-(piperazin-1-yl)pyridine-3-carboxamide
N-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-3-(1-methyl-1H-pyrazol-4-yl)propanamide
N-(cyclopropylmethyl)-4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
3-(1-benzyl-3-phenyl-1H-1,2,4-triazol-5-yl)-1λ6-thiane-1,1-dione
1-{4-[2-(morpholin-3-yl)acetyl]piperazin-1-yl}-2-phenoxyethan-1-one
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-6-(pyridin-4-yl)pyridine-3-carboxamide
dimethyl(2-{2-[1-(3-methylpyridin-4-yl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-(methylsulfanyl)benzamide
methyl 5-[(1-cyclohexylethyl)amino]-3-(furan-2-amido)-1-(2-methoxyethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N,N-dimethyl-4-[4-({[1-(2-phenylethyl)piperidin-3-yl]methyl}amino)piperidin-1-yl]benzamide
4-(2-ethoxybenzoyl)-1-(4-methylphenyl)piperazin-2-one