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8-[2-methyl-5-(2-methyl-1,3-oxazol-5-yl)benzenesulfonyl]-1-oxa-8-azaspiro[4.5]decane
1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-methyl-N-[2-(4-methylphenoxy)ethyl]piperidin-4-amine
cyclopentyl 4-({methyl[(2-methylpyridin-4-yl)methyl]carbamoyl}amino)benzoate
2-({[1-(1-benzofuran-2-ylmethyl)piperidin-3-yl]oxy}methyl)pyridine
N-cyclopropyl-3-{5-[(2-methyl-1,3-thiazol-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
N-(4-{4-[3-(methoxymethyl)piperidin-1-yl]piperidin-1-yl}phenyl)-2,4-dimethylbenzamide
4-({2-[2-(dimethylamino)ethoxy]phenyl}methyl)-N,N-dimethylpiperazine-1-carboxamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-{[(4-phenylphenyl)methyl]amino}-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
2-[(3S,4R)-4-amino-1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl]ethan-1-ol
3-(3-methylphenyl)-N-[4-(2-oxopyrrolidin-1-yl)phenyl]piperidine-1-carboxamide
[(5-{[2-(2-methoxyphenyl)pyrimidin-5-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]dimethylamine
N-{2-methoxy-5-[4-(1H-1,2,4-triazol-1-yl)butanamido]phenyl}furan-2-carboxamide
2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)-7-(3-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-ethyl-3-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]-1-[2-(1H-pyrazol-1-yl)ethyl]urea
1-[2-(furan-2-yl)pyrrolidin-1-yl]-3-[4-(3-methylphenyl)piperazin-1-yl]propan-1-one
ethyl 2-{N-methyl-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propanamido}acetate
4-(2H-1,3-benzodioxole-5-carbonyl)-1-(2-methylpropyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
1-benzyl-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-phenylpiperidine-4-carboxamide
(3S,4S)-3-({[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}(methyl)amino)-4-hydroxy-1λ6-thiolane-1,1-dione
3-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-N-methylpropanamide
(1H-imidazol-2-ylmethyl)(methyl)({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)amine
6-(1,4-oxazepan-4-yl)-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
2-methyl-N-{2-[2-(trifluoromethyl)phenyl]ethyl}-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
methyl 4-({4-[2-oxo-2-(piperidin-1-yl)ethyl]piperazin-1-yl}methyl)thiophene-2-carboxylate
N-(2,2-diphenylethyl)-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]acetamide
4-(4-fluorophenyl)-1-[4-(pyridin-3-yl)pyrimidin-2-yl]piperidin-4-ol
N-[2-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)ethyl]-1H-1,3-benzodiazole-2-carboxamide
4,6-dimethyl-N-[1-(4-methylpyridin-2-yl)propyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
2-methoxy-N-{1-[4-(4-methyl-3-phenylpiperazine-1-carbonyl)phenyl]-1H-pyrazol-4-yl}acetamide
(3aR,6aR)-2-(ethylcarbamoyl)-5-(6-methylpyridazin-3-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[(dimethylamino)methyl]-4-{1-[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]-1H-imidazol-2-yl}phenol
7-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-4-(thiophene-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}-3-[3-(propan-2-yloxy)benzoyl]piperidine
2-(dimethylamino)-1-[(1R,3R,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octan-8-yl]ethan-1-one
2-{[4-(2-hydroxyethyl)piperazin-1-yl]sulfonyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]-2-[2-(thiophen-2-yl)ethyl]piperidine
2-{5-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carbonyl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
(1-{[4-(furan-2-yl)phenyl]methyl}-4-(2-phenoxyethyl)piperidin-4-yl)methanol
1-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-[2-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazole
3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}propanamide
2-(dimethylamino)-N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}acetamide
N-benzyl-N-methyl-2-(1H-pyrrole-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
7-methyl-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-2,3-dihydro-1,4-benzodioxine-6-carboxamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-1-[(3R,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]ethan-1-one
(2R,3S,6R)-5-(cyclopropanesulfonyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(2S,4S)-1-benzyl-N-(2-methoxyethyl)-4-[(1-propylpiperidin-4-yl)amino]pyrrolidine-2-carboxamide
1-(benzenesulfonyl)-3-[4-(methylsulfanyl)benzoyl]piperidine
1-[7-(3-chlorophenyl)-9-(thiophen-3-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methylpropan-1-one
4-[5-(5-methyl-1-propyl-1H-pyrazol-4-yl)-1,2,4-oxadiazol-3-yl]pyridine