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2-{2-[(4-cyclopentyl-1,4-diazepan-1-yl)methyl]phenyl}-6-(methoxymethyl)-3,4-dihydropyrimidin-4-one
4-[9-oxo-8-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecane-2-carbonyl]benzonitrile
5-ethyl-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-(1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
(3S,9aR)-3-ethyl-8-(naphthalene-1-sulfonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(2-chlorobenzoyl)-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]piperidine
ethyl 4-(2-methoxyethyl)-1-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}piperidine-4-carboxylate
5-ethyl-2,3-dimethyl-7-{3-methyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}pyrazolo[1,5-a]pyrimidine
N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]acetamide
N-{1-[1-(2,3-dihydroxypropyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopentanecarboxamide
N-(1-methyl-1H-pyrazol-4-yl)-2-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}acetamide
(1R,5R)-3-[(2,5-dimethylthiophen-3-yl)sulfonyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
N-[3-(2,6-dimethylphenoxy)propyl]-N-methyl-2-{1-oxo-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-2-yl}acetamide
2-(4-hydroxyhepta-1,6-dien-4-yl)-7-(3-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
5-(4-fluoro-2-methoxyphenyl)-1-phenyl-1H,4H-pyrazolo[3,4-d]imidazole
2-(3-{3-oxa-9-azaspiro[5.5]undecane-9-carbonyl}pyrazolo[1,5-a]pyrimidin-6-yl)ethan-1-ol
4-[1-(1-benzoylpiperidin-4-yl)piperidine-3-carbonyl]morpholine
ethyl 4-(2-methoxyethyl)-1-{[5-(oxan-2-yl)thiophen-2-yl]methyl}piperidine-4-carboxylate
3-[2-(3-benzoylpiperidin-1-yl)-2-oxoethyl]-5,5-dimethylimidazolidine-2,4-dione
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-4-methylpyrimidine-5-carboxamide
4-[4-(propan-2-yloxy)phenyl]pyrimidine
(4aS,7aR)-1-[3-(2-hydroxyphenyl)-1H-pyrazole-5-carbonyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[3-(1H-imidazol-1-yl)propyl]-2-(propan-2-yl)pyrimidine-5-carboxamide
5-[4-(cyclopropylmethyl)piperazin-1-yl]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-(pyridin-2-ylmethyl)-4-[6-(pyrrolidin-1-yl)pyridazin-3-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
3-[methyl({6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl})amino]propane-1,2-diol
4-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-3,4-dihydro-2H-1,4-benzothiazin-3-one
2-[(4-methoxyphenyl)methyl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)-1,3-benzoxazole-6-carboxamide
N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
4-[2-(4-methylphenoxy)acetyl]-1-phenylpiperazin-2-one
ethyl 1-[5-(benzylcarbamoyl)-1-cyclopropyl-4-oxo-1,4-dihydropyridine-3-carbonyl]piperidine-2-carboxylate
N-benzyl-5-({[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)amino}methyl)pyrimidin-2-amine
4,4-difluoro-1-{[5-(thiophene-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}piperidine
N-benzyl-N-methyl-1-[3-(pyridin-4-yl)propanoyl]piperidine-4-carboxamide
[(1-ethyl-1H-imidazol-2-yl)methyl](methyl){[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
N-(2-fluorophenyl)-3-({[2-(1H-imidazol-2-yl)ethyl]carbamoyl}methyl)morpholine-4-carboxamide
5-fluoro-2-[1-(1H-pyrrole-3-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
(1R,2S,6R,7S)-4-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-4-azatricyclo[5.2.2.02,6]undecane
N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-2-(trimethyl-1H-pyrazol-1-yl)acetamide
1-methyl-N,N-bis(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{[3-(2,6-dichlorophenyl)-5-methyl-1,2-oxazol-4-yl]methyl}-3-methoxy-1,2-dihydropyridin-2-one
1-(4-fluorophenyl)-4-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]butane-1,4-dione
7-(furan-3-carbonyl)-2-methyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-(2-methoxyphenyl)-4-(5-methyl-1H-indole-2-carbonyl)piperazin-2-one
3-{[(2S,5R)-2,5-dimethylpiperazin-1-yl]methyl}-N-(2-oxo-2,3-dihydro-1H-indol-5-yl)benzamide
5-(pyrrolidin-1-yl)-2-(3,3,4,4-tetrafluorobutyl)-2,3-dihydropyridazin-3-one
N-[(5-methyl-1,2-oxazol-3-yl)methyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-(3-methyl-1,2,4-thiadiazol-5-yl)-1-[(2-phenyl-1,3-thiazol-4-yl)methyl]urea
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)-1H-pyrazole-3-carboxamide
2-methoxyethyl 2-[(5-methylpyrazin-2-yl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxylate
2-(2-ethenylphenyl)pyridine-4-carboxamide