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1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]propan-1-one
9-[5,6-dimethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
(4aS,8aS)-2-[2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]-decahydroisoquinoline
4-(1-ethylpiperidine-4-carbonyl)-2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}morpholine
2-{1-[(3,4-difluorophenyl)methyl]-4-(3-phenylprop-2-yn-1-yl)piperazin-2-yl}ethan-1-ol
4-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]-4-oxobutane-1-sulfonamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
N-({4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-3-(4-methylphenyl)propanamide
1-benzyl-4-[4-(hydroxymethyl)-1,3-thiazol-2-yl]-1,4-diazepan-6-ol
2-methyl-5-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]pyrazine
N-[1-(cyclohexylmethyl)piperidin-3-yl]-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
2-[1-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-1H-imidazol-2-yl]-4,5,6,7-tetrahydro-1,3-benzothiazole
1-(5-{3-[5-(2-chlorophenyl)pyrimidin-4-yl]piperidine-1-carbonyl}thiophen-2-yl)ethan-1-one
4-[2-(7-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propyl]phenol
(3S,4S)-4-[(2-hydroxyethyl)(methyl)amino]-1-{5-[(phenylsulfanyl)methyl]furan-2-carbonyl}pyrrolidin-3-ol
3-[4-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)piperazin-1-yl]-1λ6-thiolane-1,1-dione
{[2-(4-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[(1-methyl-1H-pyrazol-4-yl)methyl](propan-2-yl)amine
7-{[4-(benzyloxy)piperidin-1-yl]methyl}-4-(2-methylpropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(3R,4S)-4-(propan-2-yl)-1-(propane-1-sulfonyl)pyrrolidin-3-yl]pyrimidin-2-amine
N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-(4H-1,2,4-triazol-4-yl)benzamide
4-hydroxy-N-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-2-[(phenylsulfanyl)methyl]pyrimidine-5-carboxamide
3-(5-methyl-1,3,4-thiadiazol-2-yl)-1-(piperidin-3-yl)urea
5-(methoxymethyl)-N-methyl-N-(pyridin-3-ylmethyl)-1,3,4-oxadiazole-2-carboxamide
(1-benzothiophen-2-ylmethyl)(methyl)[(4-{2-[4-(5-methylthiophene-2-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl]amine
1-{1-[(3-fluoro-2-methylphenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
2-{2-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
1-[cyclohexyl(methyl)amino]-3-(4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}-2-methoxyphenoxy)propan-2-ol
1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
3-{[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]methyl}pyridine
1'-[2-(1-ethylpiperidin-4-yl)acetyl]-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
3-chloro-4-({1-[(2-chlorophenyl)methyl]piperidin-4-yl}oxy)-N-[2-(dimethylamino)ethyl]benzamide
N-[(5-fluoro-2-methylphenyl)methyl]-3-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propanamide
2-amino-4-[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]-6-(furan-2-yl)pyridine-3-carbonitrile
5-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
(4aS,8aR)-N-(cyclohexylmethyl)-1-[2-(methylamino)ethyl]-2-oxo-decahydro-1,6-naphthyridine-6-carboxamide
3-ethyl-8-(2-oxo-6-phenyl-1,2-dihydropyridine-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[4-(2,8-dimethylquinoline-4-carbonyl)piperazin-1-yl]pyridine-3-carbonitrile
N-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]-5-(oxolan-2-yl)thiophene-2-carboxamide
N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-3-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
2-(4-chlorophenyl)-4-[6-(methoxymethyl)pyrimidin-4-yl]morpholine
1-[(2R,6S)-6-phenyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
[(1-cyclopentylpiperidin-4-yl)methyl]({[5-(methoxymethyl)furan-2-yl]methyl})(oxolan-2-ylmethyl)amine
1-{4-[(1-cyclopentylpiperidin-4-yl)oxy]-3-methoxybenzoyl}piperidin-3-ol
4-[4-(2-fluorophenyl)-5-methyl-1H-imidazol-2-yl]-1-(propan-2-yl)pyrrolidin-2-one
2-[(1-phenoxypropan-2-yl)amino]-N-(propan-2-yl)acetamide
N-({3-[(2-fluorophenyl)methoxy]-4-methoxyphenyl}methyl)-2,3-dimethyl-N-(pyridin-4-ylmethyl)-1H-indole-5-carboxamide
4-{4-[(benzylamino)methyl]-1H-1,2,3-triazol-1-yl}-N-tert-butylpiperidine-1-carboxamide
(3S,4S)-3-hydroxy-4-[({4-methoxy-3-[(4-methylphenyl)methoxy]phenyl}methyl)amino]-1λ6-thiolane-1,1-dione
ethyl 4-[(3-methoxyphenyl)methyl]-1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidine-4-carboxylate
1-(2-{1-[2-(3-methylphenyl)benzoyl]piperidin-4-yl}ethyl)pyrrolidin-2-one