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2-(4-fluorophenyl)-1-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine
3-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-methyl-N-{3-[methyl(phenyl)amino]propyl}pyrazolo[1,5-a]pyrimidin-7-amine
N-methyl-2-(3-phenylpyrrolidin-1-yl)-N-(1,3-thiazol-2-ylmethyl)acetamide
3-[3-(2-methylphenoxy)azetidine-1-carbonyl]phenol
3-[(2-fluorophenyl)formamido]-N-[2-(2-hydroxyethoxy)ethyl]propanamide
2-amino-3-ethyl-N-[4-(pyridin-2-yl)butyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
4-[3-(morpholin-4-ylmethyl)piperidin-1-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
4-methyl-6-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyrimidine
(1S,5R)-6-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2,3,5-trimethyl-N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)pyrazolo[1,5-a]pyrimidin-7-amine
N-[4-(2-fluorophenoxy)phenyl]-1-(1-methyl-1H-pyrazole-5-carbonyl)piperidine-4-carboxamide
1-(4-{2-[(2S)-2-(hydroxymethyl)pyrrolidine-1-carbonyl]phenoxy}piperidin-1-yl)-2-methoxyethan-1-one
6-{1-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]piperidin-4-yl}-2-methylpyrimidin-4-ol
ethyl 1-(1H-1,3-benzodiazol-2-ylmethyl)-4-[(3-fluorophenyl)methyl]piperidine-4-carboxylate
[(3R,4R)-4-(morpholin-4-ylmethyl)-1-[2-(trifluoromethyl)benzoyl]pyrrolidin-3-yl]methanol
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(2,6-dimethylpyrimidine-4-carbonyl)pyrrolidin-3-yl]methanol
(1S,9aR)-1-{[4-(3-chloropyridin-2-yl)piperazin-1-yl]methyl}-octahydro-1H-quinolizine
2-methyl-8-{[5-(1,3-oxazol-5-yl)thiophen-2-yl]sulfonyl}-2,8-diazaspiro[4.5]decane
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)cyclopentanecarboxamide
3-[4-(benzyloxy)piperidine-1-carbonyl]-6-(propan-2-yl)-1,2-dihydropyridin-2-one
methyl 4-[5-(acetamidomethyl)-1,2,4-oxadiazol-3-yl]benzoate
1-[2-(1-butyl-1H-1,2,4-triazol-5-yl)ethyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-butyl-4-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-1-methylpiperazin-2-one
N-benzyl-N-(cyclobutylmethyl)-2-(hydroxymethyl)-1H-1,3-benzodiazole-5-carboxamide
4-(3-benzyl-1H-1,2,4-triazol-5-yl)-6-(2-methylpropyl)-1,2-dihydropyrimidin-2-one
1-[(3-chloro-4,5-dimethoxyphenyl)methyl]-4-(2-methoxyethoxy)piperidine
N-(2-ethoxyphenyl)-N'-(prop-2-en-1-yl)-N'-(pyridin-2-ylmethyl)propanediamide
2-[2-(azepan-1-ylmethyl)phenyl]-6-propyl-3,4-dihydropyrimidin-4-one
N-({3-[(3-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
1-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
1-(azepan-1-yl)-3-(2-methoxy-4-{[methyl(prop-2-en-1-yl)amino]methyl}phenoxy)propan-2-ol
2-cyclopentyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-2-phenylacetamide
7-(2-methoxyphenyl)-2-(thiophen-3-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-methoxy-3-[4-methoxy-2-(1H-pyrazol-1-yl)phenyl]pyrazine
(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-[2-(methylsulfanyl)pyridine-3-carbonyl]pyrrolidin-3-amine
(3R,4S)-N,N-dimethyl-1-[(2-methylpyrimidin-5-yl)methyl]-4-propylpyrrolidin-3-amine
4-[(4aS,8aR)-decahydroisoquinolin-2-yl]-N-(2-hydroxyethyl)pyridine-2-carboxamide
1-[3,5-difluoro-4-(trifluoromethyl)phenyl]-3-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]urea
4-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidine-1-carbonyl]-5,6,7,8-tetrahydroquinazolin-2-amine
2-hydroxy-2-methyl-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)propanamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(1,3-thiazol-4-ylmethyl)pyrrolidin-3-yl]-2-hydroxypyridine-3-carboxamide
N-({3-methoxy-4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)-2-methyl-N-[(3S)-2-oxoazepan-3-yl]propanamide
N-{2-[5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl]ethyl}-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
4-methyl-3-(2-oxoimidazolidin-1-yl)-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}benzamide
2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)benzamide
3-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
2-methyl-N-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)-1,3-thiazole-4-carboxamide
1-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]-2-(4-phenylpiperidin-1-yl)ethan-1-one
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(ethanesulfonyl)piperidine