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3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N,4-dimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-2-(propan-2-yl)pyrimidine-5-carboxamide
1-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine
5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-[(4-methyl-1H-imidazol-2-yl)methyl]benzamide
2-[(4-benzylpiperazin-1-yl)methyl]-N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-1,3-oxazole-4-carboxamide
N-{[(2R,3R,5S)-2-(2-fluorophenyl)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]methyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
3-(1-methyl-1H-pyrrol-2-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]-1H-pyrazole-5-carboxamide
3-(4-ethylphenyl)-N-(2-methanesulfonylethyl)-1H-pyrazole-5-carboxamide
1-(5-methyl-1,3-oxazole-4-carbonyl)-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-3-carboxamide
N-[1-(2-oxo-2-{spiro[indene-1,4'-piperidine]-1'-yl}ethyl)-1H-pyrazol-4-yl]-2-phenoxyacetamide
4-(2,4-dioxoimidazolidin-1-yl)-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]benzamide
(3R,4R)-1-{[2-(cyclopentyloxy)phenyl]methyl}-4-(morpholin-4-yl)piperidin-3-ol
1-benzyl-5-(2,6-dimethylpyrimidine-4-carbonyl)-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(oxan-4-ylmethyl)-2-[4-(trifluoromethyl)phenyl]-1H-imidazole
2-({[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]amino}methyl)-6-methylquinolin-4-ol
6-oxo-N-({4-[(3-phenylpropyl)amino]quinazolin-2-yl}methyl)-1,4,5,6-tetrahydropyridazine-3-carboxamide
4-ethyl-1-methyl-3-(1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)methylamine
3,5,7-trimethyl-N-[2-(methylsulfamoyl)ethyl]-1H-indole-2-carboxamide
(4aS,7aR)-1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)[2-(piperidin-1-yl)ethyl]amine
(1S,5R)-3-(4-methyl-1,3-thiazole-5-carbonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(5-methylthiophen-2-yl)methyl]piperidine
ethyl 4-(2-phenoxyethyl)-1-(thian-4-yl)piperidine-4-carboxylate
9-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]acetyl}-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
7-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-[2-(azepan-1-yl)-2-oxoethyl]-4-[(3,4-dimethoxyphenyl)methyl]piperazin-2-one
6-methyl-2-{[(oxolan-3-ylmethyl)amino]methyl}quinolin-4-ol
methyl 3-(4-methoxybenzamido)-1-methyl-5-(propylamino)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-({5-[(3,5-dimethylphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
1-[5-(methoxymethyl)pyrazolo[1,5-a]pyrimidin-7-yl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
5-(1-acetylpyrrolidin-2-yl)-N-(2H-1,3-benzodioxol-5-yl)thiophene-2-carboxamide
2-(2H-1,3-benzodioxol-4-yl)-1-methyl-1H-1,3-benzodiazole
4-cyclobutaneamido-N-[2-(2-fluorophenyl)ethyl]benzamide
3-[methyl(2-oxo-2-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethyl)amino]-1λ6-thiolane-1,1-dione
(1S,5R)-6-(2,3-difluoro-4-methylbenzoyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-[(1S,5R)-6-[(trimethyl-1H-pyrazol-4-yl)sulfonyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
(3S,7S,8aS)-3-[(benzyloxy)methyl]-7-{[(2-chlorophenyl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
3-(2-methoxyethyl)-1-(oxan-4-ylmethyl)piperidine-3-carboxylic acid
1-methyl-4-(6-methylpyrimidin-4-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
7-hydroxy-6-methyl-4-(6-phenoxypyridin-3-yl)-1,2,3,4-tetrahydroquinolin-2-one
4-({3-[(furan-2-ylmethyl)sulfanyl]propyl}carbamoyl)benzoic acid
3-(5-methylthiophen-2-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H-pyrazole-5-carboxamide
5-benzoyl-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-(2-{[(cyclohexylmethyl)amino]methyl}-5-methoxyphenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
(5-methyl-7-{5-methyl-6-[(2-methylpyridin-3-yl)oxy]pyrimidin-4-yl}-2,3-dihydro-1-benzofuran-2-yl)methanamine
6-methyl-2-{[(2-methylpropyl)(pyridin-2-ylmethyl)amino]methyl}pyridin-3-ol
2-methyl-N-(1-{[({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)carbamoyl]methyl}-1H-pyrazol-4-yl)furan-3-carboxamide
1-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-3,5-dimethyl-1H-1,2,4-triazole
5-[4-(cyclopropylmethyl)-5-oxo-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]pyridine-2-carbonitrile