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6,8-dimethyl-3-{[methyl({[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}-1,2-dihydroquinolin-2-one
4-[1-(2-methylpropyl)-5-oxopyrrolidine-3-carbonyl]-1-phenylpiperazin-2-one
1-[(1R,2R)-2-(benzyloxy)cyclopentyl]-4-(1,3-thiazol-2-yl)-1H-1,2,3-triazole
4-cyclobutyl-N,6-dimethyl-N-(pyridin-3-ylmethyl)pyrimidin-2-amine
1-butyl-3-(furan-2-yl)-5-[3-(1H-pyrazol-4-yl)propyl]-1H-1,2,4-triazole
2-amino-N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetamide
N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
ethyl 1-[(3S,4R)-4-ethoxyoxolan-3-yl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylate
[(2-ethyl-3-methyl-1H-indol-5-yl)methyl][(4-fluoro-3-methoxyphenyl)methyl]amine
4-(hydroxymethyl)-1-(7-methyl-2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidin-4-ol
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(2-fluorobenzoyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
7-[(3,4-difluorophenyl)methyl]-2-methanesulfonyl-2,7-diazaspiro[4.5]decan-6-one
2-(azocan-1-yl)-N-ethyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]acetamide
5-[3-(3-ethylphenoxy)azetidine-1-carbonyl]-2-(pyridin-3-yl)pyrimidine
4-(2-methoxyphenoxy)-1-(2-methyl-1,3-thiazole-4-carbonyl)piperidine
2-[7-(hydroxymethyl)-9-[2-(1H-imidazol-4-yl)acetyl]-3,9-diazaspiro[5.5]undecan-3-yl]acetamide
3-[2-({1-[4-(furan-2-yl)phenyl]piperidin-4-yl}amino)ethyl]-1,3-oxazinan-2-one
N-[3-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-3-[(methylsulfanyl)methyl]piperidine-1-carboxamide
1-[2-(6-{[2-(dimethylamino)ethyl]amino}-1H-pyrrolo[2,3-b]pyridin-4-yl)phenyl]ethan-1-one
(3S,9aR)-2-methyl-8-{[1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-{[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}azetidin-3-ol
5-[2-methoxy-5-(pyrrolidin-1-ylmethyl)phenoxy]isoquinoline
[(4aS,8aR)-6-[(2-phenyl-1,3-thiazol-5-yl)methyl]-decahydro-1,6-naphthyridin-4a-yl]methanol
1-{2-[methyl({[4-(methylsulfanyl)phenyl]methyl})amino]ethyl}piperidin-2-one
2-(5-acetylthiophen-3-yl)-1-[4-(3-methylpyridin-2-yl)piperazin-1-yl]ethan-1-one
6,7-dimethoxy-2-{1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-1,2,3,4-tetrahydroisoquinoline
(2R,6R)-4-(1-ethyl-1H-pyrazole-5-carbonyl)-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-ethyl-2-{4-[(2-ethylpyrimidin-4-yl)methyl]piperazin-1-yl}acetamide
1-(3-{2-[3-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}propyl)pyrrolidin-2-one
4-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}benzonitrile
3-[(methylsulfanyl)methyl]-N-[4-(pyridin-3-yloxy)phenyl]piperidine-1-carboxamide
N,N-dimethyl-3-[({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]benzamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-2-(pyrimidin-2-ylsulfanyl)acetamide
N-(cyclohexylmethyl)-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-[1-(3-phenylpropyl)piperidin-3-yl]-2-(pyridin-3-yl)acetamide
5-methyl-4-(1-methyl-1H-pyrazol-4-yl)-2-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-yl}pyrimidine
4-[4-(1,3-thiazol-2-yl)piperazin-1-yl]pyrimidine-5-carboxylic acid
(3S,4S)-1-{6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}-4-(naphthalen-2-yl)piperidin-3-ol
2-(1-benzofuran-2-yl)-4-{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]pyrrolidin-3-yl}pyridine
3-chloro-4-[(1-cyclobutylpiperidin-4-yl)oxy]-N-[2-(dimethylamino)ethyl]benzamide
3-(2-phenylpropyl)-8-[2-(propylsulfanyl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-methoxy-N-[3-methyl-1-(7-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)butyl]acetamide
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanamide
N-[(4-hydroxyphenyl)methyl]-3-(2-oxopiperidin-1-yl)-N-(pyridin-3-ylmethyl)propanamide
(2R)-1-{[2-(3,4-dimethoxyphenyl)-7-methylquinolin-3-yl]methyl}pyrrolidine-2-carboxamide
(2H-1,3-benzodioxol-5-ylmethyl)[(5-ethylpyridin-2-yl)methyl](pyridin-3-ylmethyl)amine
1-cyclopentyl-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-6-oxopiperidine-3-carboxamide
2-(1H-imidazole-4-carbonyl)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane
2-[3-(3-chloro-1H-1,2,4-triazol-5-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one