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2-chloro-4-{3-cyclopropyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}pyridine
2-[(2S,4S)-2-(diethylcarbamoyl)-4-(2-methoxypyridine-3-amido)pyrrolidin-1-yl]acetic acid
2-[(4-benzylpiperazin-1-yl)methyl]-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]-1,3-oxazole-4-carboxamide
2-(4,6-dimethoxypyrimidin-2-yl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
1-{[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}-4-(pyridin-2-yl)piperazine
1-[1-(diphenylmethyl)-1H-1,2,3-triazole-4-carbonyl]-3-(pyrrolidin-1-ylmethyl)piperidine
ethyl 1-(2-methoxyacetyl)-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylate
N-[(3S,4R)-4-(4-methylphenyl)-1-[2-(2-oxopyrrolidin-1-yl)acetyl]pyrrolidin-3-yl]acetamide
4-[7-(cyclobutylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-2-methoxypyridine-3-carbonitrile
N-{[4-amino-6-(dimethylamino)-1,3,5-triazin-2-yl]methyl}-2-benzyl-1,3-thiazole-4-carboxamide
1'-(pyrimidin-4-yl)-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
1-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-(morpholin-3-yl)ethan-1-one
1-[2-(2,3-dihydro-1H-inden-1-yl)acetyl]-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
3-(3-methyl-1H-1,2,4-triazol-5-yl)-N-[4-(2-oxopyrrolidin-1-yl)phenyl]piperidine-1-carboxamide
3-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-1-[3-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]urea
N-cyclopropyl-1-{1-[(2E)-4-methylpent-2-en-1-yl]piperidin-4-yl}piperidine-4-carboxamide
4-[4-(dimethylamino)-5-fluoropyrimidin-2-yl]-1,4-oxazepan-6-ol
1-[1-(2-carbamoylethyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
1-[(3R)-3-fluoropyrrolidin-1-yl]-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
2-(6-methoxynaphthalen-2-yl)-4-[5-(propan-2-yl)pyrimidin-4-yl]morpholine
4-[(3-hydroxypyrrolidin-1-yl)sulfonyl]-N-[2-(1H-pyrazol-1-yl)ethyl]benzamide
6-fluoro-4-[2-(3-methyl-4H-1,2,4-triazol-4-yl)ethyl]-3,4-dihydro-2H-1,4-benzoxazin-3-one
2-methyl-5-[(1R,5R)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-3,4-dihydropyrimidin-4-one
2-[2-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)ethyl]-1,3-benzothiazole
(benzylsulfamoyl)(2-hydroxyethyl)[(2-methylphenyl)methyl]amine
N-(3,3-diphenylpropyl)-6-[2-(3-methyl-1H-1,2,4-triazol-5-yl)acetyl]-6-azaspiro[2.5]octane-1-carboxamide
N-ethyl-N-[2-(4-methoxyphenoxy)ethyl]-2-(propan-2-yloxy)acetamide
N,N-dimethyl-2-(pyridin-3-yl)-7-(1H-pyrrole-2-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(3aR,6aR)-2-[(1-ethyl-1H-imidazol-5-yl)methyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-({[(2,6-dimethylpyridin-4-yl)methyl]amino}methyl)-3-hydroxy-1-(3-phenylpropyl)piperidin-2-one
(3aR,6aS)-N-(4-{[2-(pyridin-2-yl)ethyl]sulfanyl}phenyl)-octahydropyrrolo[3,4-c]pyrrole-2-carboxamide
1-(5-cyclopropyl-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-1H-pyrazole-4-carbonyl)-N,N-diethylpyrrolidin-3-amine
1-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}piperidine-3-carbonitrile
6-{[1-(phenoxymethyl)cyclopropyl]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
1-{4-[(3-methylphenyl)methyl]-3-oxopiperazin-1-yl}-4-phenylbutane-1,4-dione
5-(2-methoxyphenoxymethyl)-N-methyl-N-[1-(pyridin-3-yl)ethyl]-1,2-oxazole-3-carboxamide
2-[2-(3-ethenylphenyl)-1H-imidazol-1-yl]-N-methylbutanamide
4-[(dimethylamino)methyl]-1-(5-methylpyrimidin-2-yl)azepan-4-ol
N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-2,6,8-trimethylquinoline-4-carboxamide
(3S,4S)-1-(4-amino-5-methylpyrimidin-2-yl)-4-(naphthalen-2-yl)piperidin-3-ol
2-[({1-[(2-fluorophenyl)methyl]piperidin-3-yl}amino)methyl]-6-methoxyphenol
2-(2,5-dihydro-1H-pyrrol-1-yl)-4-[1-(4-fluorophenyl)-1H-pyrazol-4-yl]pyrimidine
1-(2-aminoethyl)-N-[3-(1,3-benzothiazol-2-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
N-benzyl-N-methyl-3-(1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidin-4-yl)propanamide
2-(1H-1,2,4-triazol-1-yl)-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}acetamide
N-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-1-[2-(morpholin-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-hydroxy-4-(oxolan-2-ylmethoxy)-5-(1H-pyrazol-3-yl)benzoic acid
5-[3-(aminomethyl)pyrrolidin-1-yl]-2-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-2,3-dihydropyridazin-3-one
N-{2-[3-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]propyl}-2,3,4,9-tetrahydro-1H-carbazole-6-carboxamide