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3-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-1-(3-methanesulfonamidophenyl)urea
N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-4-(1H-pyrazol-3-yl)benzamide
3-(2-fluorophenyl)-1-(4-methyl-1,4-diazepan-1-yl)-3-phenylpropan-1-one
1-methyl-N-[(5-methylfuran-2-yl)methyl]azepane-2-carboxamide
methyl 4-[5-methyl-4-({1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}methyl)-1,3-oxazol-2-yl]benzoate
N-({4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)pyridine-4-carboxamide
ethyl 3-benzyl-1-(1-benzyl-1H-pyrazole-4-carbonyl)piperidine-3-carboxylate
1-(2-{4-[(6-chloropyridin-3-yl)methyl]piperazin-1-yl}pyrimidin-4-yl)pyrrolidin-3-ol
N-ethyl-2-{[4-(pyridin-3-yl)piperazin-1-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
1-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3,3,3-trifluoropropan-1-one
{[3-(1-butyl-3-methyl-1H-1,2,4-triazol-5-yl)phenyl]methyl}dimethylamine
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(5-methylpyrazine-2-carbonyl)pyrrolidin-3-yl]methanol
5-(2-chloro-4-methoxyphenoxymethyl)-N-[2-(3-fluorophenyl)ethyl]-1,2-oxazole-3-carboxamide
(3S,9aR)-3-methyl-8-[(2-methylphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
1-[5-({[(5-fluoro-1H-indol-2-yl)methyl](methyl)amino}methyl)-2-methoxyphenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
N-(1-{4-[(2,3-dihydro-1-benzofuran-2-ylmethyl)(methyl)carbamoyl]phenyl}-1H-pyrazol-4-yl)oxane-4-carboxamide
5-chloro-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methylpyridine-2-carboxamide
N-[1-(6-chloropyridazin-3-yl)piperidin-4-yl]-2-(1H-pyrazol-1-yl)butanamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-sulfamoylbenzamide
2-methoxy-6-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]-5-oxo-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
(3S,4S)-1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-4-(propan-2-yloxy)pyrrolidin-3-ol
N-({1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}methyl)thiophene-2-carboxamide
2-chloro-4-({[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl](prop-2-en-1-yl)amino}methyl)phenol
2-[4-(6-cyclopropylpyrimidin-4-yl)phenyl]-2-methylpropanenitrile
N-(1-{7-[(2,6-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)pyridine-3-carboxamide
2-[(1-acetylpiperidin-4-yl)oxy]-5-methoxy-N-methyl-N-(oxan-2-ylmethyl)benzamide
2-(1,5-dimethyl-1H-indazole-3-carbonyl)-8-methyl-2,8-diazaspiro[4.5]decane
4-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-2-[(4-phenyl-1,3-thiazol-2-yl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
1-methyl-N-(pyridin-4-ylmethyl)-5-({[4-(trifluoromethoxy)phenyl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-{[4-(6-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}piperidin-3-ol
N,1-dimethyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-1H-1,2,3-benzotriazole-5-carboxamide
1-(3-{[(adamantan-1-yl)amino]methyl}-7-methoxyquinolin-2-yl)-4-[2-(dimethylamino)ethyl]-1,4-diazepan-5-one
3-(2,5-dioxoimidazolidin-4-yl)-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}propanamide
5-{[(2,3-dimethoxyphenyl)methyl]amino}-N,N-dimethyl-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
[3-methyl-1-({1-[1-(pyridin-4-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)piperidin-3-yl]methanol
1-cyclopentyl-4-[1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperazine
4-(2-fluoro-5-methylphenoxy)-1-[(2-methylpyrimidin-5-yl)methyl]piperidine-4-carboxylic acid
2,5-dimethyl-3-[3-methyl-5-(pyrrolidin-1-ylmethyl)phenoxy]pyrazine
1-{1'-cyclopentanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}-2-methoxyethan-1-one
(5S,9aS,9bS)-2-[(2-methoxyphenyl)methyl]-5-(4-phenyl-1,3-thiazol-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-[5-(2-ethoxyethyl)-1,3,4-thiadiazol-2-yl]-1-[1-(thiophen-2-yl)propyl]urea
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[3-(hydroxymethyl)-3-propylpiperidin-1-yl]ethan-1-one
N4-(furan-2-ylmethyl)-N2,N2,N4,5,6-pentamethylpyrimidine-2,4-diamine
(4aS,8aR)-6-(pyridine-4-carbonyl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
1-[(4-chlorophenyl)methyl]-N-[3-(4-methoxyphenyl)propyl]-6-oxopiperidine-3-carboxamide
(1S,5R)-6-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-[(3R,4S)-3-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanamido]-4-(propan-2-yl)pyrrolidin-1-yl]propanoic acid
ethyl 1-(cyclopropylmethyl)-5-(1H-indol-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
8-[3-(dimethylamino)pyrazin-2-yl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid