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[5-methyl-7-(thiophen-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
N4-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-2-methylpyrimidine-4,6-diamine
2-(4-methylnaphthalen-1-yl)-2-(3-oxopiperazin-1-yl)acetic acid
(5S,9aS,9bS)-2-cyclopentyl-5-[3-(2-hydroxyethoxy)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-(4-methyl-6-{[3-(1H-1,2,3-triazol-1-yl)propyl]amino}pyrimidin-2-yl)phenol
1-ethyl-N-methyl-2-oxo-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1,2-dihydropyridine-4-carboxamide
N-[(1-cyclohexylpyrrolidin-3-yl)methyl]pyrimidin-4-amine
3-(4-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)-2,5-dimethylpyrazine
3-(1-methylpiperidin-3-yl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}propanamide
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methylpropyl)acetamide
ethyl 1-(1-ethylpiperidine-2-carbonyl)-4-[(4-methoxyphenyl)methyl]piperidine-4-carboxylate
1-[(1-benzyl-4-phenylpiperidin-4-yl)methyl]-5-oxopyrrolidine-3-carboxylic acid
2-(2,4-dioxoimidazolidin-1-yl)-N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}acetamide
1-(3-methylpyridin-4-yl)-4-(thiophen-3-ylmethyl)-1,4-diazepane
(2R)-2-hydroxy-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-2-phenylacetamide
8-(2,2-dimethylpropyl)-1-ethyl-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[(2-acetamidoethyl)sulfamoyl]-N-(2-fluoroethyl)benzamide
N,6-dimethyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-2-oxo-4-(pyridin-3-yl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
2-methyl-4-(4-{[4-(2-methylpyrimidin-4-yl)piperidin-1-yl]methyl}phenyl)butan-2-ol
3-chloro-5-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,2-dihydropyridin-2-one
3-phenyl-1-{1-[2-(pyrrolidin-1-yl)-5,6,7,8-tetrahydroquinazoline-4-carbonyl]piperidin-3-yl}propan-1-one
5-cyano-N,2-dimethyl-6-oxo-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-1,6-dihydropyridine-3-carboxamide
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-({[(5-methylpyrazin-2-yl)methyl]amino}methyl)piperidin-2-one
1-(2-fluorophenyl)-4-{1-[4-(propan-2-yloxy)benzoyl]piperidin-3-yl}piperazine
N,1-dimethyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]azepane-2-carboxamide
5-{4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-1-carbonyl}-2-methylpyrimidin-4-ol
1-(6-carbamoylpyrazin-2-yl)-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
1-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-[(2-ethyl-6-methylpyridin-3-yl)oxy]ethan-1-one
8-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-3-[(4-methoxyphenyl)methyl]-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-3,4-dihydro-2H-1,4-benzoxazine-7-carboxamide
2-cyclopentyl-8-(6-methyl-4-oxo-1,4-dihydropyridine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(5-acetylpyridin-2-yl)-4-(4-methylphenoxy)piperidine-4-carboxylic acid
3-(3-chlorobenzoyl)-N-(4-methoxyphenyl)piperidine-1-carboxamide
N-(3-methoxypropyl)-1-methyl-5-{1-[3-(trifluoromethyl)phenyl]propan-2-yl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[1-benzyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-3-methoxypropanamide
N-(2-cyclopentylethyl)-1-[2-(4-methoxyphenyl)ethyl]-6-oxopiperidine-3-carboxamide
3-[(3S,4R)-4-(morpholin-4-yl)-1-(pyridin-4-ylmethyl)piperidin-3-yl]-N-[2-(piperidin-1-yl)ethyl]propanamide
6-(3-methylpyrazin-2-yl)-2-[3-(thiomorpholin-4-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
3-[1-(4-chlorobenzenesulfonyl)piperidin-4-yl]-N-[(4-fluorophenyl)methyl]propanamide
3-cyclopentyl-5-[(4-fluorophenyl)methyl]-5-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
N-[(2-fluorophenyl)methyl]-3-[(4-methylpiperazin-1-yl)sulfonyl]-5-phenylbenzamide
N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-5-(oxolan-2-yl)thiophene-2-carboxamide
(3S)-3-ethyl-4-[2-(1H-pyrazol-1-yl)benzoyl]morpholine
(2S,4R)-1-[(3-hydroxyphenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]-N-(quinoxalin-6-yl)pyrrolidine-2-carboxamide
4-chloro-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
3-(3-methylbutyl)-8-(1-methylpiperidine-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(4aS,7aR)-1-(1H-indole-5-carbonyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-cyclopropyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1,3,4-oxadiazol-2-amine
(2S,3R)-3-hydroxy-2-[(2-methyl-5-propylpyrimidin-4-yl)amino]butanamide
2-methyl-5-{5-methylthieno[2,3-d]pyrimidin-4-yl}quinoline