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N5-ethyl-N3-methyl-1-(2-methylpropyl)-4-oxo-N3-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
4-{4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]benzoyl}-1-phenylpiperazin-2-one
2-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]pyridine-4-carboxamide
{5-chloro-7-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
2-methyl-4-(4-{[3-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl}phenyl)butan-2-ol
3-(5-acetyl-2,4-dimethyl-1H-pyrrole-3-carbonyl)-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
(4S,4aS,8aS)-1-(2-methyl-1,3-thiazole-4-carbonyl)-4-phenyl-decahydroquinolin-4-ol
1-(carbamoylmethyl)-N-{5H,6H,7H,8H,9H,10H-cyclohepta[b]indol-2-ylmethyl}piperidine-4-carboxamide
1-[4-({[2-(2-chlorophenyl)ethyl]amino}methyl)-2-methoxyphenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
3-chloro-4-{[2-(1,3-thiazol-2-yl)piperidin-1-yl]methyl}pyridine
4-[3-(4-ethoxypiperidine-1-carbonyl)phenyl]-2-methylbutan-2-ol
N-[2-(2-chloro-6-fluorophenyl)ethyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
methyl 5-(cyclopentylamino)-3-acetamido-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-({2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}sulfonyl)azepane
5-{[2-(2-phenylethyl)morpholin-4-yl]methyl}-N-(propan-2-yl)pyrimidin-2-amine
1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-N-ethyl-N-(pyridin-4-ylmethyl)piperidin-3-amine
2-ethyl-1-[(4-methoxyphenyl)methyl]-6-methyl-N-{[1-(morpholin-4-yl)cycloheptyl]methyl}-4-oxo-1,4-dihydropyridine-3-carboxamide
({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(cyclopropylmethyl)propylamine
N-methyl-3-(5-methylthiophen-2-yl)-N-[2-(phenylsulfanyl)ethyl]-1H-pyrazole-5-carboxamide
N-(1-methoxypropan-2-yl)-5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-amine
1-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-2-methyl-4-(2-methylphenyl)piperazine
2-(dimethyl-1,2-oxazol-4-yl)-1-{7-[2-hydroxy-4-(1H-pyrazol-1-yl)butan-2-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}ethan-1-one
methyl 1-{2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]acetyl}piperidine-4-carboxylate
6-[2-({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)ethyl]-2-methylpyrimidin-4-ol
N-({7-[(5-acetamidothiophen-2-yl)methyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(phenylsulfanyl)acetamide
5-[5-(ethoxymethyl)-1,2,4-oxadiazol-3-yl]-6-methyl-2-[(2R)-oxolane-2-carbonyl]-1,2,3,4-tetrahydro-2,7-naphthyridine
5-methoxy-N-(2-methoxyethyl)-1,2-dimethyl-N-[(3-methylthiophen-2-yl)methyl]-1H-indole-3-carboxamide
2-[1-(2-phenylethyl)-4-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}piperazin-2-yl]ethan-1-ol
1-(1-benzofuran-2-ylmethyl)-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
butyl 3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxylate
N-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]-1H-pyrazole-4-carboxamide
2-methyl-4-{4-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]phenyl}butan-2-ol
N-[3-(azepan-1-yl)propyl]-1-[(2-chlorophenyl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
5-({4-[(4-chlorophenyl)methyl]piperazin-1-yl}methyl)-2-(furan-2-yl)pyrimidine
3-[2-(dimethylamino)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1,4,6-trimethyl-1,2-dihydropyridin-2-one
9-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-phenyl-1-[1-(pyridin-4-yl)piperidin-4-yl]propan-1-ol
2,3-dimethyl-N-({1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}methyl)benzamide
(1S,5R)-6-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-({5-[(2,3-difluoro-4-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxyacetamide
(2S)-2-amino-2-cyclohexyl-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}acetamide
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(1,3-dihydroxypropan-2-yl)acetamide
3-(2,5-dihydro-1H-pyrrol-1-yl)-N-(2-ethoxyphenyl)-3-oxopropanamide
methyl 2-oxo-1-(prop-2-en-1-yloxy)-8-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-1,8-diazaspiro[4.5]decane-4-carboxylate
N-cyclobutyl-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
1-[2-(1H-imidazol-1-yl)ethyl]-2-(4-methanesulfonylphenyl)-1H-imidazole
N-{[4-(2-methoxyethoxy)phenyl]methyl}-5,6-dimethylpyrimidin-4-amine
1-(3-fluorophenyl)-3-(1-{1-[3-(pyridin-3-yl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
3-{[5-(5-ethylfuran-2-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1λ6-thiolane-1,1-dione
5-{[(2,6-difluoro-3-methylphenyl)methyl]amino}-1-ethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid