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6-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carbonyl}-2-methyl-2,3-dihydropyridazin-3-one
(1R,5R)-6-[2-(difluoromethoxy)benzoyl]-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
3-{1-methyl-4-[4-(pyrrolidin-1-yl)piperidin-1-yl]-1H-pyrazolo[3,4-d]pyrimidin-6-yl}pyridine
3-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(2-methoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(2,4-dioxo-1,3-diazinan-1-yl)-N-[2-(3-methylpyridin-2-yl)ethyl]benzamide
1-({5-[3-(2-fluorophenyl)-1H-pyrazol-5-yl]-1,2,4-oxadiazol-3-yl}methyl)-4-methylpiperazine
4-[5-(3-fluorobenzoyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperazin-2-one
7-(5-methylthiophen-2-yl)-4-(2-propoxyethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-3-(3-fluorophenyl)benzamide
3-(3-hydroxy-3-methylbutyl)-N-[2-(1,3-thiazol-4-yl)ethyl]benzamide
N3-ethyl-N5-[2-(3-fluorophenyl)ethyl]-N3-(2-methylprop-2-en-1-yl)-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-methyl-1,3-benzoxazole-6-carboxamide
(4aR,7aS)-1-benzyl-4-(6-oxo-1,6-dihydropyridine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(6-methoxy-2-oxo-2,3-dihydro-1H-indol-3-yl)acetamide
1-{3-[1-(2-phenylethyl)piperidin-4-yl]pyrrolidin-1-yl}-3-(pyridin-3-yl)propan-1-one
2-{1-[(5-methylfuran-2-yl)methyl]-4-(pyridin-4-ylmethyl)piperazin-2-yl}ethan-1-ol
1-amino-N-{[1-(2-methylpropyl)piperidin-3-yl]methyl}cyclopentane-1-carboxamide
2-(azocan-1-yl)-1-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}ethan-1-one
1-(2-methylphenyl)-3-{1-[1-(2-oxobutanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
N-(1-{1-[(2-chloro-4-fluorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2,2-dimethylpropanamide
N-cyclopropyl-N-{[2-(3,4-dimethoxyphenyl)-7-methylquinolin-3-yl]methyl}-1,3-thiazole-5-carboxamide
1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
3-[(2R,3R,6R)-5-(5-methylpyrazine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
1-({2-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)-4-(pyrrolidin-3-yl)piperazine
3-{1-[(2,3-difluoro-6-methoxyphenyl)methyl]piperidin-2-yl}propanoic acid
[3-(cyclopropylmethyl)-1-{[6-(dimethylamino)pyridin-3-yl]methyl}piperidin-3-yl]methanol
5-(azepane-1-carbonyl)-1-(butan-2-yl)-N-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-4-oxo-1,4-dihydropyridine-3-carboxamide
1-[5-(methanesulfonylmethyl)pyridin-2-yl]-4-(pentan-3-yl)piperazine
[1-(2-chlorophenyl)ethyl]({[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
methyl 2-{2-[2-amino-3-cyano-6-(propan-2-yl)pyridin-4-yl]phenoxy}acetate
N-methyl-N-[1-(pyridin-2-yl)propan-2-yl]-3-(4H-1,2,4-triazol-4-yl)benzamide
1-(3-chlorophenyl)-4-[(3-{2-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-2-yl]ethoxy}phenyl)methyl]piperazine
4-benzyl-3-ethyl-1-(2-fluoro-6-methoxybenzoyl)-1,4-diazepan-5-one
(4aR,7aS)-1-acetyl-4-{imidazo[1,2-a]pyridine-2-carbonyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-amino-6-(propan-2-yl)-4-[1-(pyridin-2-yl)-1H-pyrrol-2-yl]pyridine-3-carbonitrile
N-(8-chloro-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-2-(1,3-thiazol-2-yl)pyrrolidine-1-carboxamide
N-(1-{7-[(5-ethylfuran-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)pyridine-3-carboxamide
1-(6-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}pyridin-3-yl)ethan-1-one
N-cyclopentyl-N-[2-(dimethylamino)ethyl]-5-[(dimethylamino)methyl]furan-2-carboxamide
2-[8-(3-methylbutyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]acetamide
8-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
1-(2-fluorophenyl)-4-{1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-3-yl}piperazine
1-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-5-oxopyrrolidine-3-carboxylic acid
2-{[(3S)-2-oxoazepan-3-yl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
1-(3-{2-[2-(4-hydroxyphenyl)ethyl]piperidine-1-carbonyl}phenyl)imidazolidin-2-one
2-{5-[(1E)-1-(furan-2-yl)prop-1-en-2-yl]-4-phenyl-1H-imidazol-1-yl}-N-methylethane-1-sulfonamide
5-(2,6-difluorophenoxymethyl)-N-{[2-(trifluoromethoxy)phenyl]methyl}-1,2-oxazole-3-carboxamide
1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}-4-(3-methylpiperidine-1-carbonyl)piperidine
1-[({[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}carbamoyl)methyl]piperidine-4-carboxamide
1-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one