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2-{8-methylimidazo[1,2-a]pyridin-3-yl}-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]acetamide
1-[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]-2-(1-methyl-1H-pyrrol-2-yl)ethane-1,2-dione
3-(2-{6-azabicyclo[3.2.1]octan-6-yl}-2-oxoethyl)-1-cyclopentyl-3-(4-methoxyphenyl)pyrrolidine-2,5-dione
2-chloro-5-(piperidin-1-yl)-N-[1-(pyrazin-2-yl)propan-2-yl]benzamide
2-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]-1-(piperazin-1-yl)ethan-1-one
N-{[7-(9H-fluoren-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}acetamide
5-ethyl-N-[(1-phenylpyrrolidin-3-yl)methyl]pyrimidin-2-amine
2-hydroxy-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)butanamide
N-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-2-methylpyrido[2,3-d]pyrimidin-4-amine
(3R,5S)-5-[4-(dimethylamino)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]pyrrolidin-3-ol
N-[2-(6-hydroxypyrimidin-4-yl)ethyl]-2,3-dimethyl-1H-indole-7-carboxamide
2-[1-(3,5-dimethyl-1-benzofuran-2-carbonyl)piperidin-4-yl]-5-methyl-1H-1,3-benzodiazole
2-[3-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyrazine
N-{2-hydroxy-2-[2-(trifluoromethyl)phenyl]ethyl}-3-(4H-1,2,4-triazol-4-yl)benzamide
1-(3-chloro-4-fluorophenyl)-5-(oxan-2-yl)-1H-1,2,4-triazole
(3S)-1-{5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-yl}pyrrolidin-3-ol
(2,1,3-benzothiadiazol-5-ylmethyl)({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)methylamine
2-(3-fluorophenyl)-1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
4-(1-aminocyclobutanecarbonyl)-7-(1-benzothiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[(4-fluorophenyl)methyl]-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[(4-methylphenyl)methyl]-7-(pyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-{1'-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}-2-methoxyethan-1-one
2-cyclopropyl-N-(2-{[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]methyl}propyl)pyrimidine-5-carboxamide
2-[methyl(oxan-2-ylmethyl)amino]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
methyl({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl})(quinolin-2-ylmethyl)amine
(3aS,6aS)-2-ethyl-5-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
methyl 2-{[2-(2-fluorophenyl)ethyl]sulfamoyl}-6-(4-methylpentanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-methyl-5-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
methyl (2S,4R)-4-(2-methylpropanamido)-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxylate
2-(2,5-dimethoxyphenyl)-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
7-(cyclopropylmethyl)-2-(morpholine-4-sulfonyl)-2,7-diazaspiro[4.5]decan-6-one
3-cyclohexyl-N-(furan-2-ylmethyl)-N-(pyridin-4-ylmethyl)-1H-pyrazole-4-carboxamide
8-[2-(dimethyl-1,3-thiazol-4-yl)acetyl]-2-(3-methylphenyl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
2-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}acetic acid
N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-3-(2-methoxyphenyl)-N-(pyridin-3-ylmethyl)propanamide
2-(3-phenylpropyl)-N-[2-(1H-pyrazol-4-yl)ethyl]-1,3-benzoxazole-5-carboxamide
7-(cyclopropylmethyl)-2-(4-methyl-1,3-thiazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]-4-(1H-pyrazol-1-yl)butanamide
2-(3,4-dihydro-2H-1-benzopyran-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
5-methyl-N-[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]pyrazolo[1,5-a]pyrimidin-7-amine
3-[4-(1-methylpiperidin-4-yl)piperazine-1-carbonyl]-1H-pyrazol-5-amine
N-{5-[(1E)-pent-1-en-1-yl]pyridin-2-yl}methanesulfonamide
N-{imidazo[1,2-a]pyridin-2-ylmethyl}-5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[cyclopropyl(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-hydroxy-2-phenylpyrimidine-5-carboxamide
3-chloro-N-({3,5-dimethoxy-4-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]benzene-1-sulfonamide
methyl[1-(pyrimidin-4-yl)ethyl]{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]{[4-(5-methylpyridin-2-yl)piperidin-4-yl]methyl}amine
(2S,4S)-1-{[4-(diethylamino)phenyl]methyl}-4-{[(2-fluorophenyl)methyl]amino}-N-methylpyrrolidine-2-carboxamide
1-[4-(benzyloxy)piperidin-1-yl]-2-(oxan-2-ylmethoxy)ethan-1-one
ethyl 4-[3-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]piperidine-1-carboxylate