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N-{[2-(4-acetylpiperazin-1-yl)-6-methylquinolin-3-yl]methyl}-N-[2-(cyclohex-1-en-1-yl)ethyl]-2-methoxyacetamide
5-chloro-3-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
methyl({[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
(3R,4R)-1-[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]-4-(morpholin-4-yl)piperidin-3-ol
3-fluoro-N-[(3R)-piperidin-3-yl]imidazo[1,2-a]pyridine-2-carboxamide
3-methyl-1-[(3-methylphenyl)methyl]-4-[2-(pyridin-4-yl)pyrimidine-5-carbonyl]piperazin-2-one
1-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-6-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-6-azaspiro[2.5]octane
6-fluoro-2-{[(oxan-4-yl)amino]methyl}quinolin-4-ol
3-(3-hydroxyquinoxalin-2-yl)-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}propanamide
5-{[2-(morpholin-4-yl)quinolin-3-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-methylbenzamide
3-phenyl-5-(thiophene-3-sulfonyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
4-butyl-11-({[2-fluoro-4-(trifluoromethyl)phenyl]methyl}amino)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
ethyl 1-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylate
4-{[(4-methyl-1H-imidazol-5-yl)methyl]amino}-1-(2-phenylethyl)pyrrolidin-2-one
N-(4-{thieno[3,2-d]pyrimidin-4-yl}-1H-pyrrolo[2,3-b]pyridin-6-yl)piperidin-4-amine
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[(2-fluoro-3-methylphenyl)methyl]pyrrolidine-3-carboxylic acid
N-[(5-chlorothiophen-2-yl)methyl]-2-(2,5-dioxoimidazolidin-1-yl)acetamide
3-(oxan-4-ylmethyl)-5-(piperidin-4-yl)-5-propylimidazolidine-2,4-dione
1-methyl-1'-[2-(1H-pyrazol-1-yl)butanoyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
1-benzyl-4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-1-yl]ethan-1-one
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-[(2-fluorophenyl)methyl]-1H-pyrazole-4-carboxamide
2-[2-(2,3-dihydro-1H-inden-5-yloxy)-2-methylpropanoyl]-2,7-diazaspiro[4.5]decan-6-one
2-chloro-9-methyl-3-({methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}methyl)-4H-pyrido[1,2-a]pyrimidin-4-one
N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-3,5-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
N-[(3R,5S)-5-(ethylcarbamoyl)-1-[(2E)-3-phenylprop-2-en-1-yl]pyrrolidin-3-yl]pyridine-2-carboxamide
2,4-dimethyl-5-[3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyrimidine
1-(2-fluorophenyl)-4-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]piperidine
(4aR,7aS)-1-ethyl-4-({9-hydroxy-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]pyrrolidin-3-yl]methanol
1-{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(methoxymethyl)piperidine
4-({[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}carbamoyl)pyridin-1-ium-1-olate
(3S,4S)-1-cyclopentyl-4-cyclopropylpyrrolidine-3-carboxylic acid
8-(2-methyl-1H-pyrrole-3-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-(3-ethoxypropyl)-2-(4-methanesulfonylphenyl)-1H-imidazole
7-(2-methylphenyl)-4-(4-methylpyrimidin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(1'-{[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)propan-1-one
2-[3-(2-methoxyphenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(quinoxalin-6-ylmethyl)acetamide
N-({1-[(2-butyl-1H-imidazol-4-yl)methyl]piperidin-3-yl}methyl)pyridine-3-carboxamide
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
4-(1-{[3-(1H-imidazol-2-yl)phenyl]methyl}piperidin-4-yl)morpholine
3,5-dimethyl-N-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1-(prop-2-en-1-yl)-1H-pyrazole-4-carboxamide
5-cyclopropyl-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-1,3-oxazole-4-carboxamide
4-({4-methyl-5-[1-(pyridin-4-yl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
N-cyclopentyl-4-[5-(morpholin-4-ylmethyl)pyridin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
1-[2-({[5-(4-methoxyphenyl)-1,2-oxazol-3-yl]methyl}amino)-4-methylpyrimidin-5-yl]ethan-1-one
N-(1-{7-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)methanesulfonamide
8-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}quinoline
1-cyclopentyl-N-[(3,5-dimethoxyphenyl)methyl]-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide