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4-[({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl)amino)methyl]-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
ethyl 2-cyclohexyl-2-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)acetate
1-(methoxymethyl)-N-[2-(2-methyl-1H-indol-1-yl)ethyl]cyclobutane-1-carboxamide
N-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]phenyl}acetamide
2-(2-aminoethyl)-5,6-dimethyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]thieno[2,3-d]pyrimidin-4-amine
2-(3-fluorophenoxymethyl)-N-[2-(oxan-2-yl)ethyl]-1,3-oxazole-4-carboxamide
1-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
N4,N4,N6-trimethyl-N6-[2-(pyrrolidin-1-ylmethyl)propyl]pyrimidine-4,6-diamine
N-{2-[2-(thiophen-3-yl)acetyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}pyridine-4-carboxamide
2-(2-propoxyethyl)-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
4-({1-[2-(ethylamino)pyrimidine-5-carbonyl]pyrrolidin-3-yl}methyl)benzoic acid
N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]-1-[3-(pyridin-3-yl)azetidin-1-yl]butan-1-one
4-(4-chlorophenyl)-1-[4-(oxolane-2-carbonyl)piperazin-1-yl]butan-1-one
4-methoxy-6-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyrimidine
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[(2-ethylphenyl)methyl]pyrrolidin-3-yl]methanol
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-4-(piperidin-3-yl)benzamide
N-(2-hydroxyethyl)-2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-N-methyl-1,3-oxazole-4-carboxamide
4-(pyridin-3-yl)-1-[(4-{[3-(trifluoromethyl)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methyl]piperidin-4-ol
4-[2-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]-1,3-thiazol-2-amine
5-[1-(2-methylbutanoyl)piperidin-4-yl]-5-(pyridin-3-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
methyl (2S,4S)-4-(2,6-dimethoxypyrimidine-4-amido)-1-methylpyrrolidine-2-carboxylate
N-[(2-methylphenyl)(pyridin-4-yl)methyl]-2-(pyridin-2-yl)acetamide
N-[(1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)methyl]acetamide
dimethyl[1-(4-{1-[2-(morpholin-4-yl)ethyl]-1H-imidazol-2-yl}phenyl)ethyl]amine
N-methyl-N-[2-(pyridin-2-yl)ethyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
2-[(3,5-difluorophenyl)methyl]-8-(1,2-oxazole-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
N-[2-(2-fluoro-5-methoxyphenyl)pyridin-3-yl]-2-methylpropanamide
N-{[(3S,4S)-3-hydroxy-1-(1-hydroxycyclopentanecarbonyl)piperidin-4-yl]methyl}-2-methylbenzamide
1-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)-2-{methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}ethan-1-one
1-(cyclopentylmethyl)-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol
8-[3-(4-fluorophenoxy)propyl]-2-methyl-2,8-diazaspiro[4.5]decan-3-one
N-cyclopropyl-1,3-dimethyl-N-[(3-methylthiophen-2-yl)methyl]-1H-indole-2-carboxamide
(3R)-1-[2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carbonyl]-3-methylpiperazine
2-ethoxy-3-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]pyridine
3-{[1-(1,4-dioxane-2-carbonyl)piperidin-4-yl]methyl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]ethan-1-one
1-[1-(3-chlorobenzoyl)piperidin-4-yl]-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(pyrrolidine-1-carbonyl)piperidine
N-[(3R,5S)-5-(ethylcarbamoyl)-1-[(3-hydroxyphenyl)methyl]pyrrolidin-3-yl]pyrazine-2-carboxamide
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-N-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]acetamide
N-{2-[4-(hydroxymethyl)piperidin-1-yl]-5,6,7,8-tetrahydroquinazolin-5-yl}-6-methylpyridine-3-carboxamide
N-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-[(trimethyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
(3R,5S)-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]-1-[(3,4-dimethoxyphenyl)methyl]-N-[2-(dimethylamino)ethyl]piperidine-3-carboxamide
4-(3,5-difluoro-4-methoxyphenyl)-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(1-methyl-1H-pyrazole-4-carbonyl)-decahydro-1,6-naphthyridin-2-one
3-phenyl-N-{1-[7-(quinolin-8-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}propanamide
2-{1-[(4-fluorophenyl)methyl]-5-[1-(1H-1,2,4-triazol-1-yl)ethyl]-1H-1,2,4-triazol-3-yl}pyridine
{2-[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-1,3-thiazol-4-yl}methanol