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3-[(1-cycloheptyl-5-oxopyrrolidin-3-yl)carbamoyl]pyridin-1-ium-1-olate
1-(2-chloro-4,6-dimethylphenyl)-3-methyl-3-[(3-methyl-1H-pyrazol-4-yl)methyl]urea
2-chloro-5-{3-[1-(dimethylamino)ethyl]phenyl}benzamide
2-ethyl-4-methyl-N-[3-(3-phenylpropanamido)phenyl]-1,3-oxazole-5-carboxamide
1-(azocan-1-yl)-3-{4-[(dimethylamino)methyl]-2-methoxyphenoxy}propan-2-ol
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl](methyl){[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}amine
1-{[1-(2,4-difluoro-3-methoxybenzoyl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
(2R,3R)-3-{methyl[3-(4-methylphenoxy)propyl]amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}-1-(morpholin-4-yl)propan-1-one
5-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]-N-phenylpyrimidin-2-amine
(1S,5R)-6-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-3-(2-phenylethyl)piperidine
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-1H-indazol-6-amine
2-(2-methyl-1,3-thiazol-4-yl)-N-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]acetamide
N-[1-(3-methoxyphenyl)-5-oxopyrrolidin-3-yl]-2-methylimidazo[1,2-a]pyridine-6-carboxamide
2-(4-methyl-1,4-diazepan-1-yl)-1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
4-{2-[(4-fluorophenyl)methyl]-3H-imidazo[4,5-b]pyridin-3-yl}-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine
8-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(2H-1,3-benzodioxole-5-carbonyl)-1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)piperidine
1-[(diethylcarbamoyl)methyl]-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1H-1,2,3-triazole-4-carboxamide
N1-(pyridin-3-yl)-N2-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}ethane-1,2-diamine
(2R,3R,6R)-5-(furan-2-ylmethyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-8-fluoro-1,4-dihydroquinolin-4-one
(2R)-2-amino-1-[4-(1H-imidazol-2-yl)piperidin-1-yl]-4-methylpentan-1-one
4-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl}-N,N-dimethylaniline
N-[5-(3-methanesulfonamidopropanamido)-2-methylphenyl]-3-methylbenzamide
5-(2-{3-[(4-methylpiperazin-1-yl)methyl]-1,2,4-oxadiazol-5-yl}ethyl)-1,2-oxazol-3-ol
N-(4-{3-[(3-fluorophenyl)amino]piperidine-1-carbonyl}phenyl)acetamide
(3aR,6aR)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-2-(pyrimidin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
1-{3-[3-(2-methylphenyl)piperidin-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
8-[(2-methyl-1,3-thiazol-4-yl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
4-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-7-(phenoxathiin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-(3-chloro-4-methoxyphenyl)-3-[1-(pyridine-3-carbonyl)piperidin-3-yl]propanamide
3-{1-[1-(cyclohexylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-2-yl}propan-1-ol
(4aR,8aR)-4a-hydroxy-7-[(4-methoxypyridin-2-yl)methyl]-N,N-dimethyl-decahydro-2,7-naphthyridine-2-sulfonamide
5-(1,3-benzothiazol-2-ylmethyl)-1-(cyclopropylmethyl)-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-ol
3-[(4-fluorophenyl)formamido]-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}propanamide
1-(1-{2-methyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl}piperidin-4-yl)-3-phenylpropan-1-ol
ethyl[(3-fluoro-2-methoxyphenyl)methyl][(trimethyl-1H-pyrazol-4-yl)methyl]amine
1-{[5-(1H-imidazol-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-4-methanesulfonylpiperazine
methyl 3-(2-methoxyacetamido)-1-(3-methylbutyl)-5-[(naphthalen-1-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-[(3-methylphenyl)methyl]piperazin-2-one
6-ethyl-2-(1-propyl-1H-pyrazol-4-yl)-4-(pyrrolidine-1-carbonyl)quinoline
N-[1-(1H-imidazol-1-yl)butan-2-yl]-6-oxo-1,6-dihydropyridine-3-carboxamide
6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]-N-[2-(pyridin-3-yloxy)ethyl]piperidine-3-carboxamide
4-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}-3-propylmorpholine
9-(2-chloro-6-fluorobenzoyl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-1-ethyl-1H-pyrazole-4-carboxamide
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-3-(3-hydroxy-1,2-oxazol-5-yl)propanamide