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3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-(thiophen-3-ylmethyl)propanamide
{[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}[(1-ethyl-1H-imidazol-2-yl)methyl]methylamine
4-[1-(4-chloro-2-methylphenyl)-3-methyl-1H-1,2,4-triazol-5-yl]-2-(4H-1,2,4-triazol-4-yl)pyridine
9-[(4-fluoro-3-methylphenyl)methyl]-3-oxa-9-azaspiro[5.5]undecane
3-({7-[(2-methyl-1,3-oxazol-4-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]pyrrolidine-1-carboxamide
1-(2-butoxyacetyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-methoxy-N-({2-methoxy-5-oxo-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)acetamide
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-(dimethyl-1,3-oxazole-5-carbonyl)pyrrolidine-3-carboxylic acid
1-(dimethylamino)-2-(4-{[4-(propan-2-yloxy)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)propan-2-ol
2-phenoxy-N-{2-[7-(1,3-thiazol-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}acetamide
2-[3-(2-methylpropyl)-5-[2-(trimethyl-1H-pyrazol-4-yl)ethyl]-1H-1,2,4-triazol-1-yl]pyridine
8-cyclopropanecarbonyl-2-[(2-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-[1-(1-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
2-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane
N-(dimethyl-1H-1,2,4-triazol-3-yl)-3,3-difluoropiperidine-1-carboxamide
ethyl 2-[4-(4-fluorobenzenesulfonyl)-1-[(5-methylthiophen-2-yl)methyl]piperidin-4-yl]acetate
3-(1H-pyrazol-4-yl)-N-{2-[(pyridin-3-yl)amino]ethyl}benzamide
3-ethyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
1-(2-cyclohexylethyl)-3-hydroxy-3-({[2-(6-methylpyridin-2-yl)ethyl]amino}methyl)piperidin-2-one
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carboxamide
(1S,5R)-6-(cyclopropylmethyl)-3-[(5-fluoro-2-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
dimethyl({4-[1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)piperidin-2-yl]phenyl}methyl)amine
N-benzyl-N,1-diethyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
[(3R,4R)-1-[2-(methylamino)pyrimidine-5-carbonyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-methylbut-2-enamide
N-(furan-3-ylmethyl)-N,7-dimethyl-2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
7-(cyclobutylmethyl)-2-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
ethyl 1-[3-(furan-2-yl)propanoyl]-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
4-{1-[(2,3-difluoro-6-methoxyphenyl)methyl]azetidin-3-yl}morpholine
2-{[4-(oxolan-2-ylmethyl)phenyl]sulfanyl}acetamide
3-[2-(4-fluorophenyl)piperidin-1-yl]propanamide
2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1-[4-(pyrrolidin-1-ylmethyl)phenyl]-1H-imidazole
7-(1,3-benzothiazol-2-yl)-4-(6-methylpyridazin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]benzamide
N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-3-[5-(thiophen-2-yl)furan-2-yl]propanamide
3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}-2-(4-methoxyphenyl)imidazo[1,2-a]pyridine
2-{[1-(2-methoxyphenoxy)propan-2-yl]amino}-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
6-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N,N-dimethylpyridine-3-carboxamide
4-[(3-fluorophenyl)methyl]-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-[3-(2-chlorophenyl)pyrrolidine-1-carbonyl]-2-propyl-1,3-thiazole
N-butyl-4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}benzamide
5-[(dimethylamino)methyl]-N-[(4-methoxyphenyl)methyl]-N-methyl-1,3,4-oxadiazole-2-carboxamide
8-(4-hydroxy-3-methoxybenzoyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-butyl-1-(3-methylphenyl)-4-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]piperazin-2-one
(3S,4S)-1-(2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carbonyl)piperidine-3,4-diol
8-(4,6-dimethylpyridine-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
5-{1-[3-(2,3-dihydro-1H-isoindol-2-yl)propanoyl]pyrrolidin-2-yl}thiophene-2-carboxamide
ethyl 1-methyl-5-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-tert-butyl-3-cyclopentyl-5-[(methylsulfanyl)methyl]-1H-1,2,4-triazole