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3-(2-methoxyethyl)-1-(2-phenylethyl)-8-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)[(2,4,5-trimethoxyphenyl)methyl]amine
ethyl 2-[1-(8-fluoroquinoline-2-carbonyl)piperidin-2-yl]acetate
ethyl 6-{4-[(3-methyl-1H-pyrazol-5-yl)methyl]piperazin-1-yl}pyridine-3-carboxylate
2-{[(5-chloro-1-benzothiophen-3-yl)methyl]amino}-N-(pyrazin-2-yl)acetamide
{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(1-methoxybutan-2-yl)amine
9-[2-(2-fluorophenyl)acetyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N2-(4-methylphenyl)-6-(thiophen-2-yl)-1,3,5-triazine-2,4-diamine
N-(2-ethyl-2-methyl-4-oxo-3,4-dihydro-2H-1-benzopyran-6-yl)-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carboxamide
3-{1-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]piperidin-3-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(2S,4R)-1-[(3-chlorophenyl)methyl]-4-{[(2,5-difluorophenyl)methyl]amino}-N-ethylpyrrolidine-2-carboxamide
(1R,5S,6R)-3-(2,3-dihydroxypropyl)-N-[2-(3-fluorophenyl)ethyl]-3-azabicyclo[3.1.0]hexane-6-carboxamide
3-{2-[4-(1-hydroxypropyl)piperidin-1-yl]-2-oxoethyl}-1-methyl-3-(4-phenylphenyl)pyrrolidine-2,5-dione
1-(2-aminoethyl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]-1H-1,2,3-triazole-4-carboxamide
5-[4-(hydroxymethyl)phenyl]-2-methoxybenzamide
4-(1-ethyl-3-methyl-1H-pyrazole-4-carbonyl)-1-(2-methoxyphenyl)-2,2-dimethylpiperazine
3-(1-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}piperidin-3-yl)benzoic acid
1-{3-[benzyl(methyl)amino]piperidin-1-yl}-4-phenylbutan-1-one
3-[({2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}amino)methyl]piperidin-3-ol
3-cyclohexyl-N-[2-(4-phenylpyrimidin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
1-(4-{4-[(1,3-benzothiazol-2-ylmethyl)amino]piperidin-1-yl}benzoyl)piperidin-3-ol
5-{2,7-diazaspiro[4.5]decane-7-carbonyl}-2-(methylsulfanyl)-3,4-dihydropyrimidin-4-one
5-chloro-2-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
3-[(2-fluorophenyl)methyl]-1-{furo[3,2-c]pyridin-4-yl}piperidine-3-carboxylic acid
2-[(2-hydroxyethyl)(methyl)amino]-2-(4-{[(propan-2-yl)carbamoyl]amino}phenyl)acetic acid
2-(2-methyl-1,3-thiazol-4-yl)-1-(6-methyl-2-phenyl-1,2-diazinan-1-yl)ethan-1-one
methyl 2-(diethylsulfamoyl)-6-[(4-methoxy-2,3-dimethylphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-(thiophene-2-carbonyl)piperazine
1-(cyclopropylmethyl)-4-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2-(propan-2-yl)-1,4-diazepane
2-[(4-cyclopentyl-1,4-diazepan-1-yl)methyl]-1-methyl-1H-indole
4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1H-1,2,4-triazole-5-carbonyl)piperidine
2-(4-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)pyrimidine
N,N-dimethyl-2-{[(2-methyl-6-propylpyrimidin-4-yl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
2-(dimethylamino)-2-(2-fluorophenyl)-N-methyl-N-(quinolin-3-ylmethyl)acetamide
N-methyl-N-(pyrazin-2-ylmethyl)-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
3-(oxolan-3-yl)-5-(2-phenylethyl)-1,2,4-oxadiazole
ethyl 5-(2-phenoxyacetyl)-1-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-({[2-(2,4-dimethylphenoxy)ethyl](methyl)amino}methyl)benzoic acid
N-(2-methoxyethyl)-3-(3-methyl-1H-pyrazol-1-yl)-N-{[6-methyl-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}propanamide
2-{5-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
7,7-dimethyl-2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-{[(2-fluorophenyl)methyl]amino}-N-[3-(methylsulfanyl)phenyl]-5-(pyrrolidine-1-sulfonyl)benzamide
1-(4-chloro-2-fluorobenzoyl)-4-[(dimethylamino)methyl]azepan-4-ol
7-fluoro-N-[2-(4-hydroxyphenyl)ethyl]-3-methyl-1-benzofuran-2-carboxamide
(1S,5R)-3-[(5-methoxy-1,3,4-thiadiazol-2-yl)methyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
1-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-2-(1-propylpiperidin-4-yl)ethan-1-one
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-butoxyethan-1-one
3-benzyl-4-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
1-[3-(1H-imidazol-1-yl)propyl]-1-(pyridin-3-ylmethyl)-3-(2,4,6-trimethylpyridin-3-yl)urea
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}(3-phenylpropyl)amine