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1-{4-[(2-methylprop-2-en-1-yl)oxy]phenyl}-3-[2-(1-methylpyrrolidin-2-yl)ethyl]urea
8-(1-hydroxypropan-2-yl)-3-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-[(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)methyl]-1,2,4-oxadiazole-3-carboxamide
3-(1H-1,3-benzodiazol-1-yl)-1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]propan-1-one
1-{3-[4-(3,5-dimethylphenyl)-3-oxopiperazin-1-yl]-3-oxopropyl}azepan-2-one
N-(piperidin-4-ylmethyl)-4-(propan-2-yl)pyrimidin-2-amine
6-methyl-2-{2-[4-(2-phenylpropyl)-1H-1,2,3-triazol-1-yl]ethyl}-3,4-dihydropyrimidin-4-one
1-(furan-2-carbonyl)-4-[4-(pyrrolidin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]piperidine
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)cyclopropanecarboxamide
(1R,5S,8S)-3-[3-(dimethylamino)benzoyl]-N,N-dimethyl-3-azabicyclo[3.2.1]octan-8-amine
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(pyridin-4-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]({[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
3-[1-(2,3-difluoro-4-methylbenzoyl)piperidin-3-yl]benzoic acid
2-(dimethyl-1,3-thiazol-5-yl)-N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
2-(2-fluorophenyl)-1-[4-hydroxy-4-(hydroxymethyl)azepan-1-yl]ethan-1-one
1-methyl-4-(4-{[(4-methylphenyl)amino]methyl}benzoyl)piperazin-2-one
1-[7-(1-hydroxy-2,2-diphenylethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(1,3-thiazol-4-yl)ethan-1-one
1-[(4-{2-hydroxy-3-[methyl(propan-2-yl)amino]propoxy}-3-methoxyphenyl)methyl]-1,4-diazepan-5-one
[3-(cyclopropylmethyl)-1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-3-yl]methanol
2-({1-[2-(2-ethylphenoxy)ethyl]piperidin-4-yl}oxy)pyrimidine
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}piperazine
2-{1-[3-(1H-imidazol-1-yl)propyl]-1H-imidazol-2-yl}-4-phenyl-1,3-thiazole
2-[methyl(pyridin-2-ylmethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1,3-benzothiazole-5-carboxamide
N-{[3-(pyrrolidin-1-yl)phenyl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N'-cyclooctyl-N-[(3S,4R)-4-ethoxyoxolan-3-yl]butanediamide
4-{[2-(5-methylfuran-2-yl)-1H-imidazol-1-yl]methyl}-2-(pyrrolidin-1-yl)-1,3-thiazole
1-(azepan-1-yl)-3-(3-{[4-(2-methoxyethoxy)piperidin-1-yl]methyl}phenoxy)propan-2-ol
3-{3-[benzyl(methyl)amino]piperidine-1-carbonyl}-2H-chromen-2-one
5-fluoro-N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-1H-indole-2-carboxamide
(2S,4R)-4-[3-(dimethylamino)benzamido]-N-ethyl-1-(3-hydroxypropanoyl)pyrrolidine-2-carboxamide
2-ethoxy-4-{[3-(2-hydroxyethyl)-4-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-1-yl]methyl}phenol
1-{[4-(1H-imidazol-1-yl)phenyl]methyl}-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
3-(pentan-2-yl)-8-(1H-1,2,4-triazole-5-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(5-methylpyrazin-2-yl)methyl]-1-(oxan-4-yl)piperidine-3-carboxamide
N-[2-(1-methylpyrrolidin-2-yl)ethyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
6-{[(3R,4S)-1-[2-(morpholin-4-yl)-2-oxoethyl]-4-(propan-2-yl)pyrrolidin-3-yl]amino}pyridine-2-carbonitrile
N-(1-{2-oxo-2-[2-(pyridin-2-yl)piperidin-1-yl]ethyl}-1H-pyrazol-4-yl)-2-(phenylsulfanyl)acetamide
2-{[4-(cyclohex-3-ene-1-carbonyl)-2-oxo-1-(2-phenylethyl)-1,4-diazepan-6-yl]oxy}-N,N-diethylacetamide
1-(2-hydroxy-3-{3-[(3,3,4-trimethylpiperazin-1-yl)methyl]phenoxy}propyl)piperidin-4-ol
4-{1-benzyl-5-[(5-methylfuran-2-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperazin-2-one
8-(3-hydroxypyrrolidine-1-carbonyl)-2-methyl-1,4-dihydroquinolin-4-one
N-({5-[(oxolan-2-ylmethyl)sulfanyl]-4-[3-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl}methyl)-3-phenyl-1,2-oxazole-5-carboxamide
(benzylsulfamoyl)(ethyl)[2-(1H-pyrazol-1-yl)ethyl]amine
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)-3-methoxyphenyl]methyl}-2-(4-fluorophenyl)-N-(oxolan-2-ylmethyl)acetamide
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperazine
7-methyl-2-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
N-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(4S)-3,3,4-trimethyl-1-[4-(4-methylpiperazine-1-carbonyl)pyridin-2-yl]piperidin-4-ol
methyl 5-[(3,3-dimethylcyclohexyl)amino]-1-(2-methoxyethyl)-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate